A Novel Synthesis of a 1,3-Disubstituted 1,3-Dihydro-2H-imidazo[4,5-b]pyridin-2-one. Application to GW808990 a CRF1 Receptor Antagonist

Heterocycles ◽  
2010 ◽  
Vol 82 (1) ◽  
pp. 297 ◽  
Author(s):  
Jerome F. Hayes ◽  
Matthew E. Popkin
Keyword(s):  
Receptor Antagonist ◽  
Crf1 Receptor ◽  
Novel Synthesis ◽  
Crf1 Receptor Antagonist

Discovery of 4-chloro-2-(2,4-dichloro-6-methylphenoxy)-1-methyl-7-(pentan-3-yl)-1H-benzimidazole, a novel CRF1 receptor antagonist

2017 ◽  
Vol 25 (5) ◽  
pp. 1556-1570 ◽  
Author(s):  
Michiyo Mochizuki ◽  
Takuto Kojima ◽  
Katsumi Kobayashi ◽  
Etsuo Kotani ◽  
Yuji Ishichi ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Crf1 Receptor ◽  
Crf1 Receptor Antagonist

P.4.c.003 Preliminary evidence of efficacy of a CRF1 receptor antagonist in the 7.5% CO2 model of anxiety

2008 ◽  
Vol 18 ◽  
pp. S494 ◽  
Author(s):  
J.E. Bailey ◽  
A. Papadopoulos ◽  
A. Diaper ◽  
S. Phillips ◽  
M. Schmidt ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Preliminary Evidence ◽  
Crf1 Receptor ◽  
Crf1 Receptor Antagonist

scholarly journals Effect of the CRF1-receptor antagonist pexacerfont on stress-induced eating and food craving

2016 ◽  
Vol 233 (23-24) ◽  
pp. 3921-3932 ◽  
Author(s):  
David H. Epstein ◽  
Ashley P. Kennedy ◽  
Melody Furnari ◽  
Markus Heilig ◽  
Yavin Shaham ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Food Craving ◽  
Crf1 Receptor ◽  
Crf1 Receptor Antagonist
Sign in / Sign up

Export Citation Format

Share Document