Facile and Efficient Synthesis of Dendrimers and One-Pot Preparation of Dendritic–Linear Polymer Conjugates via a Single Chemistry: Utilization of Kinetically Selective Thiol–Michael Addition Reactions

2014 ◽  
Vol 47 (15) ◽  
pp. 4894-4900 ◽  
Author(s):  
Shunsuke Chatani ◽  
Maciej Podgórski ◽  
Chen Wang ◽  
Christopher N. Bowman
Keyword(s):  
Michael Addition ◽  
Linear Polymer ◽  
Addition Reactions ◽  
Efficient Synthesis ◽  
One Pot ◽  
Polymer Conjugates

The first peripherally masked thiol dendrimers: a facile and highly efficient functionalization strategy of polyester dendrimers via one-pot xanthate deprotection/thiol–acrylate Michael addition reactions

2014 ◽  
Vol 50 (50) ◽  
pp. 6574-6577 ◽  
Author(s):  
Sam E. R. Auty ◽  
Oliver Andrén ◽  
Michael Malkoch ◽  
Steven P. Rannard
Keyword(s):  
Michael Addition ◽  
Addition Reactions ◽  
One Pot ◽  
Highly Efficient

We present the first xanthate surface functional dendrimers which undergo rapid one-pot deprotection to thiols and subsequent acrylate Michael addition .

Efficient Synthesis of 3-Amino-1,5-benzodiazepine-2-one Derivatives

Synlett ◽  
2017 ◽  
Vol 28 (10) ◽  
pp. 1183-1186 ◽  
Author(s):  
Nobuhiro Obara ◽  
Takeshi Watanabe ◽  
Tomohiro Asakawa ◽  
Toshiyuki Kan ◽  
Takao Tanaka
Keyword(s):  
Michael Addition ◽  
Convenient Method ◽  
Addition Reaction ◽  
Efficient Synthesis ◽  
Michael Addition Reaction ◽  
One Pot ◽  
Simple Method ◽  
The Michael Addition

A convenient method for synthesizing 3-amino-1,5-benzodiazepine-2-one via the Michael addition reaction of o-phenylenediamine with dehydroalanine ester derivatives, followed by cyclization, was developed. This simple method was used to obtain a variety of N-substituted 3-amino-1,5-benzodiazepine-2-ones in one pot with good yields.

ChemInform Abstract: Buchwald-Hartwig Coupling/Michael Addition Reactions: One-Pot Synthesis of 1,2-Disubstituted 4-Quinolones from Chalcones and Primary Amines.

ChemInform ◽  
2012 ◽  
Vol 43 (40) ◽  
pp. no-no
Author(s):  
Xiang-Dong Fei ◽  
Zhou Zhou ◽  
Wen Li ◽  
Yong-Ming Zhu ◽  
Jing-Kang Shen
Keyword(s):  
Michael Addition ◽  
Primary Amines ◽  
Addition Reactions ◽  
One Pot ◽  
One Pot Synthesis

Efficient Synthesis of11C-Acrylesters,11C-Acrylamides and Their Application in Michael Addition Reactions for PET Tracer Development

2017 ◽  
Vol 2017 (34) ◽  
pp. 5154-5162 ◽  
Author(s):  
Ulrike Filp ◽  
Anna L. Pees ◽  
Carlotta Taddei ◽  
Aleksandra Pekošak ◽  
Antony D. Gee ◽  
...  
Keyword(s):  
Michael Addition ◽  
Addition Reactions ◽  
Efficient Synthesis ◽  
Pet Tracer ◽  
Tracer Development

One-Pot Synthesis of 1,3,5-Tribenzoylbenzenes by Three Consecutive Michael Addition Reactions of 1-Phenyl-2-propyn-1-ones in Pressurized Hot Water in the Absence of Added Catalysts

2010 ◽  
Vol 17 (2) ◽  
pp. 606-612 ◽  
Author(s):  
Makoto Tanaka ◽  
Kazuya Nakamura ◽  
Tatsuya Iwado ◽  
Toshiyuki Sato ◽  
Masaki Okada ◽  
...  
Keyword(s):  
Michael Addition ◽  
Hot Water ◽  
Addition Reactions ◽  
One Pot ◽  
One Pot Synthesis

Solvent free one-pot multi-component synthesis of β-azaarene substituted ketones via a Sn-catalyzed C(sp3)–H functionalization of 2-alkylazaarenes

RSC Advances ◽  
2015 ◽  
Vol 5 (125) ◽  
pp. 103091-103094 ◽  
Author(s):  
Santosh S. Chavan ◽  
Mohsinkhan Y. Pathan ◽  
Shafeek A. R. Mulla
Keyword(s):  
Michael Addition ◽  
Cascade Reaction ◽  
Solvent Free ◽  
Efficient Synthesis ◽  
One Pot

A tin-catalyzed solvent free one-pot multi-component cascade reaction strategy for the efficient synthesis of β-azaarene substituted ketones via an aldol–Michael addition/C(sp3)–H functionalization of 2-alkylazaarenes has been developed.

A stereocontrolled synthesis of Hagen's gland lactones via iterative proline catalyzed α-aminoxylation and oxa-Michael addition reactions

RSC Advances ◽  
2015 ◽  
Vol 5 (75) ◽  
pp. 61000-61005 ◽  
Author(s):  
Shruti Vandana Kauloorkar ◽  
Vishwajeet Jha ◽  
Ganesh Jogdand ◽  
Pradeep Kumar
Keyword(s):  
Michael Addition ◽  
Addition Reactions ◽  
Efficient Synthesis ◽  
Stereocontrolled Synthesis

A simple and efficient synthesis of Hagen's gland lactones was achieved using a sequential α-aminoxylation/oxa-Michael approach in a highly diastereoselective manner with assignment of relative configurations.

Sign in / Sign up

Export Citation Format

Share Document