Faculty Opinions recommendation of Design, Synthesis, and Pharmacological Characterization of a Neutral, Non-Prodrug Thrombin Inhibitor with Good Oral Pharmacokinetics.

2020 ◽  
Author(s):  
Miles Congreve ◽  
Mark Pickworth
Keyword(s):  
Thrombin Inhibitor ◽  
Pharmacological Characterization ◽  
Design Synthesis ◽  
Oral Pharmacokinetics

scholarly journals Design, Synthesis, and Pharmacological Characterization of a Neutral, Non-Prodrug Thrombin Inhibitor with Good Oral Pharmacokinetics

2020 ◽  
Vol 63 (21) ◽  
pp. 12574-12594
Author(s):  
Alexander Hillisch ◽  
Kersten M. Gericke ◽  
Swen Allerheiligen ◽  
Susanne Roehrig ◽  
Martina Schaefer ◽  
...  
Keyword(s):  
Thrombin Inhibitor ◽  
Pharmacological Characterization ◽  
Design Synthesis ◽  
Oral Pharmacokinetics

scholarly journals Structure-Based Design, Synthesis, and Biochemical and Pharmacological Characterization of Novel Salvinorin A Analogues as Active State Probes of the κ-Opioid Receptor

Biochemistry ◽  
2009 ◽  
Vol 48 (29) ◽  
pp. 6898-6908 ◽  
Author(s):  
Feng Yan ◽  
Ruslan V. Bikbulatov ◽  
Viorel Mocanu ◽  
Nedyalka Dicheva ◽  
Carol E. Parker ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Active State ◽  
Salvinorin A ◽  
Pharmacological Characterization ◽  
Design Synthesis

Design, Synthesis and Pharmacological Characterization of a Potent Radioiodinated and Photoactivatable Peptidic Oxytocin Antagonist∞

2001 ◽  
Vol 44 (18) ◽  
pp. 3022-3030 ◽  
Author(s):  
Eric Carnazzi ◽  
André Aumelas ◽  
Bernard Mouillac ◽  
Christophe Breton ◽  
Laurent Guillou ◽  
...  
Keyword(s):  
Pharmacological Characterization ◽  
Design Synthesis ◽  
Oxytocin Antagonist

Design, Synthesis and Pharmacological Characterization of Endomorphin Analogues with Non-Cyclic Amino Acid Residues in Position 2

2010 ◽  
Vol 106 (2) ◽  
pp. 106-113 ◽  
Author(s):  
Renata Perlikowska ◽  
Jakub Fichna ◽  
Anna WyrÄ™bska ◽  
Jeroen Poels ◽  
Jozef Vanden Broeck ◽  
...  
Keyword(s):  
Amino Acid ◽  
Amino Acid Residues ◽  
Pharmacological Characterization ◽  
Design Synthesis
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