Tyrosine modified analogues of the α4β7 integrin inhibitor biotin-R8ERY prepared via Click Chemistry: Synthesis and biological evaluation

2012 ◽  
Vol 20 (8) ◽  
pp. 2638-2644 ◽  
Author(s):  
Stefanie Papst ◽  
Anaïs Noisier ◽  
Margaret A. Brimble ◽  
Yi Yang ◽  
Geoffrey W. Krissansen
Keyword(s):  
Click Chemistry ◽  
Biological Evaluation ◽  
Synthesis And Biological Evaluation ◽  
Integrin Inhibitor

Synthesis and Biological Evaluation of Triazolyl Monastrol Analogues Using Cu-Catalyzed Click Chemistry

Heterocycles ◽  
2017 ◽  
Vol 94 (10) ◽  
pp. 1856 ◽  
Author(s):  
Hani Mutlak A. Hassan ◽  
Iuliana Denetiu ◽  
Kaltoom Sakkaf ◽  
Khalid A. Khan ◽  
Peter N. Pushparaj ◽  
...  
Keyword(s):  
Click Chemistry ◽  
Biological Evaluation ◽  
Synthesis And Biological Evaluation

Synthesis and biological evaluation of fluorinated analogues of ripostatin A

2019 ◽  
Vol 17 (6) ◽  
pp. 1362-1364 ◽  
Author(s):  
Vladyslav Shenderman ◽  
Evgeny V. Prusov
Keyword(s):  
Click Chemistry ◽  
Biological Evaluation ◽  
Last Stage ◽  
Synthesis And Biological Evaluation ◽  
Derivatives Of

A last stage click-chemistry approach to synthesize the heterocycle-containing derivatives of fluorinated ripostatin A was developed.

Design, synthesis and biological evaluation of novel triazole-core reversal agents against P-glycoprotein-mediated multidrug resistance

RSC Advances ◽  
2016 ◽  
Vol 6 (31) ◽  
pp. 25819-25828 ◽  
Author(s):  
Bo Zhang ◽  
Tianxiao Zhao ◽  
Jie Zhou ◽  
Qianqian Qiu ◽  
Yuxuan Dai ◽  
...  
Keyword(s):  
Multidrug Resistance ◽  
Click Chemistry ◽  
Biological Evaluation ◽  
Glycoprotein P ◽  
Design Synthesis ◽  
Reversal Agents ◽  
P Glycoprotein ◽  
Synthesis And Biological Evaluation

We designed and synthesized a novel series of P-glycoprotein (P-gp)-mediated multidrug resistance (MDR) inhibitors bearing a triazolphenethyl–tetrahydroisoquinoline scaffold through click chemistry.

Synthesis and biological evaluation of glycal-derived novel tetrahydrofuran 1,2,3-triazoles by ‘click’ chemistry

2010 ◽  
Vol 345 (11) ◽  
pp. 1515-1521 ◽  
Author(s):  
L. Vijaya Raghava Reddy ◽  
P. Venkat Reddy ◽  
Nripendra N. Mishra ◽  
Praveen K. Shukla ◽  
Garima Yadav ◽  
...  
Keyword(s):  
Click Chemistry ◽  
Biological Evaluation ◽  
Synthesis And Biological Evaluation

Synthesis and biological evaluation of tyrosine modified analogues of the α4β7 integrin inhibitor biotin-R8ERY

2012 ◽  
Vol 20 (17) ◽  
pp. 5139-5149 ◽  
Author(s):  
Stefanie Papst ◽  
Anaïs F.M. Noisier ◽  
Margaret A. Brimble ◽  
Yi Yang ◽  
Geoffrey W. Krissansen
Keyword(s):  
Biological Evaluation ◽  
Synthesis And Biological Evaluation ◽  
Integrin Inhibitor
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