A Mild and Efficient Method for Copper-Catalyzed Ullmann-Type N-Arylation of Aliphatic Amines and Amino Acids.

ChemInform ◽  
2007 ◽  
Vol 38 (48) ◽  
Author(s):  
Qun Jiang ◽  
Deshou Jiang ◽  
Yuyang Jiang ◽  
Hua Fu ◽  
Yufen Zhao
Synlett ◽  
2007 ◽  
Vol 2007 (12) ◽  
pp. 1836-1842 ◽  
Author(s):  
Yuyang Jiang ◽  
Hua Fu ◽  
Qun Jiang ◽  
Deshou Jiang ◽  
Yufen Zhao

2019 ◽  
Author(s):  
Yongzheng Ding ◽  
Shuai Fan ◽  
Xiaoxi Chen ◽  
yuzhen gao ◽  
Gang Li

A Pdᴵᴵ-catalyzed, ligand-enabled gamma-C(sp3)–H arylation of free primary aliphatic amines and amino esters without using an exogenous directing group is reported. This reaction is compatible with unhindered free aliphatic amines, and it is also be applicable to the rapid synthesis of biologically and synthetically valuable unnatural α-amino acids. Large scale synthesis is also feasible using this method.<br>


1999 ◽  
Vol 23 (7) ◽  
pp. 424-425
Author(s):  
T. Naqvi ◽  
M. Bhattacharya ◽  
W. Haq
Keyword(s):  

Reduction of pentachlorophenyl esters of Boc protected amino acids and peptides to the corresponding alcohols is described.


2016 ◽  
Vol 14 (2) ◽  
pp. 556-563 ◽  
Author(s):  
Veladi Panduranga ◽  
Girish Prabhu ◽  
Roopesh Kumar ◽  
Basavaprabhu Basavaprabhu ◽  
Vommina V. Sureshbabu

A simple and efficient method for the synthesis of N,N’-orthogonally protected imide tethered peptidomimetics is presented. The imide peptidomimetics were synthesized by coupling the in situ generated selenocarboxylate of Nα-protected amino acids with Nα-protected amino acid azides in good yields.


2009 ◽  
Vol 131 (30) ◽  
pp. 10711-10718 ◽  
Author(s):  
Mathieu Branca ◽  
Sébastien Pena ◽  
Régis Guillot ◽  
Didier Gori ◽  
Valérie Alezra ◽  
...  

2019 ◽  
Vol 58 (17) ◽  
pp. 5633-5638 ◽  
Author(s):  
Srimanta Guin ◽  
Pravas Dolui ◽  
Xinglong Zhang ◽  
Satyadip Paul ◽  
Vikas Kumar Singh ◽  
...  

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