Characterization of the thromboxane synthase pathway product 12-oxoheptadeca-5(Z)-8(E)-10(E)-trienoic acid as a thromboxane A2 
 receptor antagonist with minimal intrinsic activity

Protective Effects of G 619, a Dual Thromboxane Synthase Inhibitor and Thromboxane A2 Receptor Antagonist, in Splanchnic Artery Occlusion Shock

Journal of Cardiovascular Pharmacology ◽

10.1097/00005344-199201000-00016 ◽

1992 ◽

Vol 19 (1) ◽

pp. 115-119 ◽

Cited By ~ 12

Author(s):

Francesco Squadrito ◽

Domenica Altavilla ◽

Basilia Zingarelli ◽

Maria P. Ioculano ◽

Giuseppe M. Campo ◽

...

Keyword(s):

Receptor Antagonist ◽

Thromboxane A2 ◽

Artery Occlusion ◽

Protective Effects ◽

Thromboxane Synthase ◽

Thromboxane A2 Receptor ◽

Thromboxane Synthase Inhibitor ◽

Splanchnic Artery ◽

Synthase Inhibitor

Pharmacological Characterization of N-tert-Butyl-N′-[2-(4′-methylphenylamino)-5-nitrobenzenesulfonyl]urea (BM-573), a Novel Thromboxane A2 Receptor Antagonist and Thromboxane Synthase Inhibitor in a Rat Model of Arterial Thrombosis and Its Effects on Bleeding Time

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.103.063610 ◽

2004 ◽

Vol 309 (2) ◽

pp. 498-505 ◽

Cited By ~ 23

Author(s):

Jean-Michel Dogné ◽

Julien Hanson ◽

Xavier de Leval ◽

Philippe Kolh ◽

Vincent Tchana-Sato ◽

...

Keyword(s):

Receptor Antagonist ◽

Rat Model ◽

Arterial Thrombosis ◽

Bleeding Time ◽

Thromboxane A2 ◽

Thromboxane A2 Receptor ◽

Thromboxane Synthase Inhibitor ◽

Synthase Inhibitor

Pharmacological characterization of EK112, a new combined angiotensin II and thromboxane A2 receptor antagonist

General Pharmacology The Vascular System ◽

10.1016/s0306-3623(00)00046-x ◽

2000 ◽

Vol 34 (1) ◽

pp. 25-31 ◽

Cited By ~ 2

Author(s):

Tsong-Long Hwang ◽

Yung-An Yeh ◽

Ji-Wang Chern ◽

Che-Ming Teng

Keyword(s):

Angiotensin Ii ◽

Receptor Antagonist ◽

Thromboxane A2 ◽

Intrinsic activity of the non-prostanoid thromboxane A2 receptor antagonist, daltroban (BM 13,505), in human platelets in vitro and in the rat vasculature in vivo

British Journal of Pharmacology ◽

10.1111/j.1476-5381.1995.tb16341.x ◽

1995 ◽

Vol 115 (1) ◽

pp. 210-216 ◽

Cited By ~ 6

Author(s):

Frédéric Bertolino ◽

Jean-Pierre Valentin ◽

Myriam Maffre ◽

Françoise Grelac ◽

Anne-Marie Bessac ◽

...

Keyword(s):

Receptor Antagonist ◽

Thromboxane A2 ◽

Human Platelets ◽

Intrinsic Activity ◽

Pharmacological characterization of cinnamophilin, a novel dual inhibitor of thromboxane synthase and thromboxane A2 receptor

British Journal of Pharmacology ◽

10.1111/j.1476-5381.1994.tb14824.x ◽

1994 ◽

Vol 111 (3) ◽

pp. 906-912 ◽

Cited By ~ 20

Author(s):

Sheu-Meei Yu ◽

Tian-Shung Wu ◽

Che-Ming Teng

Keyword(s):

Thromboxane A2 ◽

Dual Inhibitor ◽

Thromboxane Synthase ◽

Characterization of the pharmacokinetics and pharmacodynamics of a new oral thromboxane A2-receptor antagonist AA-2414 in normal subjects: Population analysis

Clinical Pharmacology & Therapeutics ◽

10.1038/clpt.1994.54 ◽

1994 ◽

Vol 55 (4) ◽

pp. 441-450 ◽

Cited By ~ 5

Author(s):

Ziad Hussein ◽

Emil Samara ◽

Charles S Locke ◽

Margaret A Orchard ◽

Gary L Ringham ◽

...

Keyword(s):

Receptor Antagonist ◽

Population Analysis ◽

Thromboxane A2 ◽

Normal Subjects ◽

Pharmacokinetics And Pharmacodynamics ◽

Electromechanical Characterization

Electromechanical characterization of cinnamophilin, a natural thromboxane A2 receptor antagonist with anti-arrhythmic activity, in guinea-pig heart

British Journal of Pharmacology ◽

10.1038/sj.bjp.0707541 ◽

2008 ◽

Vol 153 (1) ◽

pp. 110-123 ◽

Cited By ~ 2

Author(s):

G-J Chang ◽

M-J Su ◽

T-S Wu ◽

W-P Chen ◽

C-M Kuo

Keyword(s):

Guinea Pig ◽

Receptor Antagonist ◽

Thromboxane A2 ◽

Guinea Pig Heart ◽

Thromboxane A2 Receptor ◽

Carrier-Mediated Active Transport of a Novel Thromboxane A2 Receptor Antagonist [2-(4-Chlorophenylsulfonylaminomethyl)indan-5-yl]acetate (Z-335) into Rat Liver

Drug Metabolism and Disposition ◽

10.1124/dmd.30.5.498 ◽

2002 ◽

Vol 30 (5) ◽

pp. 498-504 ◽

Cited By ~ 1

Author(s):

Yoshihiro Kawabata ◽

Shigeru Furuta ◽

Yutaka Shinozaki ◽

Tadashi Kurimoto ◽

Ryuichiro Nishigaki

Keyword(s):

Receptor Antagonist ◽

Active Transport ◽

Rat Liver ◽

Thromboxane A2 ◽

In Vitro and in Vivo Pharmacological Characterization of BM-613 [N-n-Pentyl-N′-[2-(4′-methylphenylamino)-5-nitrobenzenesulfonyl]urea], a Novel Dual Thromboxane Synthase Inhibitor and Thromboxane Receptor Antagonist

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.104.079301 ◽

2004 ◽

Vol 313 (1) ◽

pp. 293-301 ◽

Cited By ~ 10

Author(s):

Julien Hanson ◽

Stephanie Rolin ◽

Denis Reynaud ◽

Na Qiao ◽

Leanne P. Kelley ◽

...

Keyword(s):

Receptor Antagonist ◽

Thromboxane Synthase ◽

Thromboxane Receptor ◽

Thromboxane Synthase Inhibitor ◽

Thromboxane Receptor Antagonist ◽

Synthase Inhibitor

Antithrombotic effects of S 18886, a novel orally active thromboxane A2 receptor antagonist

Journal of Thrombosis and Haemostasis ◽

10.1111/j.1538-7933.2004.00639.x ◽

2004 ◽

Vol 2 (3) ◽

pp. 492-498 ◽

Cited By ~ 37

Author(s):

J. I. Osende ◽

D. Shimbo ◽

V. Fuster ◽

M. Dubar ◽

J. J. Badimon

Keyword(s):

Receptor Antagonist ◽

Thromboxane A2 ◽

Thromboxane A2 Receptor ◽

Antithrombotic Effects ◽

Orally Active