Design, Synthesis and Biological Activity Evaluation of 2-Mercapto-4(3H)-quinazolinone Derivatives as Novel Inhibitors of Protein Tyrosine Phosphatase 1B

Tyrosine Phosphatase ◽

Design Synthesis ◽

Protein Tyrosine ◽

Activity Evaluation ◽

Quinazolinone Derivatives

ChemInform Abstract: Design, Synthesis and Biological Activity Evaluation of 2-Mercapto-4(3H)-quinazolinone Derivatives as Novel Inhibitors of Protein Tyrosine Phosphatase 1B.

ChemInform ◽

10.1002/chin.201249175 ◽

2012 ◽

Vol 43 (49) ◽

pp. no-no

Author(s):

Hui Li ◽

Jin-Ping Wang ◽

Fan Yang ◽

Ting Liu ◽

Wen-Wei Qiu ◽

...

Keyword(s):

Biological Activity ◽

Tyrosine Phosphatase ◽

Design Synthesis ◽

Protein Tyrosine ◽

Activity Evaluation ◽

Quinazolinone Derivatives

Design, Synthesis, Biological Activity and Molecular Dynamics Studies of Specific Protein Tyrosine Phosphatase 1B Inhibitors over SHP-2

International Journal of Molecular Sciences ◽

10.3390/ijms140612661 ◽

2013 ◽

Vol 14 (6) ◽

pp. 12661-12674 ◽

Cited By ~ 5

Author(s):

Su-Xia Sun ◽

Xiao-Bo Li ◽

Wen-Bo Liu ◽

Ying Ma ◽

Run-Ling Wang ◽

...

Keyword(s):

Molecular Dynamics ◽

Biological Activity ◽

Tyrosine Phosphatase ◽

Specific Protein ◽

Design Synthesis ◽

Design, synthesis, kinetic, molecular dynamics, and hypoglycemic effect characterization of new and potential selective benzimidazole derivatives as Protein Tyrosine Phosphatase 1B inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2021.116418 ◽

2021 ◽

pp. 116418

Author(s):

Mara Ibeth Campos-Almazán ◽

Miguel Flores-Ramos ◽

Alicia Hernández-Campos ◽

Rafael Castillo ◽

Erick Sierra-Campos ◽

...

Keyword(s):

Molecular Dynamics ◽

Tyrosine Phosphatase ◽

Hypoglycemic Effect ◽

Benzimidazole Derivatives ◽

Design Synthesis ◽

Design, synthesis and biological evaluation of novel arylidine-malononitrile derivatives as non-carboxylic inhibitors of protein tyrosine phosphatase 1B

Medicinal Chemistry Research ◽

10.1007/s00044-013-0528-1 ◽

2013 ◽

Vol 22 (11) ◽

pp. 5344-5348 ◽

Cited By ~ 6

Author(s):

Girdhar Singh Deora ◽

Chandrabose Karthikeyan ◽

N. S. Hari Narayana Moorthy ◽

Vandana Rathore ◽

Arun K. Rawat ◽

...

Keyword(s):

Tyrosine Phosphatase ◽

Biological Evaluation ◽

Synthesis And Biological Evaluation

Design Synthesis ◽

Protein Tyrosine ◽

ChemInform Abstract: Design, Synthesis, and Biological Evaluation of Bromophenol Derivatives as Protein Tyrosine Phosphatase 1B Inhibitors.

ChemInform ◽

10.1002/chin.201239087 ◽

2012 ◽

Vol 43 (39) ◽

pp. no-no

Author(s):

Bo Jiang ◽

Dayong Shi ◽

Yongchao Cui ◽

Shuju Guo

Keyword(s):

Tyrosine Phosphatase ◽

Biological Evaluation ◽

Design Synthesis ◽

Protein Tyrosine ◽

Synthesis And Biological Evaluation ◽

Bromophenol Derivatives

Design, synthesis and docking studies on phenoxy-3-piperazin-1-yl-propan-2-ol derivatives as protein tyrosine phosphatase 1B inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2010.08.008 ◽

2010 ◽

Vol 20 (19) ◽

pp. 5732-5734 ◽

Cited By ~ 6

Author(s):

Swati Gupta ◽

Gyanendra Pandey ◽

Neha Rahuja ◽

Arvind K. Srivastava ◽

Anil K. Saxena

Keyword(s):

Tyrosine Phosphatase ◽

Docking Studies ◽

Design Synthesis ◽

Design, synthesis, and evaluation of bromo-retrochalcone derivatives as protein tyrosine phosphatase 1B inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2011.04.057 ◽

2011 ◽

Vol 21 (12) ◽

pp. 3755-3758 ◽

Cited By ~ 21

Author(s):

Zhiguo Liu ◽

Woojung Lee ◽

Su-Nam Kim ◽

Goo Yoon ◽

Seung Hoon Cheon

Keyword(s):

Tyrosine Phosphatase ◽

Design Synthesis ◽

Design, synthesis, and discovery of stilbene derivatives based on lithospermic acid B as potent protein tyrosine phosphatase 1B inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.06.016 ◽

2007 ◽

Vol 17 (16) ◽

pp. 4481-4486 ◽

Cited By ~ 15

Author(s):

Mankil Jung ◽

Yongnam Lee ◽

Moonsoo Park ◽

Hanjo Kim ◽

Heekyeong Kim ◽

...

Keyword(s):

Tyrosine Phosphatase ◽

Design Synthesis ◽

Protein Tyrosine ◽

Stilbene Derivatives

Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel Arylaminoacetylhydrazone Derivatives Containing Carbazole Moiety

Chinese Journal of Organic Chemistry ◽

10.6023/cjoc202102046 ◽

2021 ◽

Vol 41 (8) ◽

pp. 3157

Author(s):

Yingjun Li ◽

Ledi Lin ◽

Kun Jin ◽

Lixin Gao ◽

Li Sheng ◽

...

Keyword(s):

Inhibitory Activity ◽

Tyrosine Phosphatase ◽

Protein Tyrosine ◽

Activity Evaluation

Synthesis and biological activity of a novel class of pyridazine analogues as non-competitive reversible inhibitors of protein tyrosine phosphatase 1B (PTP1B)

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(02)00176-1 ◽

2002 ◽

Vol 10 (10) ◽

pp. 3197-3212 ◽

Cited By ~ 44

Author(s):

C Liljebris

Keyword(s):

Biological Activity ◽

Tyrosine Phosphatase ◽

Reversible Inhibitors ◽