scholarly journals Mechanistic insights into the activation of ester prodrugs of 666-15

2020 ◽  
Vol 30 (19) ◽  
pp. 127455 ◽  
Author(s):  
Fuchun Xie ◽  
Pedro Martín-Acosta ◽  
Bingbing X. Li ◽  
Xiangshu Xiao
Keyword(s):  
Ester Prodrugs

Effects of steric hindrance and electron density of ester prodrugs on controlling the metabolic activation by human carboxylesterase

2021 ◽  
pp. 100391
Author(s):  
Masato Takahashi ◽  
Ibuki Hirota ◽  
Tomoyuki Nakano ◽  
Tomoyuki Kotani ◽  
Daisuke Takani ◽  
...  
Keyword(s):  
Electron Density ◽  
Steric Hindrance ◽  
Metabolic Activation ◽  
Ester Prodrugs

Synthesis, physicochemical properties and antiviral activities of ester prodrugs of ganciclovir

2005 ◽  
Vol 305 (1-2) ◽  
pp. 75-89 ◽  
Author(s):  
Kunal Patel ◽  
Shrija Trivedi ◽  
Shuanghui Luo ◽  
Xiaodong Zhu ◽  
Dhananjay Pal ◽  
...  
Keyword(s):  
Physicochemical Properties ◽  
Antiviral Activities ◽  
Ester Prodrugs

Enhanced delivery of ketobemidone through porcine buccal mucosa in vitro via more lipophilic ester prodrugs

1992 ◽  
Vol 88 (1-3) ◽  
pp. 237-242 ◽  
Author(s):  
Laila Bach Hansen ◽  
Lona Louring Christrup ◽  
Hans Bundgaard
Keyword(s):  
Buccal Mucosa ◽  
Ester Prodrugs

Influence of chain length on thein vitrohydrolysis of model ester prodrugs by ocular esterases

1982 ◽  
Vol 2 (10) ◽  
pp. 651-656 ◽  
Author(s):  
Shih-Chieh Chang ◽  
Vincent H.L. Lee
Keyword(s):  
Chain Length ◽  
Ester Prodrugs

Skin delivery potency and antitumor activities of temozolomide ester prodrugs

2006 ◽  
Vol 244 (1) ◽  
pp. 42-52 ◽  
Author(s):  
Panassaya Suppasansatorn ◽  
Guocheng Wang ◽  
Barbara R. Conway ◽  
Weidong Wang ◽  
Yongfeng Wang
Keyword(s):  
Antitumor Activities ◽  
Skin Delivery ◽  
Ester Prodrugs

scholarly journals Synthesis of Ester Prodrugs of 9-(S)-[3-Hydroxy-2-(phosphonomethoxy)propyl]-2,6-diaminopurine (HPMPDAP) as Anti-Poxvirus Agents

2010 ◽  
Vol 86 (1) ◽  
pp. A59-A60
Author(s):  
Marcela Krecmerova ◽  
Antonin Holy ◽  
Graciela Andrei ◽  
Karel Pomeisl ◽  
Tomas Tichy ◽  
...  
Keyword(s):  
Ester Prodrugs
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