Design, synthesis and structure-activity relationship study of piperazinone-containing thieno[3,2-d]pyrimidine derivatives as new PI3Kδ inhibitors

Activity Relationship ◽

Pyrimidine Derivatives ◽

Design Synthesis ◽

Structure Activity ◽

Design, synthesis, biological evaluation and structure-activity relationship study of quinazolin-4(3H)-one derivatives as novel USP7 inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2021.113291 ◽

2021 ◽

pp. 113291

Author(s):

Peng Li ◽

Ying Liu ◽

Hua Yang ◽

Hong-Min Liu

Keyword(s):

Biological Evaluation ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Design, Synthesis and Quantitative Structure-Activity Relationship Study of N-(3-Oxo-3,4-dihydro-2H-benzo(1,4)oxazine-7-carbonyl)guanidine Derivatives as Potent Na/H Exchange Inhibitors.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.45.1975 ◽

1997 ◽

Vol 45 (12) ◽

pp. 1975-1983 ◽

Cited By ~ 3

Author(s):

Takeshi YAMAMOTO ◽

Manabu HORI ◽

Ikuo WATANABE ◽

Hisayoshi TSUTSUI ◽

Kengo HARADA ◽

...

Keyword(s):

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Design Synthesis ◽

Guanidine Derivatives ◽

Structure Activity ◽

Design, Synthesis, Biological Screening and Structure Activity Relationship Study of 4, 6-Dimethyl-2-(Substituted) Mercapto-3-(Substituted) Pyridines as Anti Tubercular Agents

American Journal of Infectious Diseases ◽

10.3844/ajidsp.2011.61.66 ◽

2011 ◽

Vol 7 (3) ◽

pp. 61-66 ◽

Cited By ~ 1

Author(s):

Rozita

Keyword(s):

Activity Relationship ◽

Biological Screening ◽

Design Synthesis ◽

Structure Activity ◽

Substituted Pyridines ◽

Design, synthesis and structure–activity relationship (SAR) studies of 2,4-disubstituted pyrimidine derivatives: Dual activity as cholinesterase and Aβ-aggregation inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2011.02.030 ◽

2011 ◽

Vol 19 (7) ◽

pp. 2269-2281 ◽

Cited By ~ 25

Author(s):

Tarek Mohamed ◽

Xiaobei Zhao ◽

Lila K. Habib ◽

Jerry Yang ◽

Praveen P.N. Rao

Keyword(s):

Activity Relationship ◽

Pyrimidine Derivatives ◽

Design Synthesis ◽

Sar Studies ◽

Structure Activity ◽

Aβ Aggregation ◽

Aggregation Inhibitors

Cover Picture: Design, Synthesis, and Structure-Activity Relationship Analysis of Thiazolo[3,2-a ]pyrimidine Derivatives with Anti-inflammatory Activity in Acute Lung Injury (ChemMedChem 13/2017)

ChemMedChem ◽

10.1002/cmdc.201700367 ◽

2017 ◽

Vol 12 (13) ◽

pp. 1013-1013

Author(s):

Lingfeng Chen ◽

Yiyi Jin ◽

Weitao Fu ◽

Siyang Xiao ◽

Chen Feng ◽

...

Keyword(s):

Acute Lung Injury ◽

Lung Injury ◽

Inflammatory Activity ◽

Activity Relationship ◽

Pyrimidine Derivatives ◽

Design Synthesis ◽

Relationship Analysis ◽

Structure Activity ◽

Anti Inflammatory

Design, synthesis and structure-activity relationship study of novel urea compounds as FGFR1 inhibitors to treat metastatic triple-negative breast cancer

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2020.112866 ◽

2021 ◽

Vol 209 ◽

pp. 112866

Author(s):

Md Ashraf-Uz-Zaman ◽

Sadisna Shahi ◽

Racheal Akwii ◽

Md Sanaullah Sajib ◽

Mohammad Jodeiri Farshbaf ◽

...

Keyword(s):

Breast Cancer ◽

Triple Negative Breast Cancer ◽

Triple Negative ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Study ◽

Urea Compounds

Design, synthesis, and structure–activity relationship study of bicyclic piperazine analogs of indole-3-carboxamides as novel cannabinoid CB1 receptor agonists

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2010.10.061 ◽

2010 ◽

Vol 20 (24) ◽

pp. 7327-7330 ◽

Cited By ~ 16

Author(s):

Elizabeth M. Moir ◽

Kazuya Yoshiizumi ◽

Jim Cairns ◽

Phillip Cowley ◽

Morag Ferguson ◽

...

Keyword(s):

Cb1 Receptor ◽

Activity Relationship ◽

Cannabinoid Cb1 Receptor ◽

Design Synthesis ◽

Receptor Agonists ◽

Structure Activity ◽

ChemInform Abstract: Design, Synthesis and Quantitative Structure-Activity Relationship Study of N-(3-Oxo-3,4-dihydro-2H-benzo[1,4]oxazine-7-carbonyl)guanidine Derivatives as Potent Na/H Exchange Inhibitors.

ChemInform ◽

10.1002/chin.199823160 ◽

2010 ◽

Vol 29 (23) ◽

pp. no-no

Author(s):

T. YAMAMOTO ◽

M. HORI ◽

I. WATANABE ◽

H. TSUTSUI ◽

K. HARADA ◽

...

Keyword(s):

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Design Synthesis ◽

Guanidine Derivatives ◽

Structure Activity ◽

Design, Synthesis and Structure-Activity Relationship Study of Coumarin Benzimidazole Hybrid as Potent Antibacterial and Anticancer Agents

ChemistrySelect ◽

10.1002/slct.201600665 ◽

2016 ◽

Vol 1 (15) ◽

pp. 4638-4644 ◽

Cited By ~ 13

Author(s):

Megharaja Holiyachi ◽

Samundeeswari L. Shastri ◽

Bahubali M. Chougala ◽

Lokesh A. Shastri ◽

Shrinivas D. Joshi ◽

...

Keyword(s):

Anticancer Agents ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Design, Synthesis, and Quantitative Structure−Activity Relationship Study of Herbicidal Analogues of Pyrazolo[5,1-d][1,2,3,5]tetrazin-4(3H)ones

Journal of Agricultural and Food Chemistry ◽

10.1021/jf063271n ◽

2007 ◽

Vol 55 (4) ◽

pp. 1364-1369 ◽

Cited By ~ 14

Author(s):

You-quan Zhu ◽

Chao Wu ◽

Hua-bin Li ◽

Xiao-mao Zou ◽

Xue-kai Si ◽

...

Keyword(s):

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Design Synthesis ◽

Structure Activity ◽