Synthesis and structure–activity relationship study of novel cytotoxic carbamate and N-acylheterocyclic bearing derivatives of betulin and betulinic acid

Activity Relationship ◽

Structure Activity ◽

Relationship Study ◽

Quantitative structure-activity relationship study of ATP-sensitive potassium channel openers: Derivatives of 3-alkylamino-4H-1,2,4-benzothiadiazine 1,1-dioxide

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756360701442381 ◽

2008 ◽

Vol 23 (1) ◽

pp. 1-6 ◽

Cited By ~ 5

Author(s):

B. K. Sharma ◽

S. K. Sharma ◽

P. Singh ◽

Susheela Sharma

Keyword(s):

Potassium Channel ◽

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Potassium Channel Openers ◽

Structure Activity ◽

Relationship Study ◽

Structure−Activity Relationship Study of Betulinic Acid, A Novel and Selective TGR5 Agonist, and Its Synthetic Derivatives: Potential Impact in Diabetes¶

Journal of Medicinal Chemistry ◽

10.1021/jm900872z ◽

2010 ◽

Vol 53 (1) ◽

pp. 178-190 ◽

Cited By ~ 120

Author(s):

Cédric Genet ◽

Axelle Strehle ◽

Céline Schmidt ◽

Geoffrey Boudjelal ◽

Annelise Lobstein ◽

...

Keyword(s):

Betulinic Acid ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study ◽

Potential Impact ◽

Synthetic Derivatives

Influence of lipophilicity in O ‐acyl and O ‐alkyl derivatives of juglone and lawsone: a structure–activity relationship study in the search for natural herbicide models

Pest Management Science ◽

10.1002/ps.4764 ◽

2017 ◽

Vol 74 (3) ◽

pp. 682-694 ◽

Cited By ~ 7

Author(s):

Alexandra G Durán ◽

Nuria Chinchilla ◽

José MG Molinillo ◽

Francisco A Macías

Keyword(s):

Activity Relationship ◽

Natural Herbicide ◽

Structure Activity ◽

Alkyl Derivatives ◽

Relationship Study ◽

Synthesis and In Vitro Antimicrobial Activity of Medicinally Important Novel N-alkyl, N-aryl and Urea Derivatives of 1-benzhydryl Piperizine: A Structure-Activity Relationship Study

Letters in Drug Design & Discovery ◽

10.2174/157018009787582570 ◽

2009 ◽

Vol 6 (2) ◽

pp. 146-154

Author(s):

Channapillekoppal Ananda Kumar ◽

Karunakara Murthy ◽

Marlinganadoddi Sadashiva ◽

Mallappanahally Vinaya ◽

Naraganahalli Thimmegowda ◽

...

Keyword(s):

Antimicrobial Activity ◽

Activity Relationship ◽

Urea Derivatives ◽

In Vitro Antimicrobial Activity ◽

Structure Activity ◽

Relationship Study ◽

Quantitative Structure-activity Relationship Study of Betulinic Acid Derivatives Against HIV using SMILES-based Descriptors

Current Computer - Aided Drug Design ◽

10.2174/1573409914666180112094156 ◽

2018 ◽

Vol 14 (2) ◽

pp. 152-159 ◽

Cited By ~ 3

Author(s):

Apilak Worachartcheewan ◽

Alla P. Toropova ◽

Andrey A. Toropov ◽

Suphakit Siriwong ◽

Jatupat Prapojanasomboon ◽

...

Keyword(s):

Betulinic Acid ◽

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Study

Anti-AIDS agents 73: Structure–activity relationship study and asymmetric synthesis of 3-O-monomethylsuccinyl-betulinic acid derivatives

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.09.081 ◽

2007 ◽

Vol 17 (23) ◽

pp. 6553-6557 ◽

Cited By ~ 23

Author(s):

Keduo Qian ◽

Kyoko Nakagawa-Goto ◽

Donglei Yu ◽

Susan L. Morris-Natschke ◽

Theodore J. Nitz ◽

...

Keyword(s):

Asymmetric Synthesis ◽

Betulinic Acid ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study

Prejunctional effect of quaternary derivatives of l-hyoscyamine at the rat neuromuscular junction. A structure-activity relationship study

General Pharmacology The Vascular System ◽

10.1016/0306-3623(94)90164-3 ◽

1994 ◽

Vol 25 (7) ◽

pp. 1397-1404 ◽

Cited By ~ 3

Author(s):

Caden Souccar ◽

Janete Do Carmo Soldera ◽

Roberta Monterazzo Cysneiros ◽

Maria Do Carmo Gonçalo ◽

Antonio José Lapa

Keyword(s):

Neuromuscular Junction ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study ◽

Structure-Activity Relationship Study Reveals Benzazepine Derivatives of Luteolin as New Aldose Reductase Inhibitors for Diabetic Cataract

Current Drug Discovery Technologies ◽

10.2174/1570163813666160701023100 ◽

2016 ◽

Vol 13 (3) ◽

pp. 152-163 ◽

Cited By ~ 2

Author(s):

Jomon Sebastian

Keyword(s):

Aldose Reductase ◽

Activity Relationship ◽

Diabetic Cataract ◽

Aldose Reductase Inhibitors ◽

Reductase Inhibitors ◽

Structure Activity ◽

Relationship Study ◽

Quantitative structure–activity relationship study of new potent and selective antagonists at the 5-HT1Aand adrenergic α1dreceptors: Derivatives of spiroethyl phenyl(substituted)piperazine

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756360600810175 ◽

2006 ◽

Vol 21 (5) ◽

pp. 601-607

Author(s):

B. K. Sharma ◽

P. Singh ◽

Susheela Sharma

Keyword(s):

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Selective Antagonists ◽

Relationship Study ◽

Substituted Piperazine ◽

Anti-AIDS Agents 81. Design, Synthesis, and Structure−Activity Relationship Study of Betulinic Acid and Moronic Acid Derivatives as Potent HIV Maturation Inhibitors†

Journal of Medicinal Chemistry ◽

10.1021/jm901782m ◽

2010 ◽

Vol 53 (8) ◽

pp. 3133-3141 ◽

Cited By ~ 45

Author(s):

Keduo Qian ◽

Reen-Yun Kuo ◽

Chin-Ho Chen ◽

Li Huang ◽

Susan L. Morris-Natschke ◽

...

Keyword(s):

Betulinic Acid ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Study