Selective Estrogen Receptor Modulators with Conformationally Restricted Side Chains. Synthesis and Structure−Activity Relationship of ERα-Selective Tetrahydroisoquinoline Ligands

2005 ◽  
Vol 48 (2) ◽  
pp. 364-379 ◽  
Author(s):  
Johanne Renaud ◽  
Serge François Bischoff ◽  
Thomas Buhl ◽  
Philipp Floersheim ◽  
Brigitte Fournier ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Side Chains ◽  
Conformationally Restricted ◽  
Estrogen Receptor Modulators ◽  
Structure Activity ◽  
Relationship Of ◽  
Receptor Modulators

Structure–Activity Relationships for a Family of Benzothiophene Selective Estrogen Receptor Modulators Including Raloxifene and Arzoxifene

ChemMedChem ◽  
2007 ◽  
Vol 2 (10) ◽  
pp. 1520-1526 ◽  
Author(s):  
Cassia R. Overk ◽  
Kuan-Wei Peng ◽  
Rezene T. Asghodom ◽  
Irida Kastrati ◽  
Daniel D. Lantvit ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Structure Activity Relationships ◽  
Estrogen Receptor Modulators ◽  
Structure Activity ◽  
Receptor Modulators

4-(4-Alkylpiperazin-1-yl)phenyl group: A novel class of basic side chains for selective estrogen receptor modulators

2003 ◽  
Vol 13 (24) ◽  
pp. 4317-4320 ◽  
Author(s):  
Nobuhide Watanabe ◽  
Hiroshi Nakagawa ◽  
Akihisa Ikeno ◽  
Hisao Minato ◽  
Chie Kohayakawa ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Phenyl Group ◽  
Selective Estrogen Receptor Modulators ◽  
Side Chains ◽  
Estrogen Receptor Modulators ◽  
Group A ◽  
Receptor Modulators
Sign in / Sign up

Export Citation Format

Share Document