New Anticancer Agents: Design, Synthesis, Biological Activity, and Molecular Docking of Bicyclic Phloroglucinol Derivatives

2021 ◽  
Vol 6 (7) ◽  
pp. 1453-1457
Author(s):  
Pei Yan ◽  
Qingfu Lai ◽  
Ming Li ◽  
Xiaobao Jin ◽  
Gao Wie ◽  
...  
Keyword(s):  
Biological Activity ◽  
Molecular Docking ◽  
Anticancer Agents ◽  
Design Synthesis ◽  
Phloroglucinol Derivatives

Design, synthesis, and molecular docking of novel indole scaffold-based VEGFR-2 inhibitors as targeted anticancer agents

2018 ◽  
Vol 351 (2) ◽  
pp. 1700299 ◽  
Author(s):  
Hanaa M. Roaiah ◽  
Iman A. Y. Ghannam ◽  
Islam H. Ali ◽  
Ahmed M. El Kerdawy ◽  
Mamdouh M. Ali ◽  
...  
Keyword(s):  
Molecular Docking ◽  
Anticancer Agents ◽  
Design Synthesis

scholarly journals Design, Synthesis, Molecular Docking and Antibacterial Screening of Some Quinolone Compounds

Proceedings ◽  
2019 ◽  
Vol 29 (1) ◽  
pp. 2
Author(s):  
Lucia Pintilie ◽  
Constantin Tanase ◽  
Elena Mihai ◽  
Maria Maganu ◽  
Miron Teodor Caproiu
Keyword(s):  
Biological Activity ◽  
Molecular Docking ◽  
Design Synthesis ◽  
Antibacterial Screening ◽  
Antibacterial Spectrum ◽  
Broad Antibacterial Spectrum

Drugs belonging to the quinolone compounds are characterized by a quicker biological activity and a broad antibacterial spectrum [1–4]. [...]

Design, synthesis and biological activities of pyrrole-3-carboxamide derivatives as EZH2 (enhancer of zeste homologue 2) inhibitors and anticancer agents

2020 ◽  
Vol 44 (6) ◽  
pp. 2247-2255
Author(s):  
Qifan Zhou ◽  
Lina Jia ◽  
Fangyu Du ◽  
Xiaoyu Dong ◽  
Wanyu Sun ◽  
...  
Keyword(s):  
Biological Activity ◽  
Anticancer Agents ◽  
Biological Activities ◽  
Activity Assay ◽  
Design Synthesis ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Enhancer Of Zeste

A novel series of pyrrole-3-carboxamides targeting EZH2 have been designed and synthesized. The structure–activity relationships were summarized by combining with in vitro biological activity assay and docking results.

Design, Synthesis and Biological Activity of 1,2-Benzothiazine Derivatives as Potential Anticancer Agents

2014 ◽  
Vol 34 (10) ◽  
pp. 2040 ◽  
Author(s):  
Jie Wang ◽  
Qinlong Xu ◽  
Jiaming Li ◽  
Enli Zhang ◽  
Minhua Hu ◽  
...  
Keyword(s):  
Biological Activity ◽  
Anticancer Agents ◽  
Design Synthesis
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