Structure-Activity Relationships of the Antimalarial Agent Artemisinin. 2. Effect of Heteroatom Substitution at O-11: Synthesis and Bioassay of N-Alkyl-11-aza-9-desmethylartemisinins

1995 ◽  
Vol 38 (26) ◽  
pp. 5038-5044 ◽  
Author(s):  
Mitchell A. Avery ◽  
Jason D. Bonk ◽  
Wesley K. M. Chong ◽  
Sanjiv Mehrotra ◽  
Robert Miller ◽  
...  
Keyword(s):  
Antimalarial Agent ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Heteroatom Substitution ◽  
O 11

Structure−Activity Relationships of the Antimalarial Agent Artemisinin. 4. Effect of Substitution at C-3

1996 ◽  
Vol 39 (15) ◽  
pp. 2900-2906 ◽  
Author(s):  
Mitchell A. Avery ◽  
Sanjiv Mehrotra ◽  
Jason D. Bonk ◽  
Jeffrey A. Vroman ◽  
D. Keith Goins ◽  
...  
Keyword(s):  
Antimalarial Agent ◽  
Structure Activity Relationships ◽  
Structure Activity

Structure-Activity Relationships of Analogs of Thapsigargin Modified at O-11 and O-12

1995 ◽  
Vol 38 (2) ◽  
pp. 272-276 ◽  
Author(s):  
Simon Feldbk Nielsen ◽  
Ole Thastrup ◽  
Rudi Pedersen ◽  
Carl Erik Olsen ◽  
Soren Brogger Christensen
Keyword(s):  
Structure Activity Relationships ◽  
Structure Activity ◽  
O 11

Structure−Activity Relationships of the Antimalarial Agent Artemisinin. 3. Total Synthesis of (+)-13-Carbaartemisinin and Related Tetra- and Tricyclic Structures

1996 ◽  
Vol 39 (9) ◽  
pp. 1885-1897 ◽  
Author(s):  
Mitchell A. Avery ◽  
Pingchen Fan ◽  
Jean M. Karle ◽  
Jason D. Bonk ◽  
Robert Miller ◽  
...  
Keyword(s):  
Total Synthesis ◽  
Antimalarial Agent ◽  
Structure Activity Relationships ◽  
Structure Activity

Structure−Activity Relationships of the Antimalarial Agent Artemisinin. 6. The Development of Predictive In Vitro Potency Models Using CoMFA and HQSAR Methodologies

2002 ◽  
Vol 45 (2) ◽  
pp. 292-303 ◽  
Author(s):  
Mitchell A. Avery ◽  
Maria Alvim-Gaston ◽  
Carlos R. Rodrigues ◽  
Eliezer J. Barreiro ◽  
Fred E. Cohen ◽  
...  
Keyword(s):  
Antimalarial Agent ◽  
Structure Activity Relationships ◽  
Structure Activity

Structure−Activity Relationships of the Antimalarial Agent Artemisinin. 5. Analogs of 10-Deoxoartemisinin Substituted at C-3 and C-9

1996 ◽  
Vol 39 (21) ◽  
pp. 4149-4155 ◽  
Author(s):  
Mitchell A. Avery ◽  
Sanjiv Mehrotra ◽  
Theresa L. Johnson ◽  
Jason D. Bonk ◽  
Jeffrey A. Vroman ◽  
...  
Keyword(s):  
Antimalarial Agent ◽  
Structure Activity Relationships ◽  
Structure Activity
Sign in / Sign up

Export Citation Format

Share Document