Synthesis, structure-activity relationships and biological evaluation of 7-phenyl-pyrroloquinolinone 3-amide derivatives as potent antimitotic agents

Structure Activity ◽

Amide Derivatives

Synthesis and structure activity relationships of glycine amide derivatives as novel Vascular Adhesion Protein-1 inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2016.10.025 ◽

2017 ◽

Vol 25 (1) ◽

pp. 187-201 ◽

Cited By ~ 6

Author(s):

Susumu Yamaki ◽

Daisuke Suzuki ◽

Jiro Fujiyasu ◽

Masahiro Neya ◽

Akira Nagashima ◽

...

Keyword(s):

Adhesion Protein ◽

Structure Activity ◽

Amide Derivatives ◽

Vascular Adhesion ◽

Vascular Adhesion Protein 1

Synthesis and Biological Evaluation of 14-Alkoxymorphinans. 18.1N-Substituted 14-Phenylpropyloxymorphinan-6-ones with Unanticipated Agonist Properties: Extending the Scope of Common Structure−Activity Relationships

Journal of Medicinal Chemistry ◽

10.1021/jm021118o ◽

2003 ◽

Vol 46 (9) ◽

pp. 1758-1763 ◽

Cited By ~ 23

Author(s):

Elisabeth Greiner ◽

Mariana Spetea ◽

Roland Krassnig ◽

Falko Schüllner ◽

Mario Aceto ◽

...

Keyword(s):

Biological Evaluation ◽

Synthesis And Biological Evaluation

Common Structure ◽

Structure Activity ◽

125 Synthesis, biological evaluation and structure activity relationships of a novel servies of aromatic hydroxamic acids as potent HDAC inhibitors

European Journal of Cancer Supplements ◽

10.1016/s1359-6349(04)80133-2 ◽

2004 ◽

Vol 2 (8) ◽

pp. 40-41

Author(s):

K. Van Emelen ◽

J. Arts ◽

P. Angibaud ◽

H. De Winter ◽

S. Van Brandt ◽

...

Keyword(s):

Hdac Inhibitors ◽

Hydroxamic Acids ◽

Biological Evaluation ◽

Biological Evaluation, Structure−Activity Relationships, and Three-Dimensional Quantitative Structure−Activity Relationship Studies of Dihydro-β-agarofuran Sesquiterpenes as Modulators of P-Glycoprotein-Dependent Multidrug Resistance

Journal of Medicinal Chemistry ◽

10.1021/jm070290v ◽

2007 ◽

Vol 50 (20) ◽

pp. 4808-4817 ◽

Cited By ~ 30

Author(s):

Carolina P. Reyes ◽

Francisco Muñoz-Martínez ◽

Ivan R. Torrecillas ◽

Cristina R. Mendoza ◽

Francisco Gamarro ◽

...

Keyword(s):

Multidrug Resistance ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Biological Evaluation ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

P Glycoprotein

Selective and effective anticancer agents: Synthesis, biological evaluation and structure-activity relationships of novel carbazole derivatives

Bioorganic Chemistry ◽

10.1016/j.bioorg.2021.104991 ◽

2021 ◽

pp. 104991

Author(s):

Wenbo Huang ◽

Zilin Gao ◽

Zhigang Zhang ◽

Wei Fang ◽

Zuoqian Wang ◽

...

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Carbazole Derivatives ◽

ChemInform Abstract: Indole Amide Derivatives: Synthesis, Structure-Activity Relationships, and Molecular Modeling Studies of a New Series of Histamine H1-Receptor Antagonists.

ChemInform ◽

10.1002/chin.199929124 ◽

2010 ◽

Vol 30 (29) ◽

pp. no-no

Author(s):

Sandra Battaglia ◽

Enrico Boldrini ◽

Federico Da Settimo ◽

Giulio Dondio ◽

Concettina La Motta ◽

...

Keyword(s):

Molecular Modeling ◽

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor ◽

Structure Activity ◽

Modeling Studies ◽

Amide Derivatives ◽

Molecular Modeling Studies

Synthesis, Biological Evaluation, and Structure−Activity Relationships of 3-Acylindole-2-carboxylic Acids as Inhibitors of the Cytosolic Phospholipase A2

Journal of Medicinal Chemistry ◽

10.1021/jm960863w ◽

1997 ◽

Vol 40 (17) ◽

pp. 2694-2705 ◽

Cited By ~ 20

Author(s):

Matthias Lehr

Keyword(s):

Phospholipase A2 ◽

Carboxylic Acids ◽

Biological Evaluation ◽

Cytosolic Phospholipase A2 ◽

Cytosolic Phospholipase ◽

Taxol structure-activity relationships: synthesis and biological evaluation of 10-deoxytaxol

The Journal of Organic Chemistry ◽

10.1021/jo00063a001 ◽

1993 ◽

Vol 58 (11) ◽

pp. 2927-2928 ◽

Cited By ~ 32

Author(s):

Shu Hui Chen ◽

Craig Fairchild ◽

Stephen W. Mamber ◽

Vittorio Farina

Keyword(s):

Biological Evaluation ◽

Synthesis And Biological Evaluation

Structure Activity ◽

Scaffold hopping, synthesis and structure–activity relationships of 5,6-diaryl-pyrazine-2-amide derivatives: A novel series of CB1 receptor antagonists

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2007.03.075 ◽

2007 ◽

Vol 15 (12) ◽

pp. 4077-4084 ◽

Cited By ~ 47

Author(s):

Jonas Boström ◽

Kristina Berggren ◽

Thomas Elebring ◽

Peter J. Greasley ◽

Michael Wilstermann

Keyword(s):

Cb1 Receptor ◽

Scaffold Hopping ◽

Receptor Antagonists ◽

Structure Activity ◽

Amide Derivatives ◽

Cb1 Receptor Antagonists

New platinum(II) complexes conjugated at position 7α of 17β-acetyl-testosterone as new combi-molecules against prostate cancer: Design, synthesis, structure–activity relationships and biological evaluation

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2013.08.011 ◽

2013 ◽

Vol 68 ◽

pp. 433-443 ◽

Cited By ~ 20

Author(s):

Sébastien Fortin ◽

Kevin Brasseur ◽

Nathalie Morin ◽

Éric Asselin ◽

Gervais Bérubé

Keyword(s):

Prostate Cancer ◽

Biological Evaluation ◽

Design Synthesis ◽