scholarly journals Development of novel fluorescent histamine H1-receptor antagonists to study ligand-binding kinetics in living cells

2018 ◽  
Vol 8 (1) ◽  
Author(s):  
Leigh A. Stoddart ◽  
Andrea J. Vernall ◽  
Monica Bouzo-Lorenzo ◽  
Reggie Bosma ◽  
Albert J. Kooistra ◽  
...  
Keyword(s):  
Ligand Binding ◽  
Living Cells ◽  
Binding Kinetics ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor

scholarly journals Exploring the Effect of Cyclization of Histamine H1 Receptor Antagonists on Ligand Binding Kinetics

ACS Omega ◽  
2021 ◽  
Author(s):  
Zhiyong Wang ◽  
Reggie Bosma ◽  
Sebastiaan Kuhne ◽  
Jelle van den Bor ◽  
Wrej Garabitian ◽  
...  
Keyword(s):  
Ligand Binding ◽  
Binding Kinetics ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor

scholarly journals Design of Phthalazinone Amide Histamine H1 Receptor Antagonists for Use in Rhinitis

2017 ◽  
Vol 8 (5) ◽  
pp. 577-581 ◽  
Author(s):  
Panayiotis A. Procopiou ◽  
Alison J. Ford ◽  
Paul M. Gore ◽  
Brian E. Looker ◽  
Simon T. Hodgson ◽  
...  
Keyword(s):  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor

Anti-Inflammatory Actions of Histamine H1 Receptor Antagonists Unrelated to H1 Receptor Blockade

1996 ◽  
Vol 5 (6) ◽  
pp. 449-464 ◽  
Author(s):  
Claus Kroegel ◽  
Verena Herzog ◽  
Birgit Knöchel ◽  
Peter Julius ◽  
Dirk Wagnetz ◽  
...  
Keyword(s):  
Receptor Blockade ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor ◽  
Anti Inflammatory

Identification of selective 8-(piperidin-4-yloxy)quinoline sulfone and sulfonamide histamine H1 receptor antagonists for use in allergic rhinitis

2017 ◽  
Vol 27 (21) ◽  
pp. 4914-4919 ◽  
Author(s):  
Panayiotis A. Procopiou ◽  
Alison J. Ford ◽  
Paul M. Gore ◽  
Ashley P. Hancock ◽  
Simon T. Hodgson ◽  
...  
Keyword(s):  
Allergic Rhinitis ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor
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