Synthesis and Pharmacological Characterization of a Novel Sigma Receptor Ligand with Improved Metabolic Stability and Antagonistic Effects Against Methamphetamine

Receptor Ligand ◽

Antagonistic Effects

Pharmacological Characterization of an Optimized Sigma Receptor Ligand

10.33915/etd.3561 ◽

2012 ◽

Author(s):

Michael Seminerio

Keyword(s):

Sigma Receptor ◽

Abstract 2559: Pharmacological characterization of sigma-2 receptor ligand-induced metabolic stimulation in human SK-N-SH neuroblastoma cells

10.1158/1538-7445.am2020-2559 ◽

2020 ◽

Author(s):

Bridget M. McVeigh ◽

Alissa K. Oakes ◽

Cheri Z. Liu ◽

Christophe Mesangeau ◽

Walid F. Alsharif ◽

...

Keyword(s):

Neuroblastoma Cells ◽

Receptor Ligand ◽

Metabolic Stimulation

Synthesis and Pharmacological Characterization of Sila-panamesine, a Sila-Analogue of the σ Receptor Ligand Panamesine (EMD 57445)

Organometallics ◽

10.1021/om060562c ◽

2006 ◽

Vol 25 (22) ◽

pp. 5396-5408 ◽

Cited By ~ 26

Author(s):

Rainer Ilg ◽

Christian Burschka ◽

Dirk Schepmann ◽

Bernhard Wünsch ◽

Reinhold Tacke

Keyword(s):

Neurochemical characterization of dopaminergic effects of opipramol, a potent sigma receptor ligand, in vivo

Neuropharmacology ◽

10.1016/0028-3908(90)90044-r ◽

1990 ◽

Vol 29 (12) ◽

pp. 1191-1197 ◽

Cited By ~ 13

Author(s):

T RAO ◽

J CLER ◽

S MICK ◽

V DILWORTH ◽

P CONTRERAS ◽

...

Keyword(s):

Sigma Receptor ◽

Design, Synthesis, and Pharmacological Characterization of 4-[4,4-Dimethyl-3-(4-hydroxybutyl)-5-oxo-2-thioxo-1-imidazolidinyl]- 2-iodobenzonitrile as a High-Affinity Nonsteroidal Androgen Receptor Ligand#

Journal of Medicinal Chemistry ◽

10.1021/jm000163y ◽

2000 ◽

Vol 43 (17) ◽

pp. 3344-3347 ◽

Cited By ~ 29

Author(s):

Marcian E. Van Dort ◽

Diane M. Robins ◽

Bess Wayburn

Keyword(s):

Androgen Receptor ◽

Receptor Ligand ◽

Design Synthesis ◽

High Affinity

In vitro and in vivo pharmacological characterization of the nociceptin/orphanin FQ receptor ligand Ac-RYYRIK-ol

European Journal of Pharmacology ◽

10.1016/j.ejphar.2006.03.075 ◽

2006 ◽

Vol 539 (1-2) ◽

pp. 39-48 ◽

Cited By ~ 23

Author(s):

Özge Gündüz ◽

Anna Rizzi ◽

Anna Baldisserotto ◽

Remo Guerrini ◽

Barbara Spagnolo ◽

...

Keyword(s):

Orphanin Fq ◽

ChemInform Abstract: Design, Synthesis, and Pharmacological Characterization of 4-[4,4-Dimethyl-3-(4-hydroxybutyl)-5-oxo-2-thioxo-1-imidazolidinyl] -2-iodobenzonitrile as a High-Affinity Nonsteroidal Androgen Receptor Ligand.

ChemInform ◽

10.1002/chin.200050122 ◽

2000 ◽

Vol 31 (50) ◽

pp. no-no

Author(s):

Marcian E. Van Dort ◽

Diane M. Robins ◽

Bess Wayburn

Keyword(s):

Androgen Receptor ◽

Receptor Ligand ◽

Design Synthesis ◽

High Affinity

Synthesis and Characterization of a Novel γ-Aminobutyric Acid Type A (GABAA) Receptor Ligand That Combines Outstanding Metabolic Stability, Pharmacokinetics, and Anxiolytic Efficacy

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.6b01332 ◽

2016 ◽

Vol 59 (23) ◽

pp. 10800-10806 ◽

Cited By ~ 16

Author(s):

Michael M. Poe ◽

Kashi Reddy Methuku ◽

Guanguan Li ◽

Ashwini R. Verma ◽

Kelly A. Teske ◽

...

Keyword(s):

Gabaa Receptor ◽

Type A ◽

Metabolic Stability ◽

Aminobutyric Acid ◽

Synthesis And Characterization ◽

Receptor Ligand ◽

Acid Type

Pharmacological characterization of the novel nociceptin/orphanin FQ receptor ligand, ZP120: in vitro and in vivo studies in mice

British Journal of Pharmacology ◽

10.1038/sj.bjp.0704894 ◽

2002 ◽

Vol 137 (3) ◽

pp. 369-374 ◽

Cited By ~ 40

Author(s):

Anna Rizzi ◽

Daniela Rizzi ◽

Giuliano Marzola ◽

Domenico Regoli ◽

Bjarne Due Larsen ◽

...

Keyword(s):

In Vivo Studies ◽

The Novel ◽

Orphanin Fq ◽

In vitro pharmacological characterization of (±)-4-[2-(1-methyl-2-pyrrolidinyl)ethyl]thio]phenol hydrochloride (SIB-1553A), a nicotinic acetylcholine receptor ligand

Brain Research ◽

10.1016/s0006-8993(03)02979-2 ◽

2003 ◽

Vol 981 (1-2) ◽

pp. 85-98 ◽

Cited By ~ 15

Author(s):

Tadimeti S. Rao ◽

Pamala B. Adams ◽

Lucia D. Correa ◽

Emily M. Santori ◽

Aida I. Sacaan ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Nicotinic Acetylcholine Receptor ◽

Receptor Ligand ◽

Nicotinic Acetylcholine