conformationally restricted analogs Recently Published Documents

Aba Receptor ◽

Conformationally restricted analogs of (+)-PAO4, an abscisic acid receptor antagonist, were synthesized to improve its potency.

Synthesis of novel non-natural spiro[2.3]hexane amino acids, the conformationally restricted analogs of γ-aminobutyric acid

Russian Chemical Bulletin ◽

10.1007/s11172-017-1912-7 ◽

2017 ◽

Vol 66 (8) ◽

pp. 1483-1490 ◽

Cited By ~ 1

Author(s):

N. V. Yashin ◽

E. B. Averina ◽

D. A. Vasilenko ◽

Yu. K. Grishin ◽

D. I. Osolodkin ◽

...

Keyword(s):

Amino Acids ◽

Aminobutyric Acid ◽

Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted Analogs

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.7b00247 ◽

2017 ◽

Vol 60 (10) ◽

pp. 4304-4315 ◽

Cited By ~ 6

Author(s):

Alessio Lodola ◽

Serena Bertolini ◽

Matteo Biagetti ◽

Silvia Capacchi ◽

Fabrizio Facchinetti ◽

...

Keyword(s):

Conformational Equilibria ◽

A structure–function study of PACAP using conformationally restricted analogs: Identification of PAC1 receptor-selective PACAP agonists

Peptides ◽

10.1016/j.peptides.2015.01.009 ◽

2015 ◽

Vol 66 ◽

pp. 26-42 ◽

Cited By ~ 18

Author(s):

Irene Ramos-Álvarez ◽

Samuel A. Mantey ◽

Taichi Nakamura ◽

Bernardo Nuche-Berenguer ◽

Paola Moreno ◽

...

Keyword(s):

Structure Function ◽

Pac1 Receptor ◽

Function Study ◽

Synthesis of conformationally restricted Analogs of γ-aminobutyric acid

Review Journal of Chemistry ◽

10.1134/s2079978014040049 ◽

2014 ◽

Vol 4 (4) ◽

pp. 253-275 ◽

Cited By ~ 3

Author(s):

N. V. Yashin ◽

T. N. Chmovzh ◽

E. B. Averina ◽

T. S. Kuznetsova ◽

N. S. Zefirov

Keyword(s):

Aminobutyric Acid ◽

Conformationally restricted analogs of the direct thrombin inhibitor FM 19

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2011.10.045 ◽

2011 ◽

Vol 19 (24) ◽

pp. 7425-7434 ◽

Cited By ~ 5

Author(s):

Elizabeth A. Girnys ◽

Vanessa R. Porter ◽

Henry I. Mosberg

Keyword(s):

Direct Thrombin Inhibitor ◽

Thrombin Inhibitor ◽

Assessment of dopamine D1 receptor affinity and efficacy of three tetracyclic conformationally-restricted analogs of SKF38393

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2011.07.057 ◽

2011 ◽

Vol 19 (18) ◽

pp. 5420-5431 ◽

Cited By ~ 6

Author(s):

Alia H. Clark ◽

John D. McCorvy ◽

Val J. Watts ◽

David E. Nichols

Keyword(s):

Dopamine D1 Receptor ◽

D1 Receptor ◽

Receptor Affinity ◽

ChemInform Abstract: Synthesis of Some Conformationally Restricted Analogs of Serotonin.

ChemInform ◽

10.1002/chin.199109187 ◽

2010 ◽

Vol 22 (9) ◽

pp. no-no

Author(s):

J. E. MACOR ◽

K. RYAN

Keyword(s):

ChemInform Abstract: Novel Conformationally Restricted Analogs of Norepinephrine: Synthesis and Structure Activity

ChemInform ◽

10.1002/chin.199151340 ◽

2010 ◽

Vol 22 (51) ◽

pp. no-no

Author(s):

F. Z. BASHA

Keyword(s):

Structure Activity ◽

ChemInform Abstract: Stereocontrolled Syntheses of Some Conformationally Restricted Analogs of Serotonin.

ChemInform ◽

10.1002/chin.199208289 ◽

2010 ◽

Vol 23 (8) ◽

pp. no-no

Author(s):

A. GHOSH ◽

W. WANG ◽

J. P. FREEMAN ◽

J. S. ALTHAUS ◽

P. F. VON VOIGTLANDER ◽

...

Keyword(s):