Organocatalytic asymmetric synthesis of benzothiazolopyrimidines via [4+2] cycloaddition of azlactones with 2-benzothiazolimines
An easily available L-proline-derived guanidine-amide was found efficient to catalyze [4+2] cycloaddition of azlactones with 2-benzothiazolimines, affording various benzothiazolopyrimidines bearing adjacent tertiary and quaternary stereogenic centers in excellent results at...
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