Radioiodination and biological evaluation of Cladribine as potential agent for tumor imaging and therapy

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AbstractCladribine, a purine analogue antimetabolite, was radioiodinated with

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The novel complex 99mTc(FA-PEG2-HYNIC)(tricine/TPPTS) was clearly visualized at 120 min p.i. at the FR-positive tumor, highlighting its potential as an effective folate receptor tumor imaging agent.


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