The second extracellular loop of GPCRs determines subtype-selectivity and controls efficacy as evidenced by loop exchange study at A2 adenosine receptors

2013 ◽  
Vol 85 (9) ◽  
pp. 1317-1329 ◽  
Author(s):  
Benjamin F. Seibt ◽  
Anke C. Schiedel ◽  
Dominik Thimm ◽  
Sonja Hinz ◽  
Farag F. Sherbiny ◽  
...  
Keyword(s):  
Adenosine Receptors ◽  
Extracellular Loop ◽  
Subtype Selectivity ◽  
Exchange Study ◽  
A2 Adenosine Receptors

A2A and A2B adenosine receptors: The extracellular loop 2 determines high (A2A) or low affinity (A2B) for adenosine

2020 ◽  
Vol 172 ◽  
pp. 113718 ◽  
Author(s):  
Elisabetta De Filippo ◽  
Sonja Hinz ◽  
Veronica Pellizzari ◽  
Giuseppe Deganutti ◽  
Ali El-Tayeb ◽  
...  
Keyword(s):  
Adenosine Receptors ◽  
Extracellular Loop ◽  
Loop 2

A1 and A2 Adenosine Receptors in Synovial Cells from Patients with Rheumatic Diseases

1989 ◽  
pp. 429-433 ◽  
Author(s):  
Claudia Martini ◽  
Gino Giannaccini ◽  
Antonio Lucacchini ◽  
Laura Bazzichi ◽  
Annalia Soletti ◽  
...  
Keyword(s):  
Rheumatic Diseases ◽  
Adenosine Receptors ◽  
Synovial Cells ◽  
A2 Adenosine Receptors

Homospecific regulation of A1 and A2 adenosine receptors

1990 ◽  
Vol 22 ◽  
pp. 431
Author(s):  
A.M. Rosati ◽  
C. Florio ◽  
U. Traversa ◽  
R. Vertua
Keyword(s):  
Adenosine Receptors ◽  
A2 Adenosine Receptors

scholarly journals Xanthine functionalized congeners as potent ligands at A2-adenosine receptors

1987 ◽  
Vol 30 (1) ◽  
pp. 211-214 ◽  
Author(s):  
Kenneth A. Jacobson ◽  
Dieter Ukena ◽  
William Padgett ◽  
John W. Daly ◽  
Kenneth L. Kirk
Keyword(s):  
Adenosine Receptors ◽  
A2 Adenosine Receptors

scholarly journals Characterization of Human Striatal A2-Adenosine Receptors Using Radioligand Binding and Photoaffinity Labeling

1992 ◽  
Vol 12 (2) ◽  
pp. 149-169 ◽  
Author(s):  
Xiao-Duo Ji ◽  
Gary L. Stiles ◽  
Philip J.M. van Galen ◽  
Kenneth A. Jacobson
Keyword(s):  
Adenosine Receptors ◽  
Radioligand Binding ◽  
Photoaffinity Labeling ◽  
A2 Adenosine Receptors
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