Synthesis and Biological Evaluation of 2-Alkynyl-N6-methyl-5′-N-methylcarboxamidoadenosine Derivatives as Potent and Highly Selective Agonists for the Human Adenosine A3Receptor‡

2009 ◽  
Vol 52 (23) ◽  
pp. 7897-7900 ◽  
Author(s):  
Rosaria Volpini ◽  
Michela Buccioni ◽  
Diego Dal Ben ◽  
Catia Lambertucci ◽  
Carmen Lammi ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Selective Agonists ◽  
Synthesis And Biological Evaluation

ChemInform Abstract: Substituted Hexahydrobenzo(f)thieno(c)quinolines as Dopamine D1- Selective Agonists: Synthesis and Biological Evaluation in vitro and in vivo.

ChemInform ◽  
2010 ◽  
Vol 28 (39) ◽  
pp. no-no
Author(s):  
M. R. MICHAELIDES ◽  
Y. HONG ◽  
S. JUN. DIDOMENICO ◽  
E. K. BAYBURT ◽  
K. E. ASIN ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Selective Agonists ◽  
Synthesis And Biological Evaluation

Design, synthesis, and biological evaluation of a new class of MT2-selective agonists

RSC Advances ◽  
2014 ◽  
Vol 4 (49) ◽  
pp. 25871-25874 ◽  
Author(s):  
Xuan Zhang ◽  
Zhilong Wang ◽  
Qingqing Huang ◽  
Yu Luo ◽  
Xin Xie ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
New Class ◽  
Selective Agonists ◽  
Synthesis And Biological Evaluation

In this study, we have designed and synthesized a novel class of chiral 2,3-dihydro-1H-indene derivatives as highly selective MT2 agonists.

Design, synthesis and biological evaluation of novel TRβ selective agonists sustained by ADME-toxicity analysis

2020 ◽  
Vol 188 ◽  
pp. 112006 ◽  
Author(s):  
Massimiliano Runfola ◽  
Simona Sestito ◽  
Lorenza Bellusci ◽  
Valeria La Pietra ◽  
Vincenzo Maria D’Amore ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Toxicity Analysis ◽  
Selective Agonists ◽  
Synthesis And Biological Evaluation

Synthesis and biological evaluation of halogenated curcumin analogs as potential nuclear receptor selective agonists

2013 ◽  
Vol 21 (3) ◽  
pp. 693-702 ◽  
Author(s):  
Shane Batie ◽  
Jamie H. Lee ◽  
Rabia A. Jama ◽  
Drew O. Browder ◽  
Luis A. Montano ◽  
...  
Keyword(s):  
Nuclear Receptor ◽  
Biological Evaluation ◽  
Curcumin Analogs ◽  
Selective Agonists ◽  
Synthesis And Biological Evaluation
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