In Vitro Pharmacological Characterization of a Novel Allosteric Modulator of α7 Neuronal Acetylcholine Receptor, 4-(5-(4-Chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744), Exhibiting Unique Pharmacological Profile

Neuronal Acetylcholine Receptor

In Vitro Pharmacological Characterization of a Novel Selective α7 Neuronal Nicotinic Acetylcholine Receptor Agonist ABT-107

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.110.167072 ◽

2010 ◽

Vol 334 (3) ◽

pp. 863-874 ◽

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Author(s):

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David J. Anderson ◽

Jens H. Grønlien ◽

Jianguo Ji ◽

William H. Bunnelle ◽

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Keyword(s):

Acetylcholine Receptor ◽

Receptor Agonist ◽

Neuronal Nicotinic Acetylcholine Receptor ◽

In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator

European Journal of Pharmacology ◽

10.1016/j.ejphar.2016.08.032 ◽

2016 ◽

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Carla Lobina ◽

Daniela Giunta ◽

Maurizio Solinas ◽

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Keyword(s):

Allosteric Modulator ◽

Pharmacological Characterization

P2-065: IN VITRO PHARMACOLOGICAL CHARACTERIZATION OF S68890, AN ALLOSTERIC MODULATOR OF ALPHA7 NICOTINIC RECEPTORS

Alzheimer s & Dementia ◽

10.1016/j.jalz.2019.06.2472 ◽

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Kumiko Kambara ◽

Sonia Bertrand ◽

Daniel Bertrand ◽

Alain Benoist ◽

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Keyword(s):

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Allosteric Modulator ◽

Pharmacological Characterization

Pharmacological Characterization of the Allosteric Modulator Desformylflustrabromine and Its Interaction with α4β2 Neuronal Nicotinic Acetylcholine Receptor Orthosteric Ligands

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.110.167684 ◽

2010 ◽

Vol 334 (3) ◽

pp. 917-926 ◽

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Author(s):

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Keyword(s):

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Neuronal Nicotinic Acetylcholine Receptor ◽

Allosteric Modulator ◽

Nicotinic Acetylcholine ◽

Orthosteric Ligands

The GABAB receptor positive allosteric modulator COR659: In vitro metabolism, in vivo pharmacokinetics in rats, synthesis and pharmacological characterization of metabolically protected derivatives

European Journal of Pharmaceutical Sciences ◽

10.1016/j.ejps.2020.105544 ◽

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Paola Maccioni ◽

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Antonella Brizzi ◽

Federica Fara ◽

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Keyword(s):

Gabab Receptor ◽

In Vitro Metabolism ◽

Allosteric Modulator ◽

Pharmacokinetics In Rats ◽

In Vivo Pharmacokinetics

In vitro pharmacological characterization of (±)-4-[2-(1-methyl-2-pyrrolidinyl)ethyl]thio]phenol hydrochloride (SIB-1553A), a nicotinic acetylcholine receptor ligand

Brain Research ◽

10.1016/s0006-8993(03)02979-2 ◽

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Author(s):

Tadimeti S. Rao ◽

Pamala B. Adams ◽

Lucia D. Correa ◽

Emily M. Santori ◽

Aida I. Sacaan ◽

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Keyword(s):

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Receptor Ligand ◽

In vitro pharmacological characterization of ABT-779, a novel positive allosteric modulator of α7 nAChRs

Biochemical Pharmacology ◽

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Α7 Nachrs

Identification and in vitro pharmacological characterization of a novel and selective α7 nicotinic acetylcholine receptor agonist, Br-IQ17B

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Receptor Agonist ◽

Α7 Nicotinic Acetylcholine Receptor ◽

Pharmacological Characterization of the Novel and Selective α7 Nicotinic Acetylcholine Receptor–Positive Allosteric Modulator BNC375

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Joshua D. Vardigan ◽

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Keyword(s):

Acetylcholine Receptor ◽

Allosteric Modulator ◽

The Novel ◽

Α7 Nicotinic Acetylcholine Receptor ◽

Characterization of the pharmacological profile of the potent LTB4 antagonist CP-105,696 on murine LTB4 receptors in vitro.

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Keyword(s):

Pharmacological Profile