Selective Estrogen Receptor Modulators with Conformationally Restricted Side Chains. Synthesis and Structure−Activity Relationship of ERα-Selective Tetrahydroisoquinoline Ligands

2005 ◽  
Vol 48 (2) ◽  
pp. 364-379 ◽  
Author(s):  
Johanne Renaud ◽  
Serge François Bischoff ◽  
Thomas Buhl ◽  
Philipp Floersheim ◽  
Brigitte Fournier ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Side Chains ◽  
Conformationally Restricted ◽  
Estrogen Receptor Modulators ◽  
Structure Activity ◽  
Relationship Of ◽  
Receptor Modulators

scholarly journals The Structure–Activity Relationship of a Tetrahydroisoquinoline Class ofN-Methyl-d-Aspartate Receptor Modulators that Potentiates GluN2B-ContainingN-Methyl-d-Aspartate Receptors

2017 ◽  
Vol 60 (13) ◽  
pp. 5556-5585 ◽  
Author(s):  
Katie L. Strong ◽  
Matthew P. Epplin ◽  
John Bacsa ◽  
Christopher J. Butch ◽  
Pieter B. Burger ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Aspartate Receptor ◽  
Structure Activity ◽  
Relationship Of ◽  
Receptor Modulators

Structure–Activity Relationships for a Family of Benzothiophene Selective Estrogen Receptor Modulators Including Raloxifene and Arzoxifene

ChemMedChem ◽  
2007 ◽  
Vol 2 (10) ◽  
pp. 1520-1526 ◽  
Author(s):  
Cassia R. Overk ◽  
Kuan-Wei Peng ◽  
Rezene T. Asghodom ◽  
Irida Kastrati ◽  
Daniel D. Lantvit ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Structure Activity Relationships ◽  
Estrogen Receptor Modulators ◽  
Structure Activity ◽  
Receptor Modulators

scholarly journals Structure–Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists

2021 ◽  
Author(s):  
David Sedlák ◽  
Tyler A. Wilson ◽  
Werner Tjarks ◽  
Hanna S. Radomska ◽  
Hongyan Wang ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Structure Activity Relationship ◽  
Estrogen Receptor Β ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

4-(4-Alkylpiperazin-1-yl)phenyl group: A novel class of basic side chains for selective estrogen receptor modulators

2003 ◽  
Vol 13 (24) ◽  
pp. 4317-4320 ◽  
Author(s):  
Nobuhide Watanabe ◽  
Hiroshi Nakagawa ◽  
Akihisa Ikeno ◽  
Hisao Minato ◽  
Chie Kohayakawa ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Phenyl Group ◽  
Selective Estrogen Receptor Modulators ◽  
Side Chains ◽  
Estrogen Receptor Modulators ◽  
Group A ◽  
Receptor Modulators

Structure−Activity Relationships of Selective Estrogen Receptor Modulators:  Modifications to the 2-Arylbenzothiophene Core of Raloxifene

1997 ◽  
Vol 40 (2) ◽  
pp. 146-167 ◽  
Author(s):  
Timothy A. Grese ◽  
Stephen Cho ◽  
Don R. Finley ◽  
Alexander G. Godfrey ◽  
Charles D. Jones ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Structure Activity Relationships ◽  
Estrogen Receptor Modulators ◽  
Structure Activity ◽  
Receptor Modulators

Synthesis and structure–activity relationship of 3-arylbenzoxazines as selective estrogen receptor β agonists

2004 ◽  
Vol 14 (9) ◽  
pp. 2327-2330 ◽  
Author(s):  
Wu Yang ◽  
Yufeng Wang ◽  
Zhengping Ma ◽  
Rajasree Golla ◽  
Terry Stouch ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Structure Activity Relationship ◽  
Estrogen Receptor Β ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of
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