Design, synthesis and biological evaluation of pyrimidine-based derivatives as VEGFR-2 tyrosine kinase inhibitors

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

WITHDRAWN: Design, synthesis and biological evaluation of 3-substituted-4-anilinequinoline as EGFR tyrosine kinase inhibitors

10.1016/j.bmcl.2012.10.030 ◽

2012 ◽

Author(s):

Yongjun Mao ◽

Kai Xie ◽

Wenxiu Zhu ◽

Jianfeng Li ◽

Hua Xie ◽

...

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

Design, synthesis and biological evaluation of novel pyrimidine, 3-cyanopyridine and m-amino-N-phenylbenzamide based monocyclic EGFR tyrosine kinase inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2013.03.053 ◽

2013 ◽

Vol 21 (11) ◽

pp. 3090-3104 ◽

Cited By ~ 18

Author(s):

Yongjun Mao ◽

Wenxiu Zhu ◽

Xiaoguang Kong ◽

Zhen Wang ◽

Hua Xie ◽

...

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

The design, synthesis, and biological evaluation of potent receptor tyrosine kinase inhibitors

10.1016/j.bmcl.2012.06.029 ◽

2012 ◽

Vol 22 (15) ◽

pp. 4979-4985 ◽

Cited By ~ 13

Author(s):

Moon H. Kim ◽

Amy Lew Tsuhako ◽

Erick W. Co ◽

Dana T. Aftab ◽

Frauke Bentzien ◽

...

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Design, synthesis and biological evaluation of substituted pyrrolo[2,3-d]pyrimidines as multiple receptor tyrosine kinase inhibitors and antiangiogenic agents

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2008.04.019 ◽

2008 ◽

Vol 16 (10) ◽

pp. 5514-5528 ◽

Cited By ~ 22

Author(s):

Aleem Gangjee ◽

Ojas A. Namjoshi ◽

Jianming Yu ◽

Michael A. Ihnat ◽

Jessica E. Thorpe ◽

...

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Antiangiogenic Agents ◽

Design Synthesis ◽

Multiple Receptor ◽

Design, synthesis, and biological evaluation of novel 3-pyrrolo[b]cyclohexylene-2-dihydroindolinone derivatives as potent receptor tyrosine kinase inhibitors

10.1016/j.bmcl.2013.08.037 ◽

2013 ◽

Vol 23 (20) ◽

pp. 5630-5633 ◽

Cited By ~ 8

Author(s):

Lei Ding ◽

Feng Tang ◽

Wei Huang ◽

Qiu Jin ◽

Han Shen ◽

...

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Part-1: Design, synthesis and biological evaluation of novel bromo-pyrimidine analogs as tyrosine kinase inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2016.04.056 ◽

2016 ◽

Vol 119 ◽

pp. 70-82 ◽

Cited By ~ 10

Author(s):

Chandrashekar Suradhenupura Munikrishnappa ◽

Sangamesh B. Puranik ◽

G.V. Suresh Kumar ◽

Y. Rajendra Prasad

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Pyrimidine Analogs ◽

Scaffold oriented synthesis. Part 2: Design, synthesis and biological evaluation of pyrimido-diazepines as receptor tyrosine kinase inhibitors

10.1016/j.bmcl.2008.03.021 ◽

2008 ◽

Vol 18 (8) ◽

pp. 2691-2695 ◽

Cited By ~ 20

Author(s):

Vijaya Gracias ◽

Zhiqin Ji ◽

Irini Akritopoulou-Zanze ◽

Cele Abad-Zapatero ◽

Jeffrey R. Huth ◽

...

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Design, Synthesis and Biological Evaluation of Quinoxalin-2(1H)-one Derivatives as EGFR Tyrosine Kinase Inhibitors

Anti-Cancer Agents in Medicinal Chemistry ◽

10.2174/187152061502150116173357 ◽

2015 ◽

Vol 15 (2) ◽

pp. 267-273 ◽

Cited By ~ 5

Author(s):

Xuemei Qin ◽

Xiao Han ◽

Liming Hu ◽

Zhipeng Li ◽

Zhufeng Geng ◽

...

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

Design, synthesis, and biological evaluation of novel bromo-pyrimidine analogues as tyrosine kinase inhibitors

Arabian Journal of Chemistry ◽

10.1016/j.arabjc.2021.103054 ◽

2021 ◽

Vol 14 (4) ◽

pp. 103054

Author(s):

Chandrashekar S. Munikrishnappa ◽

G.V. Suresh Kumar ◽

Richie R. Bhandare ◽

Afzal B. Shaik

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Pyrimidine Analogues ◽

Design, synthesis, and biological evaluation of 1,3,5-trisubstituted pyrazoles as tyrosine kinase inhibitors

Medicinal Chemistry Research ◽

10.1007/s00044-018-2282-x ◽

2019 ◽

Vol 28 (3) ◽

pp. 267-278 ◽

Cited By ~ 3

Author(s):

Sinthiya J. Gawandi ◽

Vidya G. Desai ◽

Sunil G. Shingade

Keyword(s):

Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽