Indanesulfonamides as carbonic anhydrase inhibitors and anticonvulsant agents: Structure–activity relationship and pharmacological evaluation

Anne Thiry; Stéphanie Rolin; Daniela Vullo; Aurélie Frankart; Andrea Scozzafava; Jean-Michel Dogné; Johan Wouters; Claudiu T. Supuran; Bernard Masereel

doi:10.1016/j.ejmech.2008.02.018

Indanesulfonamides as carbonic anhydrase inhibitors and anticonvulsant agents: Structure–activity relationship and pharmacological evaluation

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2008.02.018 ◽

2008 ◽

Vol 43 (12) ◽

pp. 2853-2860 ◽

Cited By ~ 16

Author(s):

Anne Thiry ◽

Stéphanie Rolin ◽

Daniela Vullo ◽

Aurélie Frankart ◽

Andrea Scozzafava ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Carbonic Anhydrase Inhibitors ◽

Anticonvulsant Agents ◽

Pharmacological Evaluation ◽

Structure Activity

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Exploring structure-activity relationship of S-substituted 2-mercaptoquinazolin-4(3H)-one including 4-ethylbenzenesulfonamides as human carbonic anhydrase inhibitors

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756366.2020.1722121 ◽

2020 ◽

Vol 35 (1) ◽

pp. 598-609 ◽

Cited By ~ 4

Author(s):

Adel S. El-Azab ◽

Alaa A.-M. Abdel-Aziz ◽

Hany E. A. Ahmed ◽

Sivia Bua ◽

Alessio Nocentini ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity ◽

Human Carbonic Anhydrase ◽

Relationship Of

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Development of Quantitative Structure−Activity Relationship and Classification Models for a Set of Carbonic Anhydrase Inhibitors

Journal of Chemical Information and Computer Sciences ◽

10.1021/ci0100696 ◽

2001 ◽

Vol 42 (1) ◽

pp. 94-102 ◽

Cited By ~ 27

Author(s):

Brian E. Mattioni ◽

Peter C. Jurs

Keyword(s):

Carbonic Anhydrase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Classification Models ◽

Quantitative Structure ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity

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A quantitative structure–activity relationship study on some aromatic/heterocyclic sulfonamides and their charged derivatives acting as carbonic anhydrase inhibitors

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756360500067439 ◽

2005 ◽

Vol 20 (3) ◽

pp. 251-259 ◽

Cited By ~ 5

Author(s):

S. P. Gupta ◽

S. Kumaran

Keyword(s):

Carbonic Anhydrase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity ◽

Relationship Study ◽

Aromatic Heterocyclic

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Carbonic anhydrase inhibitors. Part 24. A quantitative structure-activity relationship study of positively charged sulfonamide inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/0223-5234(96)88286-9 ◽

1995 ◽

Vol 30 (9) ◽

pp. 687-696 ◽

Cited By ~ 47

Author(s):

CT Supuran ◽

BW Clare

Keyword(s):

Carbonic Anhydrase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity ◽

Relationship Study ◽

Positively Charged

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ChemInform Abstract: Development of Quantitative Structure-Activity Relationship and Classification Models for a Set of Carbonic Anhydrase Inhibitors.

ChemInform ◽

10.1002/chin.200221211 ◽

2010 ◽

Vol 33 (21) ◽

pp. no-no

Author(s):

Brian E. Mattioni ◽

Peter C. Jurs

Keyword(s):

Carbonic Anhydrase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Classification Models ◽

Quantitative Structure ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity

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Biological Activities of Drugs. VI. Structure-Activity Relationship of Sulfonamide Carbonic Anhydrase Inhibitors. (1)

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.17.1010 ◽

1969 ◽

Vol 17 (5) ◽

pp. 1010-1018 ◽

Cited By ~ 47

Author(s):

NOBUHARU KAKEYA ◽

MASARU AOKI ◽

AKIRA KAMADA ◽

NOBORU YATA

Keyword(s):

Carbonic Anhydrase ◽

Biological Activities ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity ◽

Relationship Of

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Biological Activities of Drugs. VIII. Structure-Activity Relationship of Sulfonamide Carbonic Anhydrase Inhibitors. (3)

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.17.2558 ◽

1969 ◽

Vol 17 (12) ◽

pp. 2558-2564 ◽

Cited By ~ 24

Author(s):

NOBUHARU KAKEYA ◽

NOBORU YATA ◽

AKIRA KAMADA ◽

MASARU AOKI

Keyword(s):

Carbonic Anhydrase ◽

Biological Activities ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity ◽

Relationship Of

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Structure–Activity Relationship Studies of Acetazolamide-Based Carbonic Anhydrase Inhibitors with Activity against Neisseria gonorrhoeae

ACS Infectious Diseases ◽

10.1021/acsinfecdis.1c00055 ◽

2021 ◽

Author(s):

Chad S. Hewitt ◽

Nader S. Abutaleb ◽

Ahmed E. M. Elhassanny ◽

Alessio Nocentini ◽

Xufeng Cao ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Neisseria Gonorrhoeae ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity

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Development of Quantitative Structure-Activity Relationship for a Set of Carbonic Anhydrase Inhibitors: Use of Quantum and Chemical Descriptors

Letters in Drug Design & Discovery ◽

10.2174/157018006778341138 ◽

2006 ◽

Vol 3 (9) ◽

pp. 622-635 ◽

Cited By ~ 4

Author(s):

Padmakar Khadikar ◽

Omar Deeb ◽

Amal Jaber ◽

Jyoti Singh ◽

Vijay Agrawal ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity ◽

Chemical Descriptors

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Biological Activities of Drugs. IX. Structure-Activity Relationship of Sulfonamide Carbonic Anhydrase Inhibitors.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.18.191 ◽

1970 ◽

Vol 18 (1) ◽

pp. 191-194 ◽

Cited By ~ 16

Author(s):

NOBUHARU KAKEYA ◽

NOBORU YATA ◽

AKIRA KAMADA ◽

MASARU AOKI

Keyword(s):

Carbonic Anhydrase ◽

Biological Activities ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity ◽

Relationship Of

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