ChemInform Abstract: Substituted N-Phenylcarbamates as Histamine H3 Receptor Antagonists with Improved in vivo Potency.

ChemInform ◽  
2010 ◽  
Vol 31 (24) ◽  
pp. no-no
Author(s):  
S. Reidemeister ◽  
H. Stark ◽  
X. Ligneau ◽  
C. R. Ganellin ◽  
J.-C. Schwartz ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

scholarly journals Design, synthesis, and in vitro and in vivo characterization of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines and their piperidine analogues as histamine H3 receptor antagonists

MedChemComm ◽  
2019 ◽  
Vol 10 (2) ◽  
pp. 234-251 ◽  
Author(s):  
Marek Staszewski ◽  
Anna Stasiak ◽  
Tadeusz Karcz ◽  
Daniel McNaught Flores ◽  
Wiesława Agnieszka Fogel ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Design Synthesis ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
In Vivo Characterization ◽  
Histamine H3

The prominent members of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines as histamine H3 receptor antagonists.

In vivo evaluation of effects of histamine H3 receptor antagonists on methamphetamine-induced hyperlocomotion in mice

2020 ◽  
Vol 1740 ◽  
pp. 146873
Author(s):  
Junichi Kitanaka ◽  
Nobue Kitanaka ◽  
F. Scott Hall ◽  
Yukie Amatsu ◽  
Kotaku Hashimoto ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
In Vivo Evaluation ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

ChemInform Abstract: 4-Chlorobenzyl Sulfonamide and Sulfamide Derivatives of Histamine Homologues: The Design of Potent Histamine H3 Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 31 (8) ◽  
pp. no-no
Author(s):  
Matthew J. Tozer ◽  
Ildiko M. Buck ◽  
Tracey Cooke ◽  
S. Barret Kalindjian ◽  
Iain M. McDonald ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Derivatives Of ◽  
Histamine H3

scholarly journals A Novel Potent and Selective Histamine H3 Receptor Antagonist Enerisant: In Vitro Profiles, In Vivo Receptor Occupancy, and Wake-Promoting and Procognitive Effects in Rodents

2020 ◽  
Vol 375 (2) ◽  
pp. 276-285
Author(s):  
Noriko Hino ◽  
Toshiyuki Marumo ◽  
Makiko Kotani ◽  
Toshiharu Shimazaki ◽  
Ayaka Kaku-Fukumoto ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Receptor Occupancy ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Piperidine-Containing Histamine H3 Receptor Antagonists of the Carbamate Series: The Influence of the Additional Ether Functionality

ChemInform ◽  
2003 ◽  
Vol 34 (16) ◽  
Author(s):  
D. Lazewska ◽  
K. Kiec-Kononowicz ◽  
H. H. Pertz ◽  
S. Elz ◽  
H. Stark ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Keynote review: Histamine H3 receptor antagonists reach out for the clinic

2005 ◽  
Vol 10 (23-24) ◽  
pp. 1613-1627 ◽  
Author(s):  
Sylvain Celanire ◽  
Maikel Wijtmans ◽  
Patrice Talaga ◽  
Rob Leurs ◽  
Iwan J.P. de Esch
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

scholarly journals Synthesis and evaluation of N-alkyl-S-[3-(piperidin-1-yl)propyl]isothioureas: High affinity and human/rat species-selective histamine H3 receptor antagonists

2013 ◽  
Vol 23 (23) ◽  
pp. 6415-6420 ◽  
Author(s):  
Shinya Harusawa ◽  
Koichi Sawada ◽  
Takuji Magata ◽  
Hiroki Yoneyama ◽  
Lisa Araki ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
High Affinity ◽  
H3 Receptor ◽  
Histamine H3
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