Targeting Histone Lysine Demethylases by Truncating the Histone 3 Tail to Obtain Selective Substrate-Based Inhibitors

2011 ◽  
Vol 50 (39) ◽  
pp. 9100-9103 ◽  
Author(s):  
Brian Lohse ◽  
Anders L. Nielsen ◽  
Jan B. L. Kristensen ◽  
Charlotte Helgstrand ◽  
Paul A. C. Cloos ◽  
...  
Keyword(s):  
Histone 3 ◽  
Histone Lysine ◽  
Histone Lysine Demethylases

scholarly journals Posttranslational Modifications of the Histone 3 Tail and Their Impact on the Activity of Histone Lysine Demethylases In Vitro

PLoS ONE ◽  
2013 ◽  
Vol 8 (7) ◽  
pp. e67653 ◽  
Author(s):  
Brian Lohse ◽  
Charlotte Helgstrand ◽  
Jan B. L. Kristensen ◽  
Ulrike Leurs ◽  
Paul A. C. Cloos ◽  
...  
Keyword(s):  
Posttranslational Modifications ◽  
Histone 3 ◽  
Histone Lysine ◽  
Histone Lysine Demethylases

Targeting Histone Lysine Demethylases by Truncating the Histone 3 Tail to Obtain Selective Substrate-Based Inhibitors

2011 ◽  
Vol 123 (39) ◽  
pp. 9266-9269 ◽  
Author(s):  
Brian Lohse ◽  
Anders L. Nielsen ◽  
Jan B. L. Kristensen ◽  
Charlotte Helgstrand ◽  
Paul A. C. Cloos ◽  
...  
Keyword(s):  
Histone 3 ◽  
Histone Lysine ◽  
Histone Lysine Demethylases

Abstract 2128: TACH101, a first-in-class pan inhibitor of KDM4 histone lysine demethylases

2021 ◽  
Author(s):  
Sanghee Yoo ◽  
Chandtip Chandhasin ◽  
Joselyn R. Del Rosario ◽  
Young K. Chen ◽  
Jeff Stafford ◽  
...  
Keyword(s):  
Histone Lysine ◽  
Histone Lysine Demethylases

Histone lysine demethylases as targets for anticancer therapy

2013 ◽  
Vol 12 (12) ◽  
pp. 917-930 ◽  
Author(s):  
Jonas W. Højfeldt ◽  
Karl Agger ◽  
Kristian Helin
Keyword(s):  
Anticancer Therapy ◽  
Histone Lysine ◽  
Histone Lysine Demethylases

scholarly journals Histone lysine demethylases in breast cancer

2013 ◽  
Vol 86 (2) ◽  
pp. 97-103 ◽  
Author(s):  
Elisa Paolicchi ◽  
Francesco Crea ◽  
William L. Farrar ◽  
Jeffrey E. Green ◽  
Romano Danesi
Keyword(s):  
Breast Cancer ◽  
Histone Lysine ◽  
Histone Lysine Demethylases

Honokiol inhibits HIF pathway and hypoxia-induced expression of histone lysine demethylases

2012 ◽  
Vol 422 (3) ◽  
pp. 369-374 ◽  
Author(s):  
Divya Teja Vavilala ◽  
V.K. Chaithanya Ponnaluri ◽  
Ramya Krishna Vadlapatla ◽  
Dhananjay Pal ◽  
Ashim K Mitra ◽  
...  
Keyword(s):  
Induced Expression ◽  
Histone Lysine ◽  
Histone Lysine Demethylases ◽  
Hif Pathway

scholarly journals Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7

2017 ◽  
Vol 129 (49) ◽  
pp. 15761-15765
Author(s):  
Philip A. Gerken ◽  
Jamie R. Wolstenhulme ◽  
Anthony Tumber ◽  
Stephanie B. Hatch ◽  
Yijia Zhang ◽  
...  
Keyword(s):  
Active Inhibitor ◽  
Histone Lysine ◽  
Histone Lysine Demethylases
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