Synthesis of the (3R,6S)-3-Amino-6-(2,3-difluorophenyl)azepan-2-one of Telcagepant (MK-0974), a Calcitonin Gene-Related Peptide Receptor Antagonist for the Treatment of Migraine Headache

2008 ◽  
Vol 10 (15) ◽  
pp. 3235-3238 ◽  
Author(s):  
Christopher S. Burgey ◽  
Daniel V. Paone ◽  
Anthony W. Shaw ◽  
James Z. Deng ◽  
Diem N. Nguyen ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Migraine Headache ◽  
Calcitonin Gene Related Peptide ◽  
Peptide Receptor ◽  
Related Peptide ◽  
Calcitonin Gene

Pharmacological Properties of MK-3207, a Potent and Orally Active Calcitonin Gene-Related Peptide Receptor Antagonist

2010 ◽  
Vol 333 (1) ◽  
pp. 152-160 ◽  
Author(s):  
Christopher A. Salvatore ◽  
Eric L. Moore ◽  
Amy Calamari ◽  
Jacquelynn J. Cook ◽  
Maria S. Michener ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Calcitonin Gene Related Peptide ◽  
Pharmacological Properties ◽  
Peptide Receptor ◽  
Related Peptide ◽  
Calcitonin Gene ◽  
Orally Active
Sign in / Sign up

Export Citation Format

Share Document