Rh(iii)-Catalyzed C–H allylation/annulative Markovnikov addition with 5-methylene-1,3-dioxan-2-one: formation of isoquinolinones containing a C3 quaternary centre
Rh(iii)-Catalyzed C–H allylation/annulative Markovnikov addition reaction was disclosed, offering isoquinolinones containing a C3 quaternary centre. By using this method as the key step, the US28 inverse agonist analogs were synthesized.
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2007 ◽
Vol 48
(27)
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pp. 4669-4673
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Keyword(s):
2015 ◽
Vol 137
(4)
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pp. 1452-1457
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