Renin inhibitors. Design and synthesis of a new class of conformationally restricted analogs of angiotensinogen

Design And Synthesis ◽

New Class ◽

1,2,3-Trisubstituted cyclopropanes as conformationally restricted peptide isosteres: application to the design and synthesis of novel renin inhibitors

Journal of Medicinal Chemistry ◽

10.1021/jm00088a005 ◽

1992 ◽

Vol 35 (10) ◽

pp. 1710-1721 ◽

Cited By ~ 60

Author(s):

Stephen F. Martin ◽

Richard E. Austin ◽

Christopher J. Oalmann ◽

William R. Baker ◽

Stephen L. Condon ◽

...

Keyword(s):

Renin Inhibitors ◽

Design And Synthesis ◽

Peptide Isosteres

69 Conformationally restricted analogs of a new class of potent non-nucleoside reverse transcriptase inhibitors

Antiviral Research ◽

10.1016/0166-3542(93)90447-q ◽

1993 ◽

Vol 20 ◽

pp. 77

Keyword(s):

Reverse Transcriptase ◽

Reverse Transcriptase Inhibitors ◽

Nucleoside Reverse Transcriptase Inhibitors ◽

New Class ◽

Design and synthesis of conformationally restricted renin inhibitors

Peptides ◽

10.1007/978-94-011-2264-1_330 ◽

1992 ◽

pp. 816-817 ◽

Cited By ~ 1

Author(s):

C. E. Brotherton-Pleiss ◽

S. R. Newman ◽

L. D. Waterbury ◽

M. S. Schwartzberg

Keyword(s):

Renin Inhibitors ◽

Design And Synthesis

In silico design and synthesis of N‐arylalkanyl 2‐naphthamides as a new class of non‐purine xanthine oxidase inhibitors

Drug Development Research ◽

10.1002/ddr.21782 ◽

2021 ◽

Author(s):

Sheau Ling Ho ◽

Ching‐Ting Lin ◽

Shoei‐Sheng Lee

Keyword(s):

Xanthine Oxidase ◽

In Silico ◽

In Silico Design ◽

Design And Synthesis ◽

New Class ◽

Xanthine Oxidase Inhibitors

ChemInform Abstract: 2-Phenylpyrroles as Conformationally Restricted Benzamide Analogues. A New Class of Potential Antipsychotics. Part 1.

ChemInform ◽

10.1002/chin.198815241 ◽

1988 ◽

Vol 19 (15) ◽

Author(s):

I. VAN WIJNGAARDEN ◽

C. G. KRUSE ◽

R. VAN HES ◽

J. A. M. VAN DER HEYDEN ◽

M. TH. M. TULP

Keyword(s):

New Class

A 3 dimensional model for 5-HT1A-receptor agonists based on stereoselective methyl-substituted and conformationally restricted analogs of 8-hydroxy-2-(dipropylamino)tetralin

Journal of Medicinal Chemistry ◽

10.1021/jm00106a004 ◽

1991 ◽

Vol 34 (2) ◽

pp. 497-510 ◽

Cited By ~ 47

Author(s):

Charlotta Mellin ◽

Jerk Vallgaarda ◽

David L. Nelson ◽

Lena Bjoerk ◽

Hong Yu ◽

...

Keyword(s):

Dimensional Model ◽

3 Dimensional ◽

Receptor Agonists ◽

Nucleoglycoconjugates: Design and Synthesis of a New Class of DNA–Carbohydrate Conjugates

Angewandte Chemie ◽

10.1002/1521-3757(20001016)112:20<3806::aid-ange3806>3.0.co;2-y ◽

2000 ◽

Vol 112 (20) ◽

pp. 3806-3809 ◽

Cited By ~ 2

Author(s):

Terry L. Sheppard ◽

Chi-Huey Wong ◽

Gerald F. Joyce

Keyword(s):

Design And Synthesis ◽

New Class

Synthesis of conformationally restricted analogs of kainic acid. Is the conformation of the C4-substituent of kainoid important to its neuroexcitatory activity?

Tetrahedron Letters ◽

10.1016/0040-4039(95)01094-x ◽

1995 ◽

Vol 36 (35) ◽

pp. 6235-6238 ◽

Cited By ~ 22

Author(s):

Kimiko Hashimoto ◽

Yasufumi Ohfune ◽

Haruhisa Shirahama

Keyword(s):

Kainic Acid ◽

ChemInform Abstract: Conformationally Restricted Novel Pyrazole Derivatives: Synthesis of 1,8-Disubstituted 5,5-Dimethyl-4,5-dihydro-1H-benzo[g]indazoles as a New Class of PDE4 Inhibitors.

ChemInform ◽

10.1002/chin.201239133 ◽

2012 ◽

Vol 43 (39) ◽

pp. no-no

Author(s):

S. Venkataiah ◽

et al. et al.

Keyword(s):

Pyrazole Derivatives ◽

New Class

Computer-Aided Design and Synthesis of a New Class of PEX14 Inhibitors: Substituted 2,3,4,5-Tetrahydrobenzo[F][1,4]oxazepines as Potential New Trypanocidal Agents

Journal of Chemical Information and Modeling ◽

10.1021/acs.jcim.1c00472 ◽

2021 ◽

Author(s):

Roberto Fino ◽

Dominik Lenhart ◽

Vishal C. Kalel ◽

Charlotte A. Softley ◽

Valeria Napolitano ◽

...

Keyword(s):

Computer Aided Design ◽

Design And Synthesis ◽

New Class ◽

Computer Aided ◽

Aided Design