Design, synthesis and docking studies on phenoxy-3-piperazin-1-yl-propan-2-ol derivatives as protein tyrosine phosphatase 1B inhibitors

Tyrosine Phosphatase ◽

Docking Studies ◽

Design Synthesis ◽

Design, synthesis, kinetic, molecular dynamics, and hypoglycemic effect characterization of new and potential selective benzimidazole derivatives as Protein Tyrosine Phosphatase 1B inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2021.116418 ◽

2021 ◽

pp. 116418

Author(s):

Mara Ibeth Campos-Almazán ◽

Miguel Flores-Ramos ◽

Alicia Hernández-Campos ◽

Rafael Castillo ◽

Erick Sierra-Campos ◽

...

Keyword(s):

Molecular Dynamics ◽

Tyrosine Phosphatase ◽

Hypoglycemic Effect ◽

Benzimidazole Derivatives ◽

Design Synthesis ◽

Design, synthesis and biological evaluation of novel arylidine-malononitrile derivatives as non-carboxylic inhibitors of protein tyrosine phosphatase 1B

Medicinal Chemistry Research ◽

10.1007/s00044-013-0528-1 ◽

2013 ◽

Vol 22 (11) ◽

pp. 5344-5348 ◽

Cited By ~ 6

Author(s):

Girdhar Singh Deora ◽

Chandrabose Karthikeyan ◽

N. S. Hari Narayana Moorthy ◽

Vandana Rathore ◽

Arun K. Rawat ◽

...

Keyword(s):

Tyrosine Phosphatase ◽

Biological Evaluation ◽

Synthesis And Biological Evaluation

Design Synthesis ◽

Protein Tyrosine ◽

ChemInform Abstract: Design, Synthesis, and Biological Evaluation of Bromophenol Derivatives as Protein Tyrosine Phosphatase 1B Inhibitors.

ChemInform ◽

10.1002/chin.201239087 ◽

2012 ◽

Vol 43 (39) ◽

pp. no-no

Author(s):

Bo Jiang ◽

Dayong Shi ◽

Yongchao Cui ◽

Shuju Guo

Keyword(s):

Tyrosine Phosphatase ◽

Biological Evaluation ◽

Design Synthesis ◽

Protein Tyrosine ◽

Synthesis And Biological Evaluation ◽

Bromophenol Derivatives

Synthesis, Structure-Activity Relationship and Docking Studies of Substituted Aryl Thiazolyl Phenylsulfonamides as Potential Protein Tyrosine Phosphatase 1B Inhibitors

ChemMedChem ◽

10.1002/cmdc.201200197 ◽

2012 ◽

Vol 7 (7) ◽

pp. 1185-1190 ◽

Cited By ~ 8

Author(s):

Kanika Varshney ◽

Swati Gupta ◽

Neha Rahuja ◽

Arun K. Rawat ◽

Nagendra Singh ◽

...

Keyword(s):

Tyrosine Phosphatase ◽

Structure Activity Relationship ◽

Docking Studies ◽

Activity Relationship ◽

Protein Tyrosine ◽

Structure Activity

Validation of Formylchromane Derivatives as Protein Tyrosine Phosphatase 1B Inhibitors by Pharmacophore Modeling, Atom-Based 3D-QSAR and Docking Studies

Chemical Biology & Drug Design ◽

10.1111/cbdd.12135 ◽

2013 ◽

Vol 82 (1) ◽

pp. 71-80 ◽

Cited By ~ 7

Author(s):

Priyanka Malla ◽

Rajnish Kumar ◽

Manoj Kumar

Keyword(s):

Tyrosine Phosphatase ◽

3D Qsar ◽

Pharmacophore Modeling ◽

Docking Studies ◽

ChemInform Abstract: Design, Synthesis and Biological Activity Evaluation of 2-Mercapto-4(3H)-quinazolinone Derivatives as Novel Inhibitors of Protein Tyrosine Phosphatase 1B.

ChemInform ◽

10.1002/chin.201249175 ◽

2012 ◽

Vol 43 (49) ◽

pp. no-no

Author(s):

Hui Li ◽

Jin-Ping Wang ◽

Fan Yang ◽

Ting Liu ◽

Wen-Wei Qiu ◽

...

Keyword(s):

Biological Activity ◽

Tyrosine Phosphatase ◽

Design Synthesis ◽

Protein Tyrosine ◽

Activity Evaluation ◽

Quinazolinone Derivatives

Design, synthesis, and evaluation of bromo-retrochalcone derivatives as protein tyrosine phosphatase 1B inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2011.04.057 ◽

2011 ◽

Vol 21 (12) ◽

pp. 3755-3758 ◽

Cited By ~ 21

Author(s):

Zhiguo Liu ◽

Woojung Lee ◽

Su-Nam Kim ◽

Goo Yoon ◽

Seung Hoon Cheon

Keyword(s):

Tyrosine Phosphatase ◽

Design Synthesis ◽

Design, synthesis, and discovery of stilbene derivatives based on lithospermic acid B as potent protein tyrosine phosphatase 1B inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.06.016 ◽

2007 ◽

Vol 17 (16) ◽

pp. 4481-4486 ◽

Cited By ~ 15

Author(s):

Mankil Jung ◽

Yongnam Lee ◽

Moonsoo Park ◽

Hanjo Kim ◽

Heekyeong Kim ◽

...

Keyword(s):

Tyrosine Phosphatase ◽

Design Synthesis ◽

Protein Tyrosine ◽

Stilbene Derivatives

Design, Synthesis and Biological Activity Evaluation of 2-Mercapto-4(3H)-quinazolinone Derivatives as Novel Inhibitors of Protein Tyrosine Phosphatase 1B

Heterocycles ◽

10.3987/com-12-12477 ◽

2012 ◽

Vol 85 (8) ◽

pp. 1897 ◽

Cited By ~ 3

Author(s):

Jie Tang ◽

Jia Li ◽

Jin-Ping Wang ◽

Fan Yang ◽

Ting Liu ◽

...

Keyword(s):

Biological Activity ◽

Tyrosine Phosphatase ◽

Design Synthesis ◽

Protein Tyrosine ◽

Activity Evaluation ◽

Quinazolinone Derivatives

Design, Synthesis of Lithocholic Acid Mimics and Their Inhibitory Activities against Protein Tyrosine Phosphatase 1B

Chinese Journal of Organic Chemistry ◽

10.6023/cjoc201605018 ◽

2016 ◽

Vol 36 (11) ◽

pp. 2670

Author(s):

Haibing He ◽

Hong Dai ◽

Lixin Gao ◽

Haijun Zhang ◽

Zhenga Zou ◽

...

Keyword(s):

Lithocholic Acid ◽

Tyrosine Phosphatase ◽

Design Synthesis ◽

Protein Tyrosine ◽

Inhibitory Activities