Design, synthesis and pharmacological evaluation of spirocyclic σ1 receptor ligands with exocyclic amino moiety (increased distance 1)

2011 ◽  
Vol 19 (10) ◽  
pp. 3141-3151 ◽  
Author(s):  
Elisabeth Rack ◽  
Roland Fröhlich ◽  
Dirk Schepmann ◽  
Bernhard Wünsch
Keyword(s):  
Receptor Ligands ◽  
Design Synthesis ◽  
Pharmacological Evaluation ◽  
Σ1 Receptor

Design, synthesis and pharmacological evaluation of 4-(piperazin-1-yl methyl)-N1-arylsulfonyl indole derivatives as 5-HT6 receptor ligands

2012 ◽  
Vol 22 (24) ◽  
pp. 7431-7435 ◽  
Author(s):  
Ramakrishna V.S. Nirogi ◽  
Rajeshkumar Badange ◽  
Ramasastri Kambhampati ◽  
Anil Chindhe ◽  
Amol D. Deshpande ◽  
...  
Keyword(s):  
Indole Derivatives ◽  
Receptor Ligands ◽  
Design Synthesis ◽  
Pharmacological Evaluation

Identification, pharmacological evaluation and binding mode analysis of novel chromene and chromane based σ1 receptor ligands

2014 ◽  
Vol 83 ◽  
pp. 526-533 ◽  
Author(s):  
Erik Laurini ◽  
Dipak Harel ◽  
Domenico Marson ◽  
Dirk Schepmann ◽  
Thomas J. Schmidt ◽  
...  
Keyword(s):  
Binding Mode ◽  
Mode Analysis ◽  
Receptor Ligands ◽  
Pharmacological Evaluation ◽  
Σ1 Receptor

scholarly journals Design, synthesis and pharmacological evaluation of conformationally restricted N-arylsulfonyl-3-aminoalkoxy indoles as a potential 5-HT6 receptor ligands

2011 ◽  
Vol 26 (3) ◽  
pp. 341-349 ◽  
Author(s):  
Ramakrishna V.S. Nirogia ◽  
Ramasastri Kambhampati ◽  
Anand V. Daulatabad ◽  
Parandhama Gudla ◽  
Mohammad Shaikh ◽  
...  
Keyword(s):  
Receptor Ligands ◽  
Design Synthesis ◽  
Conformationally Restricted ◽  
Pharmacological Evaluation

Design, Synthesis and Pharmacological Evaluation of 5-Hydroxytryptamine1a Receptor Ligands to Explore the Three-Dimensional Structure of the Receptor

2002 ◽  
Vol 62 (1) ◽  
pp. 15-21 ◽  
Author(s):  
Marı́a L. López-Rodrı́guez ◽  
Bruno Vicente ◽  
Xavier Deupi ◽  
Sergio Barrondo ◽  
Mireia Olivella ◽  
...  
Keyword(s):  
Three Dimensional ◽  
Dimensional Structure ◽  
Receptor Ligands ◽  
Design Synthesis ◽  
Three Dimensional Structure ◽  
Pharmacological Evaluation

Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists

2021 ◽  
pp. 104782
Author(s):  
Lin Lin ◽  
Guangyao Lin ◽  
Qingtong Zhou ◽  
Ross A.D. Bathgate ◽  
Grace Qun Gong ◽  
...  
Keyword(s):  
Design Synthesis ◽  
Pharmacological Evaluation

Design, synthesis and biological evaluation of piperazine analogues as CB1 cannabinoid receptor ligands

2008 ◽  
Vol 16 (7) ◽  
pp. 4035-4051 ◽  
Author(s):  
Kwang-Seop Song ◽  
Sung-Han Lee ◽  
Hyun Ji Chun ◽  
Jong Yup Kim ◽  
Myung Eun Jung ◽  
...  
Keyword(s):  
Cannabinoid Receptor ◽  
Biological Evaluation ◽  
Receptor Ligands ◽  
Design Synthesis ◽  
Cb1 Cannabinoid Receptor ◽  
Synthesis And Biological Evaluation

Design, Synthesis, and Pharmacological Evaluation of Glutamate Carboxypeptidase II (GCPII) Inhibitors Based on Thioalkylbenzoic Acid Scaffolds

2012 ◽  
Vol 55 (12) ◽  
pp. 5922-5932 ◽  
Author(s):  
Doris Stoermer ◽  
Dilrukshi Vitharana ◽  
Niyada Hin ◽  
Greg Delahanty ◽  
Bridget Duvall ◽  
...  
Keyword(s):  
Design Synthesis ◽  
Glutamate Carboxypeptidase Ii ◽  
Pharmacological Evaluation ◽  
Glutamate Carboxypeptidase
Sign in / Sign up

Export Citation Format

Share Document