carbonic anhydrase inhibitors Recently Published Documents

Antiproliferative effects of sulphonamide carbonic anhydrase inhibitors C18, SLC-0111 and acetazolamide on bladder, glioblastoma and pancreatic cancer cell lines

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756366.2021.2004592 ◽

2021 ◽

Vol 37 (1) ◽

pp. 280-286

Author(s):

Silvia Mussi ◽

Sara Rezzola ◽

Paola Chiodelli ◽

Alessio Nocentini ◽

Claudiu T. Supuran ◽

...

Keyword(s):

Pancreatic Cancer ◽

Carbonic Anhydrase ◽

Cell Lines ◽

Cancer Cell ◽

Pancreatic Cancer Cell ◽

Cancer Cell Lines ◽

Antiproliferative Effects

Carbonic anhydrase inhibitors: an update on experimental agents for the treatment and imaging of hypoxic tumors

Expert Opinion on Investigational Drugs ◽

10.1080/13543784.2021.2014813 ◽

2021 ◽

Author(s):

Claudiu T. Supuran

Keyword(s):

Carbonic Anhydrase ◽

1,5‐Benzodiazepines as a platform for the design of carbonic anhydrase inhibitors

Archiv der Pharmazie ◽

10.1002/ardp.202100405 ◽

2021 ◽

Author(s):

Chiraz Ismail ◽

Alessio Nocentini ◽

Claudiu T. Supuran ◽

Jean‐Yves Winum ◽

Rafik Gharbi

Keyword(s):

Carbonic Anhydrase ◽

2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and Antiglaucoma activity

10.1016/j.ejmech.2021.114026 ◽

2021 ◽

pp. 114026

Author(s):

Niccolò Chiaramonte ◽

Andrea Angeli ◽

Silvia Sgambellone ◽

Alessandro Bonardi ◽

Alessio Nocentini ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Enzyme Inhibition ◽

Computational Studies ◽

Piperazine Derivatives ◽

Human Carbonic Anhydrase ◽

Hydroxyethyl Piperazine

Natural inspired piperine-based sulfonamides and carboxylic acids as carbonic anhydrase inhibitors: Design, synthesis and biological evaluation

10.1016/j.ejmech.2021.113800 ◽

2021 ◽

Vol 225 ◽

pp. 113800

Author(s):

Diaaeldin M. Elimam ◽

Abdullah A. Elgazar ◽

Alessandro Bonardi ◽

Mohamed Abdelfadil ◽

Alessio Nocentini ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Carboxylic Acids ◽

Biological Evaluation ◽

Synthesis And Biological Evaluation

Design Synthesis ◽

Synthesis of human carbonic anhydrase inhibitors with structure of 4-substituted pyridine-3-sulfonamide

10.3390/ecmc2021-11446 ◽

2021 ◽

Author(s):

Krzysztof Szafrański ◽

Jarosław Sławiński ◽

Anna Kawiak

Keyword(s):

Carbonic Anhydrase ◽

Human Carbonic Anhydrase

Natural inspired ligustrazine-based SLC-0111 analogues as novel carbonic anhydrase inhibitors

10.1016/j.ejmech.2021.114008 ◽

2021 ◽

pp. 114008

Author(s):

Diaaeldin M. Elimam ◽

Wagdy M. Eldehna ◽

Rofaida Salem ◽

Alessandro Bonardi ◽

Alessio Nocentini ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Synthesis, biological evaluation, and in silico studies of potential activators of apoptosis and carbonic anhydrase inhibitors on isatin-5-sulfonamide scaffold

10.1016/j.ejmech.2021.113997 ◽

2021 ◽

pp. 113997

Author(s):

Stepan K. Krymov ◽

Alexander M. Scherbakov ◽

Diana I. Salnikova ◽

Danila V. Sorokin ◽

Lyubov G. Dezhenkova ◽

...

Keyword(s):

Carbonic Anhydrase ◽

In Silico ◽

Biological Evaluation ◽

In Silico Studies

Application of the dual-tail approach for the design and synthesis of novel Thiopyrimidine–Benzenesulfonamide hybrids as selective carbonic anhydrase inhibitors

10.1016/j.ejmech.2021.114004 ◽

2021 ◽

pp. 114004

Author(s):

Heba T. Abdel-Mohsen ◽

Ahmed M. El Kerdawy ◽

Mohamed A. Omar ◽

Andrea Petreni ◽

Rasha M. Allam ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Design And Synthesis