Biophysical and pharmacological characterization of α6-containing nicotinic acetylcholine receptors expressed in HEK293 cells

Acetylcholine Receptors ◽

Hek293 Cells ◽

Pharmacological Characterization of Natural Tobacco Alkaloids in the Presence of Positive Allosteric Modulators Against Human α4β2 and α7 Nicotinic Acetylcholine Receptors

Biophysical Journal ◽

10.1016/j.bpj.2019.11.790 ◽

2020 ◽

Vol 118 (3) ◽

pp. 119a

Author(s):

Omar Alijevic ◽

Damian Mc Hugh ◽

Anatoly Mazurov ◽

Julia Hoeng ◽

Manuel Peitsch

Keyword(s):

Acetylcholine Receptors ◽

Allosteric Modulators ◽

Nicotinic Acetylcholine ◽

Α7 Nicotinic Acetylcholine Receptors ◽

Tobacco Alkaloids ◽

Positive Allosteric Modulators

Pharmacological characterization of [125I]CHIBA-1006 binding, a new radioligand for α7 nicotinic acetylcholine receptors, to rat brain membranes

Brain Research ◽

10.1016/j.brainres.2010.08.095 ◽

2010 ◽

Vol 1360 ◽

pp. 130-137 ◽

Cited By ~ 8

Author(s):

Jin Wu ◽

Jun Toyohara ◽

Yuko Tanibuchi ◽

Yuko Fujita ◽

Jichun Zhang ◽

...

Keyword(s):

Rat Brain ◽

Acetylcholine Receptors ◽

Α7 Nicotinic Acetylcholine Receptors

Nicotinic Acetylcholine ◽

Brain Membranes ◽

Rat Brain Membranes ◽

Characterization of the recombinant human neuronal nicotinic acetylcholine receptors α3β2 and α4β2 stably expressed in HEK293 cells

Neuropharmacology ◽

10.1016/s0028-3908(00)00134-9 ◽

2000 ◽

Vol 39 (13) ◽

pp. 2543-2560 ◽

Cited By ~ 57

Author(s):

Laura E. Chavez-Noriega ◽

Alison Gillespie ◽

Kenneth A. Stauderman ◽

James H. Crona ◽

Brian O'Neil Claeps ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Hek293 Cells ◽

Neuronal Nicotinic Acetylcholine Receptors ◽

Synthesis and pharmacological characterization of bivalent ligands of epibatidine at neuronal nicotinic acetylcholine receptors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2003.10.071 ◽

2004 ◽

Vol 14 (8) ◽

pp. 1855-1858 ◽

Cited By ~ 9

Author(s):

Zhi-Liang Wei ◽

Yingxian Xiao ◽

Kenneth J Kellar ◽

Alan P Kozikowski

Keyword(s):

Acetylcholine Receptors ◽

Neuronal Nicotinic Acetylcholine Receptors ◽

Bivalent Ligands ◽

Identification and pharmacological characterization of 3,6-diazabicyclo[3.1.1]heptane-3-carboxamides as novel ligands for the α4β2 and α6/α3β2β3 nicotinic acetylcholine receptors (nAChRs)

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2014.08.019 ◽

2014 ◽

Vol 86 ◽

pp. 60-74 ◽

Cited By ~ 4

Author(s):

Jon-Paul Strachan ◽

David C. Kombo ◽

Anatoly Mazurov ◽

Ronald Heemstra ◽

Balwinder S. Bhatti ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Synthesis and Pharmacological Characterization of Bivalent Ligands of Epibatidine at Neuronal Nicotinic Acetylcholine Receptors

ChemInform ◽

10.1002/chin.200430239 ◽

2004 ◽

Vol 35 (30) ◽

Author(s):

Zhi-Liang Wei ◽

Yingxian Xiao ◽

Kenneth J. Kellar ◽

Alan P. Kozikowski

Keyword(s):

Acetylcholine Receptors ◽

Neuronal Nicotinic Acetylcholine Receptors ◽

Bivalent Ligands ◽

Design, Synthesis, and Pharmacological Characterization of Novel Spirocyclic Quinuclidinyl-Δ2-Isoxazoline Derivatives as Potent and Selective Agonists of α7 Nicotinic Acetylcholine Receptors

ChemMedChem ◽

10.1002/cmdc.201000514 ◽

2011 ◽

Vol 6 (5) ◽

pp. 889-903 ◽

Cited By ~ 22

Author(s):

Clelia Dallanoce ◽

Pietro Magrone ◽

Carlo Matera ◽

Fabio Frigerio ◽

Giovanni Grazioso ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

Design Synthesis ◽

Α7 Nicotinic Acetylcholine Receptors ◽

Selective Agonists

Faculty Opinions recommendation of Molecular characterization of off-target activities of telithromycin: a potential role for nicotinic acetylcholine receptors.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.7869956.8218054 ◽

2011 ◽

Author(s):

David Newman

Keyword(s):

Molecular Characterization ◽

Acetylcholine Receptors ◽

Potential Role ◽

Melatonin modulation of presynaptic nicotinic acetylcholine receptors located on short noradrenergic neurons of the rat vas deferens: a pharmacological characterization

Brazilian Journal of Medical and Biological Research ◽

10.1590/s0100-879x1999000800010 ◽

1999 ◽

Vol 32 (8) ◽

pp. 999-1006 ◽

Cited By ~ 12

Author(s):

W.M. Zago ◽

R.P. Markus

Keyword(s):

Acetylcholine Receptors ◽

Vas Deferens ◽

Rat Vas Deferens ◽

Noradrenergic Neurons ◽

Pharmacological and structural characterization of the interaction of snake toxins with nicotinic acetylcholine receptors

Cholinergic Mechanisms ◽

10.3109/9780203493878-5 ◽

2004 ◽

pp. 27-31

Author(s):

D Servent ◽

C Fruchart-Gaillard ◽

A Ménez

Keyword(s):

Structural Characterization ◽

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

Snake Toxins