AMPA Receptor Noncompetitive Inhibitors Occupy a Promiscuous Binding Site

2019 ◽  
Vol 10 (11) ◽  
pp. 4511-4521 ◽  
Author(s):  
Chamali Narangoda ◽  
Serzhan N. Sakipov ◽  
Maria G. Kurnikova
Keyword(s):  
Binding Site ◽  
Ampa Receptor ◽  
Noncompetitive Inhibitors

ChemInform Abstract: Substituted 1,2-Dihydrophthalazines: Potent, Selective, and Noncompetitive Inhibitors of the AMPA Receptor.

ChemInform ◽  
2010 ◽  
Vol 27 (19) ◽  
pp. no-no
Author(s):  
J. C. PELLETIER ◽  
D. P. HESSON ◽  
K. A. JONES ◽  
A.-M. COSTA
Keyword(s):  
Ampa Receptor ◽  
Noncompetitive Inhibitors

scholarly journals Molecular dissection of the agonist binding site of an AMPA receptor.

1995 ◽  
Vol 14 (24) ◽  
pp. 6327-6332 ◽  
Author(s):  
A. Kuusinen ◽  
M. Arvola ◽  
K. Keinänen
Keyword(s):  
Binding Site ◽  
Ampa Receptor ◽  
Molecular Dissection ◽  
Agonist Binding

Common Binding Site for Externally and Internally Applied AMPA Receptor Channel Blockers

2009 ◽  
Vol 39 (1-2) ◽  
pp. 169-174 ◽  
Author(s):  
Tatyana B. Tikhonova ◽  
Denis B. Tikhonov ◽  
Lev G. Magazanik
Keyword(s):  
Binding Site ◽  
Ampa Receptor ◽  
Channel Blockers ◽  
Receptor Channel

Identification of a putative binding site for 5-alkyl-benzothiadiazides in the AMPA receptor dimer interface

2007 ◽  
Vol 26 (1) ◽  
pp. 213-225 ◽  
Author(s):  
Kasper Harpsøe ◽  
Thomas Varming ◽  
Alex Haahr Gouliaev ◽  
Dan Peters ◽  
Tommy Liljefors
Keyword(s):  
Binding Site ◽  
Ampa Receptor ◽  
Dimer Interface ◽  
Receptor Dimer ◽  
Putative Binding Site

Substituted 1,2-Dihydrophthalazines:  Potent, Selective, and Noncompetitive Inhibitors of the AMPA Receptor

1996 ◽  
Vol 39 (2) ◽  
pp. 343-346 ◽  
Author(s):  
Jeffrey C. Pelletier ◽  
David P. Hesson ◽  
Kenneth A. Jones ◽  
Anna-Maria Costa
Keyword(s):  
Ampa Receptor ◽  
Noncompetitive Inhibitors

The binding site for allosteric modulators of AMPA receptor

2004 ◽  
Vol 399 (1-6) ◽  
pp. 351-353 ◽  
Author(s):  
I. G. Tikhonova ◽  
M. I. Lavrov ◽  
V. A. Palyulin ◽  
N. S. Zefirov
Keyword(s):  
Binding Site ◽  
Ampa Receptor ◽  
Allosteric Modulators

The AMPA Receptor Binding Site: Focus on Agonists and Competitive Antagonists

2002 ◽  
Vol 8 (10) ◽  
pp. 857-872 ◽  
Author(s):  
Tine Stensbol ◽  
Ulf Madsen ◽  
Povl Krogsgaard-Larsen
Keyword(s):  
Binding Site ◽  
Ampa Receptor ◽  
Receptor Binding ◽  
Receptor Binding Site

scholarly journals A Domain Linking the AMPA Receptor Agonist Binding Site to the Ion Pore Controls Gating and Causes lurcher Properties when Mutated

2007 ◽  
Vol 27 (45) ◽  
pp. 12230-12241 ◽  
Author(s):  
S. M. Schmid ◽  
C. Korber ◽  
S. Herrmann ◽  
M. Werner ◽  
M. Hollmann
Keyword(s):  
Binding Site ◽  
Ampa Receptor ◽  
Receptor Agonist ◽  
Agonist Binding ◽  
Ion Pore

Probing the opioid receptor complex with (+)-trans-SUPERFIT. II. Evidence that μ ligands are noncompetitive inhibitors of the δcx opioid peptide binding site

Peptides ◽  
1992 ◽  
Vol 13 (6) ◽  
pp. 1137-1143 ◽  
Author(s):  
Richard B. Rothman ◽  
Artin Mahboubi ◽  
Victor Bykov ◽  
Chong-Ho Kim ◽  
Brian R. de Costa ◽  
...  
Keyword(s):  
Binding Site ◽  
Opioid Receptor ◽  
Peptide Binding ◽  
Opioid Peptide ◽  
Receptor Complex ◽  
Peptide Binding Site ◽  
Noncompetitive Inhibitors

scholarly journals A Ligand-Binding Site in the Glua3 AMPA Receptor N-Terminal Domain Observed in Druggability Simulations and X-Ray Crystallography

2019 ◽  
Vol 116 (3) ◽  
pp. 489a
Author(s):  
Ji Young Lee ◽  
James Krieger ◽  
Beatriz Herguedas ◽  
Javier García-Nafría ◽  
Anindita Dutta ◽  
...  
Keyword(s):  
Ligand Binding ◽  
Binding Site ◽  
Ampa Receptor ◽  
Ligand Binding Site ◽  
X Ray ◽  
X Ray Crystallography ◽  
Terminal Domain
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