Structure–activity relationship study of some inhibitors of HIV-1 integrase

Journal of Molecular Structure THEOCHEM ◽

10.1016/s0166-1280(98)00558-2 ◽

1999 ◽

Vol 464 (1-3) ◽

pp. 267-272 ◽

Author(s):

M. Cyrillo ◽

D.S. Galvão

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study ◽

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Quantitative Structure-Activity Relationship Study on the Anti-HIV-1 Activity of Novel 6-Naphthylthio HEPT Analogs

Chemical Biology & Drug Design ◽

10.1111/j.1747-0285.2009.00843.x ◽

2009 ◽

Vol 74 (2) ◽

pp. 165-172 ◽

Author(s):

Siavash Riahi ◽

Eslam Pourbasheer ◽

Rassoul Dinarvand ◽

Mohammad Reza Ganjali ◽

Parviz Norouzi

Keyword(s):

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Study ◽

Anti Hiv ◽

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A facile one-pot multi-component synthesis of novel adamantine substituted imidazo[1,2-a]pyridine derivatives: identification and structure–activity relationship study of their anti-HIV-1 activity

RSC Advances ◽

10.1039/c6ra17656a ◽

2016 ◽

Vol 6 (97) ◽

pp. 95177-95188 ◽

Author(s):

Tazeem Tazeem ◽

Xin Han ◽

Qingjun Zhou ◽

Jingchen Wei ◽

Po Tien ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Pyridine Derivatives ◽

One Pot ◽

Structure Activity ◽

Relationship Study ◽

Anti Hiv ◽

A series of adamantine substituted imidazo[1,2-a]pyridine derivatives were developed through a one-pot multi-component Groebke–Blackburn–Bienaymé reaction, among them several compounds were identified to be the potent inhibitors against HIV-1 cells.

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Anti-HIV-1 activity and structure–activity-relationship study of a fucosylated glycosaminoglycan from an echinoderm by targeting the conserved CD4 induced epitope

Biochimica et Biophysica Acta (BBA) - General Subjects ◽

10.1016/j.bbagen.2013.06.003 ◽

2013 ◽

Vol 1830 (10) ◽

pp. 4681-4691 ◽

Author(s):

Wu Lian ◽

Mingyi Wu ◽

Ning Huang ◽

Na Gao ◽

Chuang Xiao ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study ◽

Anti Hiv ◽

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Quantitative Structure-Activity Relationship Study of 2-arylsulfonyl-6-substituted Benzonitriles as Non-nucleoside Reverse Transcriptase Inhibitors of HIV-1

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/1475636021000010932 ◽

2002 ◽

Vol 17 (4) ◽

pp. 219-225 ◽

Author(s):

B.K. Sharma ◽

Rajendra Kumar ◽

P. Singh

Keyword(s):

Reverse Transcriptase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Reverse Transcriptase Inhibitors ◽

Nucleoside Reverse Transcriptase Inhibitors ◽

Structure Activity ◽

Relationship Study ◽

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A quantitative structure-activity relationship study for structurally diverse HIV-1 protease inhibitors: contribution of conformational flexibility to inhibitory activity

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756360600810233 ◽

2006 ◽

Vol 21 (5) ◽

pp. 609-615

Author(s):

Keigo Gohda

Keyword(s):

Protease Inhibitors ◽

Inhibitory Activity ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Conformational Flexibility ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Study ◽

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Parallel one-pot synthesis and structure–activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2008.05.010 ◽

2008 ◽

Vol 16 (12) ◽

pp. 6353-6363 ◽

Author(s):

Sara Cesarini ◽

Andrea Spallarossa ◽

Angelo Ranise ◽

Silvia Schenone ◽

Olga Bruno ◽

...

Keyword(s):

Reverse Transcriptase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Reverse Transcriptase Inhibitors ◽

One Pot ◽

One Pot Synthesis ◽

Structure Activity ◽

Relationship Study ◽

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A quantitative structure–Activity relationship study on some sulfolanes and arylthiomethanes acting as HIV-1 protease inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(98)00157-6 ◽

1998 ◽

Vol 6 (11) ◽

pp. 2185-2192 ◽

Author(s):

S.P. Gupta ◽

M.S. Babu ◽

S. Sowmya

Keyword(s):

Protease Inhibitors ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Study ◽

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Structure–activity relationship study of flavone compounds with anti-HIV-1 integrase activity: A density functional theory study

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2006.07.005 ◽

2006 ◽

Vol 14 (21) ◽

pp. 7105-7112 ◽

Author(s):

J. Lameira ◽

I.G. Medeiros ◽

M. Reis ◽

A.S. Santos ◽

C.N. Alves

Keyword(s):

Density Functional Theory ◽

Density Functional ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Density Functional Theory Study ◽

Functional Theory ◽

Structure Activity ◽

Relationship Study ◽

Anti Hiv ◽

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A quantitative structure–activity relationship study on some HIV-1 protease inhibitors using molecular connectivity index

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(01)00210-3 ◽

2001 ◽

Vol 9 (11) ◽

pp. 3059-3063 ◽

Author(s):

P. Gayathri ◽

V. Pande ◽

R. Sivakumar ◽

S.P. Gupta

Keyword(s):

Protease Inhibitors ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Molecular Connectivity ◽

Molecular Connectivity Index ◽

Structure Activity ◽

Relationship Study ◽

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Structure-activity relationship study of the plasma membrane translocating potential of a short peptide from HIV-1 Tat protein

Letters in Peptide Science ◽

10.1007/bf02442912 ◽

1997 ◽

Vol 4 (4-6) ◽

pp. 429-436 ◽

Author(s):

Eric Virès ◽

Claude Granier ◽

Paul Prevot ◽

Bernard Lebleu

Keyword(s):

Plasma Membrane ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Tat Protein ◽

Short Peptide ◽

Structure Activity ◽

Relationship Study ◽

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