scholarly journals Synthesis and Pharmacological Evaluation of 3-[(4-Oxo-4H-pyrido[3,2-e][1,3]thiazin-2-yl)(phenyl)amino]propanenitrile Derivatives as Orally Active AMPA Receptor Antagonists

2019 ◽  
Vol 67 (7) ◽  
pp. 699-706
Author(s):  
Hiroshi Inami ◽  
Jun-ichi Shishikura ◽  
Tomoyuki Yasunaga ◽  
Masaaki Hirano ◽  
Takenori Kimura ◽  
...  
Keyword(s):  
Ampa Receptor ◽  
Receptor Antagonists ◽  
Pharmacological Evaluation ◽  
Orally Active

6-Amino quinazolinedione sulfonamides as orally active competitive AMPA receptor antagonists

2012 ◽  
Vol 22 (2) ◽  
pp. 996-999 ◽  
Author(s):  
David Orain ◽  
Silvio Ofner ◽  
Manuel Koller ◽  
David A. Carcache ◽  
Wolfgang Froestl ◽  
...  
Keyword(s):  
Ampa Receptor ◽  
Receptor Antagonists ◽  
Orally Active

Design, Synthesis, and Pharmacological Evaluation of Piperidin-4-yl amino aryl sulfonamides: Novel, Potent, Selective, Orally Active, and Brain Penetrant 5-HT6 Receptor Antagonists

2012 ◽  
Vol 55 (21) ◽  
pp. 9255-9269 ◽  
Author(s):  
Ramakrishna Nirogi ◽  
Anil Shinde ◽  
Anand Daulatabad ◽  
Ramasastri Kambhampati ◽  
Parandhama Gudla ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Design Synthesis ◽  
Pharmacological Evaluation ◽  
Orally Active

ChemInform Abstract: 5-Aminomethylquinoxaline-2,3-diones. Part 1. A Novel Class of AMPA Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 29 (18) ◽  
pp. no-no
Author(s):  
Y. P. AUBERSON ◽  
S. BISCHOFF ◽  
R. MORETTI ◽  
M. SCHMUTZ ◽  
S. J. VEENSTRA
Keyword(s):  
Ampa Receptor ◽  
Receptor Antagonists

scholarly journals Novel 3-Oxazolidinedione-6-aryl-pyridinones as Potent, Selective, and Orally Active EP3 Receptor Antagonists

2010 ◽  
Vol 1 (7) ◽  
pp. 316-320 ◽  
Author(s):  
Jian Jin ◽  
Ángel Morales-Ramos ◽  
Patrick Eidam ◽  
John Mecom ◽  
Yue Li ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Ep3 Receptor ◽  
Orally Active
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