Novel mouse GABA uptake inhibitors with enhanced inhibitory activity toward mGAT3/4 and their effect on pain threshold in mice

2020 ◽  
Vol 188 ◽  
pp. 111920 ◽  
Author(s):  
Paula Zaręba ◽  
Beata Gryzło ◽  
Katarzyna Malawska ◽  
Kinga Sałat ◽  
Georg C. Höfner ◽  
...  
Keyword(s):  
Inhibitory Activity ◽  
Pain Threshold ◽  
Gaba Uptake ◽  
Uptake Inhibitors ◽  
Gaba Uptake Inhibitors

Synthesis and Biochemical Studies of Spirocyclic Amino Acid Esters, Part 3 Activity of 2-Azaspiro[4.5]decane-6-carboxylates as GABA-Uptake Inhibitors

1996 ◽  
Vol 329 (3) ◽  
pp. 149-154 ◽  
Author(s):  
Wilhelm Fleischhacker ◽  
Silvia Lauritz ◽  
Ernst Urban ◽  
Peter Baumann ◽  
Helmut Bittiger
Keyword(s):  
Amino Acid ◽  
Gaba Uptake ◽  
Amino Acid Esters ◽  
Uptake Inhibitors ◽  
Biochemical Studies ◽  
Gaba Uptake Inhibitors ◽  
Acid Esters

GABA-A agonists and GABA uptake inhibitors: Structure-activity relationships

1990 ◽  
Vol 21 (3) ◽  
pp. 169-188 ◽  
Author(s):  
Erik Falch ◽  
Orla M. Larsson ◽  
Arne Schousboe ◽  
Povl Krogsgaard-Larsen
Keyword(s):  
Gaba Uptake ◽  
Gaba A ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Uptake Inhibitors ◽  
Gaba Uptake Inhibitors
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