New Non-Peptide Endothelin-A Receptor Antagonists:  Synthesis, Biological Properties, and Structure−Activity Relationships of 5-(Dimethylamino)-N-pyridyl-, -N-pyrimidinyl-, -N-pyridazinyl-, and -N-pyrazinyl-1-naphthalenesulfonamides

1997 ◽  
Vol 40 (6) ◽  
pp. 996-1004 ◽  
Author(s):  
Robert H. Bradbury ◽  
Colin Bath ◽  
Roger J. Butlin ◽  
Michael Dennis ◽  
Christine Heys ◽  
...  
Keyword(s):  
Biological Properties ◽  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

Selective endothelin A receptor antagonists. 2. Discovery and structure-activity relationships of 5-ketopentanoic acid derivatives

1997 ◽  
Vol 32 (6) ◽  
pp. 515-522 ◽  
Author(s):  
P.C. Astles ◽  
T.J. Brown ◽  
N.V. Harris ◽  
M.F. Harper ◽  
C McCarthy ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

Synthesis and structure-activity relationships of 9-substituted acridines as endothelin-A receptor antagonists

1996 ◽  
Vol 6 (24) ◽  
pp. 2999-3002 ◽  
Author(s):  
X.-M. Cheng ◽  
C. Lee ◽  
S. Klutchko ◽  
T. Winters ◽  
E.E. Reynolds ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

Selective Endothelin A Receptor Antagonists. 4. Discovery and Structure−Activity Relationships of Stilbene Acid and Alcohol Derivatives1-3

1998 ◽  
Vol 41 (15) ◽  
pp. 2745-2753 ◽  
Author(s):  
Peter C. Astles ◽  
Thomas J. Brown ◽  
Frank Halley ◽  
Caroline M. Handscombe ◽  
Neil V. Harris ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

ChemInform Abstract: Synthesis and Structure-Activity Relationships of 9-Substituted Acridines as Endothelin-A Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 28 (23) ◽  
pp. no-no
Author(s):  
X.-M. CHENG ◽  
C. LEE ◽  
S. KLUTCHKO ◽  
T. WINTERS ◽  
E. E. REYNOLDS ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

Selective Endothelin A Receptor Antagonists. 3. Discovery and Structure−Activity Relationships of a Series of 4-Phenoxybutanoic Acid Derivatives

1998 ◽  
Vol 41 (15) ◽  
pp. 2732-2744 ◽  
Author(s):  
Peter C. Astles ◽  
Clive Brealey ◽  
Thomas J. Brown ◽  
Vincenzo Facchini ◽  
Caroline Handscombe ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

ChemInform Abstract: Selective Endothelin A Receptor Antagonists. Part 2. Discovery and Structure-Activity Relationships of 5-Ketopentanoic Acid Derivatives.

ChemInform ◽  
2010 ◽  
Vol 28 (43) ◽  
pp. no-no
Author(s):  
P. C. ASTLES ◽  
T. J. BROWN ◽  
N. V. HARRIS ◽  
M. F. HARPER ◽  
C. MCCARTHY ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

Structure-Activity Relationships of Cyclic Pentapeptide Endothelin A Receptor Antagonists

1995 ◽  
Vol 38 (21) ◽  
pp. 4309-4324 ◽  
Author(s):  
Takehiro Fukami ◽  
Toshio Nagase ◽  
Kagari Fujita ◽  
Takashi Hayama ◽  
Kenji Niiyama ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A
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