The Evolution of Drug-Receptor Models: The Cubic Ternary Complex Model for G Protein-Coupled Receptors

Receptor Models ◽

Ternary Complex Model ◽

Drug Receptor ◽

1P388 Relevance of ternary complex model to intracellular dynamics of G protein-coupled chemoattractant receptor in living Dictyostelium cells(15. Cellular signal transduction,Poster Session,Abstract,Meeting Program of EABS & BSJ 2006)

Seibutsu Butsuri ◽

10.2142/biophys.46.s243_4 ◽

2006 ◽

Vol 46 (supplement2) ◽

pp. S243

Author(s):

Yukihiro Miyanaga ◽

Hidekazu Kuwayama ◽

Toshio Yanagida ◽

Masahiro Ueda

Keyword(s):

Signal Transduction ◽

G Protein ◽

Ternary Complex ◽

Poster Session ◽

Complex Model ◽

Cellular Signal Transduction ◽

Meeting Program ◽

Cellular Signal ◽

Ternary Complex Model ◽

Tiotidine, a Histamine H2 Receptor Inverse Agonist That Binds with High Affinity to an Inactive G-Protein—Coupled Form of the Receptor. Experimental Support for the Cubic Ternary Complex Model

Molecular Pharmacology ◽

10.1124/mol.64.2.512 ◽

2003 ◽

Vol 64 (2) ◽

pp. 512-520 ◽

Cited By ~ 33

Author(s):

Federico Monczor ◽

Natalia Fernández ◽

Bibiana Lemos Legnazzi ◽

Maria Eugenia Riveiro ◽

Alberto Baldi ◽

...

Keyword(s):

G Protein ◽

Ternary Complex ◽

Complex Model ◽

Histamine H2 Receptor ◽

H2 Receptor ◽

High Affinity ◽

Experimental Support ◽

Ternary Complex Model ◽

G Protein Coupled ◽

Receptor Inverse Agonist

G protein activation by G protein coupled receptors: ternary complex formation or catalyzed reaction?

Biochemical Pharmacology ◽

10.1016/j.bcp.2004.05.044 ◽

2004 ◽

Vol 68 (5) ◽

pp. 799-806 ◽

Cited By ~ 31

Author(s):

David J Roberts ◽

Magali Waelbroeck

Keyword(s):

Complex Formation ◽

G Protein ◽

Ternary Complex ◽

Protein Activation ◽

Ternary Complex Formation ◽

G Protein Activation ◽

Analysis of Drug-receptor Interactions Using Radioligand Binding Assays on G Protein-coupled Receptors

Affinity and Efficacy ◽

10.1142/9789814324229_0013 ◽

2014 ◽

pp. 677-730

Keyword(s):

G Protein ◽

Radioligand Binding ◽

Binding Assays ◽

Receptor Interactions ◽

Drug Receptor ◽

Signal Transduction by G Protein-Coupled Receptors - Molecular Biology Intelligence Unit ◽

The (Extended) Ternary Complex Model ([E]TCM) for G Protein Activation

10.1007/978-1-4684-1407-3_5 ◽

1997 ◽

pp. 63-73 ◽

Cited By ~ 1

Author(s):

Paul H. J. Nederkoorn ◽

Henk Timmerman ◽

Gabriëlle M. Donné-Op den Kelder

Keyword(s):

G Protein ◽

Ternary Complex ◽

Complex Model ◽

Protein Activation ◽

G Protein Activation ◽

Ternary Complex Model

Oligomerization in Health and Disease: From Enzymes to G Protein-Coupled Receptors

10.1016/s1877-1173(20)x0002-0 ◽

2020 ◽

Keyword(s):

G Protein ◽

Health And Disease ◽

G Protein-Coupled Receptors Part A

10.1016/s0091-679x(17)x0006-x ◽

2017 ◽

Keyword(s):

G Protein ◽

G Protein-Coupled Receptors - Signaling, Trafficking and Regulation

10.1016/s0091-679x(16)x0002-7 ◽

2016 ◽

Keyword(s):

G Protein ◽

Enhanced Salmonella virulence instigated by bactivorous protozoa and investigation of putative protozoan G protein-coupled receptors associated with bacterial engulfment

10.31274/etd-180810-61 ◽

2014 ◽

Author(s):

Matt T. Brewer

Keyword(s):

G Protein ◽

Salmonella Virulence ◽

Faculty Opinions recommendation of Modulation of postendocytic sorting of G protein-coupled receptors.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1008239.104108 ◽

2002 ◽

Author(s):

Silvia Arber

Keyword(s):

G Protein ◽