Preparation and in vitro/in vivo evaluation of nano-sized crystals for dissolution rate enhancement of ucb-35440-3, a highly dosed poorly water-soluble weak base

Solubility and Dissolution Rate Enhancement of Poorly Water Soluble Telmisartan by Melt Granulation Technique Using Soluplus and PEG8000 as Carrier

International Journal of Pharmaceutical Research ◽

10.31838/ijpr/2020.sp1.194 ◽

2020 ◽

Vol 12 (sp1) ◽

Keyword(s):

Dissolution Rate ◽

Water Soluble ◽

Rate Enhancement ◽

Poorly Water Soluble ◽

Melt Granulation

Microcrystals for dissolution rate enhancement of poorly water-soluble drugs

International Journal of Pharmaceutics ◽

10.1016/s0378-5173(03)00005-x ◽

2003 ◽

Vol 254 (2) ◽

pp. 137-145 ◽

Cited By ~ 137

Author(s):

Norbert Rasenack ◽

Helge Hartenhauer ◽

Bernd W Müller

Keyword(s):

Dissolution Rate ◽

Water Soluble ◽

Rate Enhancement ◽

Water Soluble Drugs ◽

Eudragit-Based Nanosuspension of Poorly Water-Soluble Drug: Formulation and In Vitro–In Vivo Evaluation

AAPS PharmSciTech ◽

10.1208/s12249-012-9833-0 ◽

2012 ◽

Vol 13 (4) ◽

pp. 1031-1044 ◽

Cited By ~ 34

Author(s):

Sarita Kumari Yadav ◽

Shivani Mishra ◽

Brahmeshwar Mishra

Keyword(s):

Drug Formulation ◽

Water Soluble ◽

In Vivo Evaluation ◽

Water Soluble Drug ◽

Poorly Water Soluble ◽

Poorly Water Soluble Drug

Practical Method for Preparing Nanosuspension Formulations for Toxicology Studies in the Discovery Stage: Formulation Optimization and in Vitro/in Vivo Evaluation of Nanosized Poorly Water-Soluble Compounds

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.c14-00232 ◽

2014 ◽

Vol 62 (11) ◽

pp. 1073-1082 ◽

Cited By ~ 11

Author(s):

Takao Komasaka ◽

Hisako Fujimura ◽

Toshiaki Tagawa ◽

Akio Sugiyama ◽

Yasunori Kitano

Keyword(s):

Practical Method ◽

Water Soluble ◽

In Vivo Evaluation ◽

Formulation Optimization ◽

Poorly Water Soluble ◽

Discovery Stage

Dissolution rate enhancement of the poorly water-soluble drug Tibolone using PVP, SiO2, and their nanocomposites as appropriate drug carriers

Drug Development and Industrial Pharmacy ◽

10.1080/03639040902787653 ◽

2009 ◽

Vol 35 (9) ◽

pp. 1128-1138 ◽

Cited By ~ 9

Author(s):

Sofia Papadimitriou ◽

Dimitrios Bikiaris

Keyword(s):

Dissolution Rate ◽

Drug Carriers ◽

Water Soluble ◽

Rate Enhancement ◽

Water Soluble Drug ◽

Poorly Water Soluble ◽

Poorly Water Soluble Drug

Solid dispersions, Part I: recent evolutions and future opportunities in manufacturing methods for dissolution rate enhancement of poorly water-soluble drugs

Expert Opinion on Drug Delivery ◽

10.1517/17425247.2011.618181 ◽

2011 ◽

Vol 8 (11) ◽

pp. 1501-1519 ◽

Cited By ~ 113

Author(s):

Dimitrios N Bikiaris

Keyword(s):

Dissolution Rate ◽

Solid Dispersions ◽

Water Soluble ◽

Rate Enhancement ◽

Water Soluble Drugs ◽

Poorly Water Soluble ◽

Manufacturing Methods

An investigation into the mechanism of dissolution rate enhancement of poorly water-soluble drugs from spray chilled gelucire 50/13 microspheres

Journal of Pharmaceutical Sciences ◽

10.1002/jps.21832 ◽

2010 ◽

Vol 99 (1) ◽

pp. 262-274 ◽

Cited By ~ 35

Author(s):

Sheng Qi ◽

Delphine Marchaud ◽

Duncan Q.M. Craig

Keyword(s):

Dissolution Rate ◽

Water Soluble ◽

Rate Enhancement ◽

Water Soluble Drugs ◽

In vitro and in vivo evaluation of porous lactose/mannitol carriers for solubility enhancement of poorly water-soluble drugs

Drying Technology ◽

10.1080/07373937.2019.1596948 ◽

2019 ◽

Vol 38 (7) ◽

pp. 889-902

Author(s):

Niyanhan Jiang ◽

Shanshan Wang ◽

Zeneng Cheng ◽

Wenjie Liu

Keyword(s):

Solubility Enhancement ◽

Water Soluble ◽

In Vivo Evaluation ◽

Water Soluble Drugs ◽

Study on Dissolution Rate Enhancement of Poorly Water Soluble Drug: Contributions of Solubility Enhancement and Relatively Low Micelle Diffusivity

Journal of Dispersion Science and Technology ◽

10.1080/01932690600859374 ◽

2006 ◽

Vol 27 (8) ◽

pp. 1141-1150 ◽

Cited By ~ 8

Author(s):

Vishal Y. Joshi ◽

Manohar R. Sawant

Keyword(s):

Dissolution Rate ◽

Solubility Enhancement ◽

Water Soluble ◽

Rate Enhancement ◽

Water Soluble Drug ◽

Poorly Water Soluble ◽

Poorly Water Soluble Drug

Solid dispersions, Part II: new strategies in manufacturing methods for dissolution rate enhancement of poorly water-soluble drugs

Expert Opinion on Drug Delivery ◽

10.1517/17425247.2011.618182 ◽

2011 ◽

Vol 8 (12) ◽

pp. 1663-1680 ◽

Cited By ~ 47

Author(s):

Dimitrios N Bikiaris

Keyword(s):

Dissolution Rate ◽

Solid Dispersions ◽

Water Soluble ◽

Rate Enhancement ◽

Water Soluble Drugs ◽

Poorly Water Soluble ◽

Manufacturing Methods ◽

New Strategies