Synthesis and In Vitro Antimicrobial Activity of Medicinally Important Novel N-alkyl, N-aryl and Urea Derivatives of 1-benzhydryl Piperizine: A Structure-Activity Relationship Study

2009 ◽  
Vol 6 (2) ◽  
pp. 146-154
Author(s):  
Channapillekoppal Ananda Kumar ◽  
Karunakara Murthy ◽  
Marlinganadoddi Sadashiva ◽  
Mallappanahally Vinaya ◽  
Naraganahalli Thimmegowda ◽  
...  
Keyword(s):  
Antimicrobial Activity ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Urea Derivatives ◽  
In Vitro Antimicrobial Activity ◽  
Structure Activity ◽  
Relationship Study ◽  
Derivatives Of

scholarly journals From in vitro to in cellulo: structure–activity relationship of (2-nitrophenyl)methanol derivatives as inhibitors of PqsD in Pseudomonas aeruginosa

2014 ◽  
Vol 12 (32) ◽  
pp. 6094-6104 ◽  
Author(s):  
Michael P. Storz ◽  
Giuseppe Allegretta ◽  
Benjamin Kirsch ◽  
Martin Empting ◽  
Rolf W. Hartmann
Keyword(s):  
Pseudomonas Aeruginosa ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Relationship Of ◽  
Derivatives Of

More than 60 derivatives of (2-nitrophenyl)methanol were synthesized and evaluated regarding their potency to inhibit PqsD. In vitro and in cellulo structure–activity relationships were derived.

Synthesis of tyrosol glycosides and their structure–activity relationship study in biochemical assays and in human cells in vitro

2017 ◽  
Vol 280 ◽  
pp. S118
Author(s):  
Eva Horvathova ◽  
Eliska Galova ◽  
Andrea Sevcovicova ◽  
Martina Klapakova ◽  
Andrej Bohac ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Human Cells ◽  
Activity Relationship ◽  
Structure Activity ◽  
Biochemical Assays ◽  
Relationship Study
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