Estrogen Receptor-β Potency-Selective Ligands:  Structure−Activity Relationship Studies of Diarylpropionitriles and Their Acetylene and Polar Analogues

Estrogen Receptor Β ◽

Activity Relationship ◽

Structure Activity ◽

Selective Ligands

Structure-based quantitative structure–activity relationship modeling of estrogen receptor β-ligands

Future Medicinal Chemistry ◽

10.4155/fmc.11.49 ◽

2011 ◽

Vol 3 (8) ◽

pp. 933-945 ◽

Cited By ~ 6

Author(s):

Xialan Dong ◽

Solomon G Hilliard ◽

Weifan Zheng

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Β ◽

Activity Relationship ◽

Quantitative Structure ◽

Quantitative structure-activity relationship of compounds binding to estrogen receptor β based on heuristic method

Science China Chemistry ◽

10.1007/s11426-010-4077-x ◽

2010 ◽

Vol 54 (1) ◽

pp. 237-243 ◽

Cited By ~ 4

Author(s):

YiMing Zhang ◽

XuShu Yang ◽

Cheng Sun ◽

LianSheng Wang

Keyword(s):

Estrogen Receptor ◽

Heuristic Method ◽

Estrogen Receptor Β ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Structure–Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.1c00555 ◽

2021 ◽

Author(s):

David Sedlák ◽

Tyler A. Wilson ◽

Werner Tjarks ◽

Hanna S. Radomska ◽

Hongyan Wang ◽

...

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Β ◽

Activity Relationship ◽

Structure Activity ◽

Synthesis and structure–activity relationship of 3-arylbenzoxazines as selective estrogen receptor β agonists

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.01.099 ◽

2004 ◽

Vol 14 (9) ◽

pp. 2327-2330 ◽

Cited By ~ 28

Author(s):

Wu Yang ◽

Yufeng Wang ◽

Zhengping Ma ◽

Rajasree Golla ◽

Terry Stouch ◽

...

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Β ◽

Activity Relationship ◽

Structure Activity ◽

Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 5: Combined A- and C-ring structure–activity relationship studies

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.08.009 ◽

2007 ◽

Vol 17 (20) ◽

pp. 5563-5566 ◽

Cited By ~ 27

Author(s):

Timothy I. Richardson ◽

Jeffrey A. Dodge ◽

Yong Wang ◽

Jim D. Durbin ◽

Venkatesh Krishnan ◽

...

Keyword(s):

Estrogen Receptor ◽

Ring Structure ◽

Estrogen Receptor Β ◽

Activity Relationship ◽

Synthesis and Structure—Activity Relationship of 3-Arylbenzoxazines as Selective Estrogen Receptor β Agonists.

ChemInform ◽

10.1002/chin.200435151 ◽

2004 ◽

Vol 35 (35) ◽

Author(s):

Wu Yang ◽

et al. et al.

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Β ◽

Activity Relationship ◽

Structure Activity ◽

Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 2: Structure–activity relationship studies on the benzopyran scaffold

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.04.051 ◽

2007 ◽

Vol 17 (13) ◽

pp. 3570-3574 ◽

Cited By ~ 25

Author(s):

Timothy I. Richardson ◽

Bryan H. Norman ◽

Charles W. Lugar ◽

Scott A. Jones ◽

Yong Wang ◽

...

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Β ◽

Activity Relationship ◽

ChemInform Abstract: Binary Quantitative Structure-Activity Relationship (QSAR) Analysis of Estrogen Receptor Ligands.

ChemInform ◽

10.1002/chin.199921263 ◽

2010 ◽

Vol 30 (21) ◽

pp. no-no

Author(s):

Hua Gao ◽

Chris Williams ◽

Paul Labute ◽

Juergen Bajorath

Keyword(s):

Estrogen Receptor ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Ligands ◽

Qsar Analysis ◽

Structure Activity ◽

Estrogen Receptor Ligands

Potent and Selective Ligands for the Dopamine Transporter (DAT): Structure−Activity Relationship Studies of Novel 4-[2-(Diphenylmethoxy)ethyl]-1-(3-phenylpropyl)piperidine Analogues

Journal of Medicinal Chemistry ◽

10.1021/jm970595h ◽

1998 ◽

Vol 41 (5) ◽

pp. 699-705 ◽

Cited By ~ 20

Author(s):

Aloke K. Dutta ◽

Lori L. Coffey ◽

Maarten E. A. Reith

Keyword(s):

Dopamine Transporter ◽

Activity Relationship ◽

Structure Activity ◽

Selective Ligands

ChemInform Abstract: Evaluation of Quantitative Structure-Activity Relationship Methods for Large-Scale Prediction of Chemicals Binding to the Estrogen Receptor.

ChemInform ◽

10.1002/chin.199845276 ◽

2010 ◽

Vol 29 (45) ◽

pp. no-no ◽

Cited By ~ 1

Author(s):

W. TONG ◽

D. R. LOWIS ◽

R. PERKINS ◽

Y. CHEN ◽

W. J. WELSH ◽

...

Keyword(s):

Estrogen Receptor ◽

Large Scale ◽

Activity Relationship ◽

Quantitative Structure ◽