Synthesis and thromboxane A2/prostaglandin H2 receptor antagonistic activity of phenol derivatives

Journal of Medicinal Chemistry ◽

10.1021/jm00090a009 ◽

1992 ◽

Vol 35 (12) ◽

pp. 2202-2209 ◽

Author(s):

Shoji Fukumoto ◽

Mitsuru Shiraishi ◽

Zenichi Terashita ◽

Yasuko Ashida ◽

Yoshiyuki Inada

Keyword(s):

Thromboxane A2 ◽

Antagonistic Activity ◽

H2 Receptor ◽

Phenol Derivatives

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ChemInform Abstract: Stereoselective Synthesis and Thromboxane A2 (TXA2) Receptor Antagonistic Activity of Optically Active Phenol Derivatives.

10.1002/chin.199643225 ◽

2010 ◽

Vol 27 (43) ◽

pp. no-no

Author(s):

S. FUKUMOTO ◽

Z. TERASHITA ◽

Y. ASHIDA ◽

S. TERAO ◽

M. SHIRAISHI

Keyword(s):

Stereoselective Synthesis ◽

Thromboxane A2 ◽

Antagonistic Activity ◽

Optically Active ◽

Phenol Derivatives ◽

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Stereoselective Synthesis and Thromboxane A2 (TXA2) Receptor Antagonistic Activity of Optically Active Phenol Derivatives.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.44.749 ◽

1996 ◽

Vol 44 (4) ◽

pp. 749-755 ◽

Author(s):

Shoji FUKUMOTO ◽

Zen-ichi TERASHITA ◽

Yasuko ASHIDA ◽

Shinji TERAO ◽

Mitsuru SHIRAISHI

Keyword(s):

Stereoselective Synthesis ◽

Thromboxane A2 ◽

Antagonistic Activity ◽

Optically Active ◽

Phenol Derivatives ◽

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A common binding site for primary prostanoids in vascular smooth muscles: a definitive discrimination of the binding for thromboxane A2/prostaglandin H2 receptor agonist from its antagonist

Biochimica et Biophysica Acta (BBA) - Molecular Cell Research ◽

10.1016/0167-4889(89)90123-7 ◽

1989 ◽

Vol 1013 (1) ◽

pp. 28-35 ◽

Author(s):

Kohji Hanasaki ◽

Hitoshi Arita

Keyword(s):

Binding Site ◽

Receptor Agonist ◽

Smooth Muscles ◽

Thromboxane A2 ◽

Vascular Smooth Muscles ◽

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ChemInform Abstract: X-Ray Crystal Structure of a Ligand at the Thromboxane A2/Prostaglandin H2 Receptor Site: (4Z)-6-((2RS,4RS,5SR)-2-(2-Chlorophenyl)-4-(2-hydroxyphenyl)-1,3-dioxan-5-yl)hex-4-enoic Acid

10.1002/chin.199043289 ◽

1990 ◽

Vol 21 (43) ◽

Author(s):

G. R. BROWN ◽

A. J. FOUBISTER ◽

M. MCPARTLIN

Keyword(s):

Crystal Structure ◽

Thromboxane A2 ◽

Receptor Site ◽

H2 Receptor ◽

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X-Ray crystal structure of a ligand at the thromboxane A2/prostaglandin H2 receptor site: (4Z)-6-[(2RS,4RS,5SR)-2-(2-chlorophenyl)-4-(2-hydroxyphenyl)-1,3-dioxan-5-yl]hex-4-enoic acid

Journal of the Chemical Society Perkin Transactions 1 ◽

10.1039/p19900002158 ◽

1990 ◽

pp. 2158 ◽

Author(s):

George R. Brown ◽

Alan J. Foubister ◽

Mary McPartlin

Keyword(s):

Crystal Structure ◽

Thromboxane A2 ◽

Receptor Site ◽

H2 Receptor ◽

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Synthesis and Optical Resolution of an Antiallergic Agent KW4099 with Thromboxane A2 Antagonistic Activity.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.40.238 ◽

1992 ◽

Vol 40 (1) ◽

pp. 238-239 ◽

Author(s):

Toru SUGAYA ◽

Yukihiro KUGE ◽

Shinji TOMIOKA ◽

Kentaro TAMAKI

Keyword(s):

Optical Resolution ◽

Thromboxane A2 ◽

Antagonistic Activity ◽

Antiallergic Agent

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Synthesis of an [125I]-azido photoaffinity probe for the human platelet thromboxane A2/prostaglandin H2 receptor

Journal of Labelled Compounds and Radiopharmaceuticals ◽

10.1002/jlcr.2580250706 ◽

1988 ◽

Vol 25 (7) ◽

pp. 731-737 ◽

Author(s):

Dale E. Mais ◽

Perry V. Halushka

Keyword(s):

Human Platelet ◽

Thromboxane A2 ◽

H2 Receptor ◽

Platelet Thromboxane

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Synthesis and Thromboxane A2 Antagonistic Activity of ((1-Aryl(or Benzyl)-1-(benzenesulfonamido)methyl)phenyl)alkanoic Acid Derivatives.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.44.765 ◽

1996 ◽

Vol 44 (4) ◽

pp. 765-777 ◽

Author(s):

Shuniciro SAKURAI ◽

Nobuo OGAWA ◽

Tomio SUZUKI ◽

Ken-ichi KATO ◽

Tetsuo OHASHI ◽

...

Keyword(s):

Thromboxane A2 ◽

Antagonistic Activity ◽

Alkanoic Acid ◽

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Purification of the human blood platelet thromboxane A2/prostaglandin H2 receptor protein

Biochemical Pharmacology ◽

10.1016/0006-2952(92)90294-s ◽

1992 ◽

Vol 43 (2) ◽

pp. 313-322 ◽

Author(s):

Kim Sun-Ok ◽

Lim Chang T. ◽

Stephen C-T. Lam ◽

Steven E. Hall ◽

Dimitri Komiotis ◽

...

Keyword(s):

Human Blood ◽

Thromboxane A2 ◽

Blood Platelet ◽

Receptor Protein ◽

H2 Receptor ◽

Human Blood Platelet ◽

Platelet Thromboxane

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Gastroprotective Mechanism of Lafutidine, a Novel Anti-ulcer Drug with Histamine H2-Receptor Antagonistic Activity

Arzneimittelforschung ◽

10.1055/s-0031-1300454 ◽

2011 ◽

Vol 49 (06) ◽

pp. 519-526

Author(s):

Sadayoshi Onodera ◽

Masahiro Shibata ◽

Masato Tanaka ◽

Niro Inaba ◽

Yoko Arai ◽

...

Keyword(s):

Antagonistic Activity ◽

Histamine H2 Receptor ◽

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