Enantioselective Synthesis of Spiro‐oxiranes: An Asymmetric Addition/Aldol/Spirocyclization Domino Cascade

2021 ◽  
Author(s):  
Ken-Loon Choo ◽  
Bijan Mirabi ◽  
Karl Z. Demmans ◽  
Mark Lautens
Keyword(s):  
Enantioselective Synthesis ◽  
Asymmetric Addition

Core-structure-inspired asymmetric addition reactions: enantioselective synthesis of dihydrobenzoxazinone- and dihydroquinazolinone-based anti-HIV agents

2015 ◽  
Vol 44 (21) ◽  
pp. 7439-7448 ◽  
Author(s):  
Shen Li ◽  
Jun-An Ma
Keyword(s):  
Asymmetric Synthesis ◽  
Core Structure ◽  
Enantioselective Synthesis ◽  
Addition Reactions ◽  
Asymmetric Addition ◽  
Anti Hiv Agents ◽  
Anti Hiv

An overview of the asymmetric synthesis of dihydrobenzoxazinone- and dihydroquinazolinone-based anti-HIV agents (Efavirenz, DPC 961, DPC 963, DPC 083) and analogues was presented.

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