Synthesis, biological evaluation and in silico studies of new pyrazoline derivatives bearing benzo[d]thiazol‐2(3H)‐one moiety as potential urease inhibitors

2022 ◽  
Author(s):  
Fatih Tok ◽  
Nimet Baltaş ◽  
Gizem Tatar ◽  
Bedia Koçyiğit-Kaymakçıoğlu
Keyword(s):  
In Silico ◽  
Biological Evaluation ◽  
Urease Inhibitors ◽  
In Silico Studies

scholarly journals Novel oxindole/benzofuran hybrids as potential dual CDK2/GSK-3β inhibitors targeting breast cancer: design, synthesis, biological evaluation, and in silico studies

2020 ◽  
Vol 36 (1) ◽  
pp. 270-285
Author(s):  
Wagdy M. Eldehna ◽  
Sara T. Al-Rashood ◽  
Tarfah Al-Warhi ◽  
Razan O. Eskandrani ◽  
Amal Alharbi ◽  
...  
Keyword(s):  
Breast Cancer ◽  
In Silico ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
In Silico Studies ◽  
Gsk 3Β

scholarly journals Synthesis, biological evaluation, and in silico studies of novel chalcone- and pyrazoline-based 1,3,5-triazines as potential anticancer agents

RSC Advances ◽  
2020 ◽  
Vol 10 (56) ◽  
pp. 34114-34129
Author(s):  
Leydi M. Moreno ◽  
Jairo Quiroga ◽  
Rodrigo Abonia ◽  
Antonino Lauria ◽  
Annamaria Martorana ◽  
...  
Keyword(s):  
Anticancer Activity ◽  
Anticancer Agents ◽  
In Silico ◽  
Biological Evaluation ◽  
In Silico Studies

A novel series of triazin-chalcones (7,8)a–g and triazin-N-(3,5-dichlorophenyl)pyrazolines (9,10)a–g were synthesized and evaluated for their anticancer activity against nine different cancer strains.

1-[(4′-Chlorophenyl) carbonyl-4-(aryl) thiosemicarbazide derivatives as potent urease inhibitors: Synthesis, in vitro and in silico studies

2018 ◽  
Vol 79 ◽  
pp. 363-371 ◽  
Author(s):  
Basharat Ali ◽  
Khalid Mohammed Khan ◽  
Uzma Salar ◽  
Kanwal ◽  
Safdar Hussain ◽  
...  
Keyword(s):  
In Silico ◽  
Urease Inhibitors ◽  
In Silico Studies ◽  
Thiosemicarbazide Derivatives

Semicarbazone derivatives as urease inhibitors: Synthesis, biological evaluation, molecular docking studies and in-silico ADME evaluation

2018 ◽  
Vol 79 ◽  
pp. 19-26 ◽  
Author(s):  
Syeda Uroos Qazi ◽  
Shafiq Ur Rahman ◽  
Asia Naz Awan ◽  
Mariya al-Rashida ◽  
Rima D. Alharthy ◽  
...  
Keyword(s):  
Molecular Docking ◽  
In Silico ◽  
Docking Studies ◽  
Biological Evaluation ◽  
Urease Inhibitors ◽  
Molecular Docking Studies

Benzylidine indane-1,3-diones: As novel urease inhibitors; synthesis, in vitro, and in silico studies

2018 ◽  
Vol 81 ◽  
pp. 658-671 ◽  
Author(s):  
Bilquees Bano ◽  
Kanwal ◽  
Khalid Mohammed Khan ◽  
Farida Begum ◽  
Muhammad Arif Lodhi ◽  
...  
Keyword(s):  
In Silico ◽  
Urease Inhibitors ◽  
In Silico Studies

Developing potential Helicobacter pylori urease inhibitors from novel oxoindoline derivatives: Synthesis, biological evaluation and in silico study

2018 ◽  
Vol 28 (19) ◽  
pp. 3182-3186 ◽  
Author(s):  
Yu-Shun Yang ◽  
Mi-Mi Su ◽  
Xu-Ping Zhang ◽  
Qi-Xing Liu ◽  
Zhen-Xiang He ◽  
...  
Keyword(s):  
Helicobacter Pylori ◽  
In Silico ◽  
Biological Evaluation ◽  
Urease Inhibitors ◽  
In Silico Study

Novel pyrazine based anti-tubercular agents: Design, synthesis, biological evaluation and in silico studies

2020 ◽  
Vol 96 ◽  
pp. 103610 ◽  
Author(s):  
Nayera W. Hassan ◽  
Manal N. Saudi ◽  
Yasser S. Abdel-Ghany ◽  
Azza Ismail ◽  
Perihan A. Elzahhar ◽  
...  
Keyword(s):  
In Silico ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
In Silico Studies

Synthesis, biological evaluation and in silico studies of novel N-substituted phthalazine sulfonamide compounds as potent carbonic anhydrase and acetylcholinesterase inhibitors

2019 ◽  
Vol 89 ◽  
pp. 103004 ◽  
Author(s):  
Cüneyt Türkeş ◽  
Mustafa Arslan ◽  
Yeliz Demir ◽  
Liridon Çoçaj ◽  
Arleta Rifati Nixha ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
In Silico ◽  
Acetylcholinesterase Inhibitors ◽  
Biological Evaluation ◽  
In Silico Studies
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