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Indole-propionic acid derivatives as potent, S1P3-sparing and EAE efficacious sphingosine-1-phosphate 1 (S1P1) receptor agonists
Bioorganic & Medicinal Chemistry Letters
◽
10.1016/j.bmcl.2012.02.083
◽
2012
◽
Vol 22
(8)
◽
pp. 2794-2797
◽
Cited By ~ 9
Author(s):
Qinghua Meng
◽
Baowei Zhao
◽
Qiongfeng Xu
◽
Xuesong Xu
◽
Guanghui Deng
◽
...
Keyword(s):
Propionic Acid
◽
Receptor Agonists
◽
S1p1 Receptor
◽
Sphingosine 1 Phosphate
Download Full-text
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References
Synthesis of 4(5)-phenylimidazole-based analogues of sphingosine-1-phosphate and FTY720: Discovery of potent S1P1 receptor agonists
Bioorganic & Medicinal Chemistry Letters
◽
10.1016/j.bmcl.2005.05.097
◽
2005
◽
Vol 15
(15)
◽
pp. 3568-3572
◽
Cited By ~ 27
Author(s):
Jeremy J. Clemens
◽
Michael D. Davis
◽
Kevin R. Lynch
◽
Timothy L. Macdonald
Keyword(s):
Receptor Agonists
◽
S1p1 Receptor
◽
Sphingosine 1 Phosphate
Download Full-text
Pyrazole derived from (+)-3-carene; a novel potent, selective scaffold for sphingosine-1-phosphate (S1P1) receptor agonists
Bioorganic & Medicinal Chemistry Letters
◽
10.1016/j.bmcl.2009.11.045
◽
2010
◽
Vol 20
(1)
◽
pp. 35-37
◽
Cited By ~ 5
Author(s):
Frédéric J. Zécri
◽
Rainer Albert
◽
Gregory Landrum
◽
Klaus Hinterding
◽
Nigel G. Cooke
◽
...
Keyword(s):
Receptor Agonists
◽
S1p1 Receptor
◽
Sphingosine 1 Phosphate
Download Full-text
Discovery of Potent 3,5-Diphenyl-1,2,4-oxadiazole Sphingosine-1-phosphate-1 (S1P1) Receptor Agonists with Exceptional Selectivity against S1P2and S1P3
Journal of Medicinal Chemistry
◽
10.1021/jm0503244
◽
2005
◽
Vol 48
(20)
◽
pp. 6169-6173
◽
Cited By ~ 69
Author(s):
Zhen Li
◽
Weirong Chen
◽
Jeffrey J. Hale
◽
Christopher L. Lynch
◽
Sander G. Mills
◽
...
Keyword(s):
Receptor Agonists
◽
S1p1 Receptor
◽
Sphingosine 1 Phosphate
Download Full-text
Faculty Opinions recommendation of Synthesis and biological evaluation of gamma-aminophosphonates as potent, subtype-selective sphingosine 1-phosphate receptor agonists and antagonists.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.1064759.517678
◽
2007
◽
Author(s):
Hugh Rosen
Keyword(s):
Biological Evaluation
◽
Receptor Agonists
◽
Sphingosine 1 Phosphate
◽
Subtype Selective
◽
Synthesis And Biological Evaluation
◽
Receptor Agonists And Antagonists
Download Full-text
Design, synthesis and docking-based 3D-QSAR study of novel 2-substituted 2-aminopropane-1,3-diols as potent and selective agonists of sphingosine-1-phosphate 1 (S1P1) receptor
MedChemComm
◽
10.1039/c3md00079f
◽
2013
◽
Vol 4
(9)
◽
pp. 1267
◽
Cited By ~ 16
Author(s):
Yulin Tian
◽
Jing Jin
◽
Xiaojian Wang
◽
Weijuan Han
◽
Gang Li
◽
...
Keyword(s):
3D Qsar
◽
Qsar Study
◽
Design Synthesis
◽
S1p1 Receptor
◽
Sphingosine 1 Phosphate
◽
Selective Agonists
Download Full-text
Immune Cell Regulation and Cardiovascular Effects of Sphingosine 1-Phosphate Receptor Agonists in Rodents Are Mediated via Distinct Receptor Subtypes
Journal of Pharmacology and Experimental Therapeutics
◽
10.1124/jpet.103.062828
◽
2004
◽
Vol 309
(2)
◽
pp. 758-768
◽
Cited By ~ 253
Author(s):
M. Forrest
◽
S.-Y. Sun
◽
R. Hajdu
◽
J. Bergstrom
◽
D. Card
◽
...
Keyword(s):
Immune Cell
◽
Cardiovascular Effects
◽
Receptor Subtypes
◽
Cell Regulation
◽
Receptor Agonists
◽
Sphingosine 1 Phosphate
Download Full-text
Sphingosine‐1‐Phosphate‐Mediated Endothelial Cell Motility Is Regulated by S1P1 Receptor, Lipid Phosphate Phosphatase‐1 and Sphingosine Kinase 1
The FASEB Journal
◽
10.1096/fasebj.20.4.a483-a
◽
2006
◽
Vol 20
(4)
◽
Author(s):
Irina Gorshkova
◽
Evgeny Berdyshev
◽
Bahman Saatian
◽
Yutong Zhao
◽
Srikanth Pendyala
◽
...
Keyword(s):
Endothelial Cell
◽
Cell Motility
◽
Sphingosine Kinase
◽
Sphingosine Kinase 1
◽
S1p1 Receptor
◽
Sphingosine 1 Phosphate
◽
Lipid Phosphate
Download Full-text
Alignment independent 3D-QSAR studies and molecular dynamics simulations for the identification of potent and selective S1P1 receptor agonists
Journal of Molecular Graphics and Modelling
◽
10.1016/j.jmgm.2019.107459
◽
2020
◽
Vol 94
◽
pp. 107459
Author(s):
Ali Akbar Alizadeh
◽
Behzad Jafari
◽
Siavoush Dastmalchi
Keyword(s):
Molecular Dynamics
◽
Molecular Dynamics Simulations
◽
3D Qsar
◽
Qsar Studies
◽
Receptor Agonists
◽
S1p1 Receptor
◽
Dynamics Simulations
Download Full-text
ChemInform Abstract: Excitatory Amino-Acid Receptor Agonists. Synthesis and Pharmacology of Analogues of 2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid.
ChemInform
◽
10.1002/chin.199739149
◽
2010
◽
Vol 28
(39)
◽
pp. no-no
Author(s):
F. A. SLOEK
◽
B. EBERT
◽
Y. LANG
◽
P. KROGSGAARD-LARSEN
◽
S. M. LENZ
◽
...
Keyword(s):
Amino Acid
◽
Propionic Acid
◽
Excitatory Amino Acid
◽
Excitatory Amino Acid Receptor
◽
Acid Receptor
◽
Receptor Agonists
Download Full-text
39 REGULATION OF SPHINGOSINE 1-PHOSPHATE-INDUCED ENDOTHELIAL CYTOSKELETAL REARRANGEMENT AND BARRIER ENHANCEMENT BY S1P1 RECEPTOR, CAVEOLIN-ENRICHED MICRODOMAINS, PI3 KINASE AND TIAM1/RAC1
Journal of Investigative Medicine
◽
10.2310/6650.2005.00206.38
◽
2005
◽
Vol 53
(2)
◽
pp. S363.3-S363
Author(s):
P. A. Singleton
◽
J. G.N. Garcia
Keyword(s):
Pi3 Kinase
◽
S1p1 Receptor
◽
Cytoskeletal Rearrangement
◽
Sphingosine 1 Phosphate
Download Full-text
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