Design, synthesis and pharmacological screening of a series of N1-(substituted)aryl-5,7-dimethyl-2-(substituted)pyrido(2,3-d)pyrimidin-4(3H)-ones as potential histamine H1-receptor antagonists

2006 ◽  
Vol 21 (6) ◽  
pp. 681-691 ◽  
Author(s):  
Bhanubhai N. Suhagia ◽  
Mahesh T. Chhabria ◽  
Ashlesha G. Makwana
Keyword(s):  
H1 Receptor ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Histamine H1 Receptor ◽  
Pharmacological Screening

scholarly journals Design of Phthalazinone Amide Histamine H1 Receptor Antagonists for Use in Rhinitis

2017 ◽  
Vol 8 (5) ◽  
pp. 577-581 ◽  
Author(s):  
Panayiotis A. Procopiou ◽  
Alison J. Ford ◽  
Paul M. Gore ◽  
Brian E. Looker ◽  
Simon T. Hodgson ◽  
...  
Keyword(s):  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor

Anti-Inflammatory Actions of Histamine H1 Receptor Antagonists Unrelated to H1 Receptor Blockade

1996 ◽  
Vol 5 (6) ◽  
pp. 449-464 ◽  
Author(s):  
Claus Kroegel ◽  
Verena Herzog ◽  
Birgit Knöchel ◽  
Peter Julius ◽  
Dirk Wagnetz ◽  
...  
Keyword(s):  
Receptor Blockade ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor ◽  
Anti Inflammatory

Identification of selective 8-(piperidin-4-yloxy)quinoline sulfone and sulfonamide histamine H1 receptor antagonists for use in allergic rhinitis

2017 ◽  
Vol 27 (21) ◽  
pp. 4914-4919 ◽  
Author(s):  
Panayiotis A. Procopiou ◽  
Alison J. Ford ◽  
Paul M. Gore ◽  
Ashley P. Hancock ◽  
Simon T. Hodgson ◽  
...  
Keyword(s):  
Allergic Rhinitis ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor
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