Design, synthesis and structure–activity relationship of novel tricyclic benzimidazolone derivatives as potent 18kDa translocator protein (TSPO) ligands

Translocator Protein ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Design, synthesis and structure–activity relationship of simple bis-amides as potent inhibitors of GlyT1

10.1016/j.bmcl.2008.09.005 ◽

2008 ◽

Vol 18 (20) ◽

pp. 5533-5536 ◽

Cited By ~ 11

Author(s):

Synèse Jolidon ◽

Daniela Alberati ◽

Adam Dowle ◽

Holger Fischer ◽

Dominik Hainzl ◽

...

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Design, synthesis, and structure–activity relationship of novel orally efficacious pyrazole/sulfonamide based dihydroquinoline γ-secretase inhibitors

10.1016/j.bmcl.2009.07.092 ◽

2009 ◽

Vol 19 (17) ◽

pp. 4920-4923 ◽

Cited By ~ 32

Author(s):

Anh P. Truong ◽

Danielle L. Aubele ◽

Gary D. Probst ◽

Martin L. Neitzel ◽

Chris M. Semko ◽

...

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationship of Novel Dinucleotide Analogues as Agents Against Herpes and Human Immunodeficiency Viruses.

ChemInform ◽

10.1002/chin.199611278 ◽

2010 ◽

Vol 27 (11) ◽

pp. no-no

Author(s):

G. H. HAKIMELAHI ◽

A. A. MOOSAVI-MOVAHEDI ◽

M. M. SADEGHI ◽

S.-C. TSAY ◽

J. R. HWU

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Human Immunodeficiency Viruses ◽

Design, Synthesis, and Structure–Activity Relationship of New Pyrimidinamine Derivatives Containing an Aryloxy Pyridine Moiety

Journal of Agricultural and Food Chemistry ◽

10.1021/acs.jafc.6b05580 ◽

2017 ◽

Vol 65 (6) ◽

pp. 1272-1280 ◽

Cited By ~ 18

Author(s):

Aiying Guan ◽

Changling Liu ◽

Wei Chen ◽

Fan Yang ◽

Yong Xie ◽

...

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Pyridine Moiety ◽

Structure Activity ◽

Design, synthesis and structure–activity relationship of N-substituted tropane muscarinic acetylcholine receptor antagonists

10.1016/j.bmcl.2012.02.015 ◽

2012 ◽

Vol 22 (9) ◽

pp. 3366-3369 ◽

Cited By ~ 3

Author(s):

Dramane I. Lainé ◽

Hongxing Yan ◽

Haibo Xie ◽

Roderick S. Davis ◽

Jeremy Dufour ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Muscarinic Acetylcholine Receptor ◽

Activity Relationship ◽

Receptor Antagonists ◽

Design Synthesis ◽

Muscarinic Acetylcholine ◽

Structure Activity ◽

Design, synthesis and structure–activity relationship of novel quinoxaline derivatives as cancer chemopreventive agent by inhibition of tyrosine kinase receptor

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2013.07.049 ◽

2013 ◽

Vol 69 ◽

pp. 115-124 ◽

Cited By ~ 21

Author(s):

Shadia A. Galal ◽

Ahmed S. Abdelsamie ◽

Salwa M. Soliman ◽

Jeremie Mortier ◽

Gerhard Wolber ◽

...

Keyword(s):

Tyrosine Kinase ◽

Activity Relationship ◽

Tyrosine Kinase Receptor ◽

Design Synthesis ◽

Chemopreventive Agent ◽

Structure Activity ◽

Quinoxaline Derivatives ◽

Triple reuptake inhibitors: Design, synthesis and structure–activity relationship of benzylpiperidine–tetrazoles

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2017.07.046 ◽

2017 ◽

Vol 25 (20) ◽

pp. 5278-5289 ◽

Cited By ~ 8

Author(s):

Suresh Paudel ◽

Xiao Min ◽

Srijan Acharya ◽

Daulat Bikram Khadka ◽

Goo Yoon ◽

...

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Design, synthesis, and structure–activity relationship of carbamate-tethered aryl propanoic acids as novel PPARα/γ dual agonists

10.1016/j.bmcl.2007.04.057 ◽

2007 ◽

Vol 17 (13) ◽

pp. 3595-3598 ◽

Cited By ~ 13

Author(s):

Nam-Jung Kim ◽

Kwang-Ok Lee ◽

Bon-Woong Koo ◽

Funan Li ◽

Ja-Kyung Yoo ◽

...

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Design, synthesis and structure–activity relationship of novel semi-synthetic flavonoids as antiproliferative agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2014.06.007 ◽

2014 ◽

Vol 82 ◽

pp. 506-520 ◽

Cited By ~ 23

Author(s):

F.A. Ragab ◽

T.A.A. Yahya ◽

M.M. El-Naa ◽

R.K. Arafa

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Antiproliferative Agents ◽

Structure Activity ◽

Design, synthesis and the structure-activity relationship of agonists targeting on the ALDH2 catalytic tunnel

Bioorganic Chemistry ◽

10.1016/j.bioorg.2020.104166 ◽

2020 ◽

Vol 104 ◽

pp. 104166

Author(s):

Ming-Che Cheng ◽

Wei-Chi Lo ◽

Yu-Wen Chang ◽

Shoei-Sheng Lee ◽

Chia-Chuan Chang

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽