scholarly journals C&EN Webinars - In Silico Design, Synthesis, and Biological Testing of Novel Antimalarial Drug Candidates Generated by Analysis of Public HTS Data

2012 ◽  
Vol 90 (17) ◽  
pp. 37
Keyword(s):  
Antimalarial Drug ◽  
In Silico ◽  
Biological Testing ◽  
Design Synthesis ◽  
In Silico Design ◽  
Drug Candidates

scholarly journals Synthesis, characterization and biological activity of organometallic derivatives of the antimalarial drug mefloquine as new antischistosomal drug candidates

MedChemComm ◽  
2018 ◽  
Vol 9 (11) ◽  
pp. 1905-1909 ◽  
Author(s):  
Faustine d'Orchymont ◽  
Jeannine Hess ◽  
Gordana Panic ◽  
Marta Jakubaszek ◽  
Lea Gemperle ◽  
...  
Keyword(s):  
Biological Activity ◽  
Antimalarial Drug ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Drug Candidates ◽  
Derivatives Of

The design, synthesis, characterization and biological evaluation of new ferrocenyl and ruthenocenyl derivatives of the antimalarial mefloquine is described.

In silico design, synthesis, characterization and pharmacological evaluation of captopril conjugates in the treatment of renal fibrosis

2019 ◽  
Vol 43 (1) ◽  
pp. 504-513 ◽  
Author(s):  
Swapnil Dashrath Jadhav ◽  
Prafulla Balkrishna Choudhari ◽  
Manish Sudesh Bhatia
Keyword(s):  
Glutamic Acid ◽  
In Silico ◽  
Renal Fibrosis ◽  
Design Synthesis ◽  
In Silico Design ◽  
Pharmacological Evaluation ◽  
P Application

Application of glutamic acid and taurine conjugates of captopril for kidney targeting.

In silico design, synthesis and activity of potential drug-like chrysin scaffold-derived selective EGFR inhibitors as anticancer agents

2019 ◽  
Vol 83 ◽  
pp. 107156 ◽  
Author(s):  
Sudhan Debnath ◽  
Manupati Kanakaraju ◽  
Minarul Islam ◽  
Ragini Yeeravalli ◽  
Debanjan Sen ◽  
...  
Keyword(s):  
Anticancer Agents ◽  
In Silico ◽  
Egfr Inhibitors ◽  
Potential Drug ◽  
Design Synthesis ◽  
In Silico Design

In Silico Design, Synthesis, and Assays of Specific Substrates for Proteinase 3: Influence of Fluorogenic and Charged Groups

2014 ◽  
Vol 57 (3) ◽  
pp. 1111-1115 ◽  
Author(s):  
Shailesh Narawane ◽  
Adnan Budnjo ◽  
Cédric Grauffel ◽  
Bengt Erik Haug ◽  
Nathalie Reuter
Keyword(s):  
In Silico ◽  
Proteinase 3 ◽  
Design Synthesis ◽  
In Silico Design

In Silico Design, Synthesis and Bioactivity of N-(2, 4-Dinitrophenyl)-3-oxo- 3-phenyl-N-(aryl) Phenyl Propanamide Derivatives as Breast Cancer Inhibitors

2017 ◽  
Vol 13 (2) ◽  
pp. 112-126 ◽  
Author(s):  
Mucheli Ramana ◽  
Rama Lokhande ◽  
Shanta Bhar ◽  
Prasanna Ranade ◽  
Ankita Mehta ◽  
...  
Keyword(s):  
Breast Cancer ◽  
In Silico ◽  
Design Synthesis ◽  
In Silico Design
Sign in / Sign up

Export Citation Format

Share Document