Anti- and Syn-Selective Cyanosilylation Reactions Promoted by a Sugar-Based Bifunctional Catalyst: Stereoselective Syntheses of Essential Building Blocks for HIV Protease Inhibitors and Bestatin

Govindaswamy Manickam; Hiroyuki Nogami; Motomu Kanai; Harald Gröger; Masakatsu Shibasaki

doi:10.1055/s-2001-13383

Anti- and Syn-Selective Cyanosilylation Reactions Promoted by a Sugar-Based Bifunctional Catalyst: Stereoselective Syntheses of Essential Building Blocks for HIV Protease Inhibitors and Bestatin

Synlett ◽

10.1055/s-2001-13383 ◽

2001 ◽

Vol 2001 (05) ◽

pp. 0617-0620 ◽

Cited By ~ 13

Author(s):

Govindaswamy Manickam ◽

Hiroyuki Nogami ◽

Motomu Kanai ◽

Harald Gröger ◽

Masakatsu Shibasaki

Keyword(s):

Protease Inhibitors ◽

Building Blocks ◽

Bifunctional Catalyst ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Stereoselective Syntheses

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ChemInform Abstract: anti- and syn-Selective Cyanosilylation Reactions Promoted by a Sugar-Based Bifunctional Catalyst: Stereoselective Syntheses of Essential Building Blocks for HIV Protease Inhibitors and Bestatin.

ChemInform ◽

10.1002/chin.200132085 ◽

2010 ◽

Vol 32 (32) ◽

pp. no-no

Author(s):

Govindaswamy Manickam ◽

Hiroyuki Nogami ◽

Motomu Kanai ◽

Harald Groeger ◽

Masakatsu Shibasaki

Keyword(s):

Protease Inhibitors ◽

Building Blocks ◽

Bifunctional Catalyst ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Stereoselective Syntheses

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ChemInform Abstract: Preparation of Aminoalkyl Chlorohydrin Hydrochlorides: Key Building Blocks for Hydroxyethylamine-Based HIV Protease Inhibitors.

ChemInform ◽

10.1002/chin.199639109 ◽

2010 ◽

Vol 27 (39) ◽

pp. no-no

Author(s):

P. L. BEAULIEU ◽

D. WERNIC

Keyword(s):

Protease Inhibitors ◽

Building Blocks ◽

Hiv Protease ◽

Hiv Protease Inhibitors

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Preparation of Aminoalkyl Chlorohydrin Hydrochlorides: Key Building Blocks for Hydroxyethylamine-Based HIV Protease Inhibitors

The Journal of Organic Chemistry ◽

10.1021/jo960109i ◽

1996 ◽

Vol 61 (11) ◽

pp. 3635-3645 ◽

Cited By ~ 75

Author(s):

Pierre L. Beaulieu ◽

Dominik Wernic

Keyword(s):

Protease Inhibitors ◽

Building Blocks ◽

Hiv Protease ◽

Hiv Protease Inhibitors

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ChemInform Abstract: Synthesis of (2R,5S)- and (2S,5S)-2-Carboxy-1,4-diaza(4.3.0) bicyclononane as Building Blocks for the Synthesis of New Potential HIV Protease Inhibitors.

ChemInform ◽

10.1002/chin.199647162 ◽

2010 ◽

Vol 27 (47) ◽

pp. no-no

Author(s):

M. FALORNI ◽

A. PORCHEDDU ◽

G. GIACOMELLI

Keyword(s):

Protease Inhibitors ◽

Building Blocks ◽

Hiv Protease ◽

Hiv Protease Inhibitors

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A concise synthesis of (2S,3S)-BocAHPBA and (R)-BocDMTA, chiral building blocks for peptide-mimetic HIV protease inhibitors

Tetrahedron Asymmetry ◽

10.1016/s0957-4166(02)00257-4 ◽

2002 ◽

Vol 13 (11) ◽

pp. 1201-1208 ◽

Cited By ~ 13

Author(s):

Masaya Ikunaka ◽

Jun Matsumoto ◽

Yukifumi Nishimoto

Keyword(s):

Protease Inhibitors ◽

Building Blocks ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Peptide Mimetic

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Synthesis of (2R, 5S)- and (2S, 5S)-2-carboxy-1,4-diaza-[4.3.0]bicyclononane as building blocks for the synthesis of new potential HIV protease inhibitors

Tetrahedron Asymmetry ◽

10.1016/0957-4166(96)00241-8 ◽

1996 ◽

Vol 7 (7) ◽

pp. 1999-2005 ◽

Cited By ~ 12

Author(s):

Massimo Falorni ◽

Andrea Porcheddu ◽

Giampaolo Giacomelli

Keyword(s):

Protease Inhibitors ◽

Building Blocks ◽

Hiv Protease ◽

Hiv Protease Inhibitors

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Determining and Overcoming Resistance to HIV Protease Inhibitors

Current Drug Targets - Infectious Disorders ◽

10.2174/1568005043340984 ◽

2004 ◽

Vol 4 (2) ◽

pp. 137-152 ◽

Cited By ~ 17

Author(s):

Jana Prejdova ◽

Milan Soucek ◽

Jan Konvalinka

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors

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A QSAR Study of HIV Protease Inhibitors Using Theoretical Descriptors

Current Computer - Aided Drug Design ◽

10.2174/1573409911006040269 ◽

2010 ◽

Vol 6 (4) ◽

pp. 269-282 ◽

Cited By ~ 4

Author(s):

Subhash C. Basak ◽

Denise Mills ◽

Rajni Garg ◽

Barun Bhhatarai

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Qsar Study

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Simultaneous determination of the HIV protease inhibitors indinavir, amprenavir, saquinavir, ritonavir and nelfinavir in human plasma by high-performance liquid chromatography

Journal of Chromatography B Biomedical Sciences and Applications ◽

10.1016/s0378-4347(00)00617-4 ◽

2001 ◽

Vol 755 (1-2) ◽

pp. 85-89 ◽

Cited By ~ 32

Author(s):

Harumi Yamada ◽

Hajime Kotaki ◽

Tetsuya Nakamura ◽

Aikichi Iwamoto

Keyword(s):

High Performance Liquid Chromatography ◽

Liquid Chromatography ◽

Simultaneous Determination ◽

Human Plasma ◽

Protease Inhibitors ◽

High Performance ◽

Hiv Protease ◽

Hiv Protease Inhibitors

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1351 SYNERGISTIC EFFECTS OF ALCOHOL AND HIV PROTEASE INHIBITORS ON CALCIUM HOMEOSTASIS, STRESS RESPONSE AND INJURY IN MOUSE AND HUMAN HEPATOCYTES

Journal of Hepatology ◽

10.1016/s0168-8278(12)61362-2 ◽

2012 ◽

Vol 56 ◽

pp. S531

Author(s):

C. Ji

Keyword(s):

Stress Response ◽

Protease Inhibitors ◽

Calcium Homeostasis ◽

Synergistic Effects ◽

Human Hepatocytes ◽

Hiv Protease ◽

Hiv Protease Inhibitors

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